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المؤلفون: Yaqin Jia, Yangliu Xia, Yuyi Feng, Zhen Wang, Lili Jiang, Jun Cao, Yong Liu, Zhe Wang, Xiaoyu Wang
المصدر: Toxicology Letters. 348:10-17
مصطلحات موضوعية: Male, 0301 basic medicine, Drug, media_common.quotation_subject, Glucuronidation, Pharmacology, Toxicology, digestive system, 03 medical and health sciences, 0302 clinical medicine, Non-competitive inhibition, In vivo, Humans, Drug Interactions, Osimertinib, Epidermal growth factor receptor, Glucuronosyltransferase, media_common, Acrylamides, Aniline Compounds, biology, Chemistry, General Medicine, In vitro, 030104 developmental biology, Microsomes, Liver, biology.protein, Microsome, 030217 neurology & neurosurgery
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المؤلفون: Emily J. Hanan, Hank La, Ivana Yen, Xiao-Hui Gu, Stephen Schmidt, Christine Yu, Timothy P. Heffron, Yuan Chen, Marian C. Bryan, Gabriele Schaefer, Peter W. Fan, Matt Baumgardner, Shiva Malek, Charles Eigenbrot, Steve Sideris, Hans E. Purkey
المصدر: Bioorganicmedicinal chemistry letters. 26(2)
مصطلحات موضوعية: 0301 basic medicine, Indazoles, Clinical Biochemistry, Mutant, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, 03 medical and health sciences, T790M, Erlotinib Hydrochloride, Mice, 0302 clinical medicine, Dogs, Growth factor receptor, Drug Discovery, Animals, Humans, Point Mutation, Growth factor receptor inhibitor, ERBB3, Epidermal growth factor receptor, Furans, Molecular Biology, Protein Kinase Inhibitors, EGFR inhibitors, Acrylamides, Aniline Compounds, Binding Sites, biology, Chemistry, Organic Chemistry, Hydrogen Bonding, Molecular biology, respiratory tract diseases, High-Throughput Screening Assays, Rats, ErbB Receptors, 030104 developmental biology, Pyrimidines, 030220 oncology & carcinogenesis, biology.protein, Hepatocytes, Microsomes, Liver, Molecular Medicine
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المؤلفون: Helena Rýdlová, Markéta Mikšanová, Eva Frei, Heinz H. Schmeiser, Miroslav Šulc, Marie Stiborová
المصدر: International Journal of Cancer. 116:667-678
مصطلحات موضوعية: Male, Cancer Research, Metabolite, o-Anisidine, medicine.disease_cause, law.invention, DNA Adducts, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, law, medicine, Animals, Deoxyguanosine, Rats, Wistar, Biotransformation, Carcinogen, Aniline Compounds, biology, Cytochrome P450, Carcinogens, Environmental, Rats, Oncology, chemistry, Biochemistry, Microsomes, Liver, biology.protein, Microsome, Recombinant DNA, Environmental Pollutants, Oxidation-Reduction, Genotoxicity
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المؤلفون: E. Karge, U. Demme, Wolfgang Klinger, M Kretzschmar
المصدر: European Journal of Drug Metabolism and Pharmacokinetics. 26:31-35
مصطلحات موضوعية: medicine.medical_specialty, Hexobarbital, In Vitro Techniques, Antioxidants, Melatonin, Lipid peroxidation, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Internal medicine, medicine, Animals, Humans, Hypnotics and Sedatives, Pharmacology (medical), Rats, Wistar, Pharmacology, Oxidase test, Aniline Compounds, biology, Chemistry, Cytochrome P450, Glutathione, Monooxygenase, Ethylmorphine, Rats, Endocrinology, Liver, Microsomes, Liver, biology.protein, Lipid Peroxidation, Sleep, NADP, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fd6fc86525038c61d6c779e73f0e4e0a
https://doi.org/10.1007/bf03190373 -
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المؤلفون: Hiroyuki Yasui, Hiromu Sakurai, Yuhko Ogura, Mayuko Osada
المصدر: Biochemical and Biophysical Research Communications. 263:392-397
مصطلحات موضوعية: Male, Aniline Compounds, Biophysics, 7-Alkoxycoumarin O-Dealkylase, Photochemistry, Biochemistry, Rats, Sprague-Dawley, Hydroxylation, Superoxide dismutase, chemistry.chemical_compound, Aniline, Cytochrome P-450 Enzyme System, Coumarins, Animals, Sodium Azide, Molecular Biology, Piperidones, Singlet Oxygen, biology, Spin trapping, Singlet oxygen, Electron Spin Resonance Spectroscopy, Free Radical Scavengers, Triacetoneamine-N-Oxyl, Cell Biology, beta Carotene, Rats, Oxygen, chemistry, Microsomes, Liver, biology.protein, Microsome, Sodium azide, Oxidation-Reduction, Spin Trapping, NADP
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المؤلفون: Yiqun Zhang, Steven J. Pernecky
المصدر: Biochemical and Biophysical Research Communications. 258:32-38
مصطلحات موضوعية: Cumene, Stereochemistry, Biophysics, Hydroxylation, Methylation, Biochemistry, Catalysis, Substrate Specificity, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Benzene Derivatives, medicine, Animals, Organic chemistry, Molecular Biology, Sequence Deletion, Demethylation, chemistry.chemical_classification, Aniline Compounds, biology, Cytochrome P450, Substrate (chemistry), Cell Biology, Amino acid, chemistry, Cumene hydroperoxide, Steroid Hydroxylases, Microsomes, Liver, Phosphatidylcholines, Microsome, biology.protein, Aryl Hydrocarbon Hydroxylases, Rabbits, Benzphetamine, medicine.drug
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المصدر: Biochimica et Biophysica Acta (BBA) - General Subjects. 1379:391-398
مصطلحات موضوعية: Cytochrome, Stereochemistry, Biophysics, Substituent, 4-Nitroaniline, Biochemistry, Enzyme activator, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Animals, RNA, Messenger, Enzyme inducer, Molecular Biology, chemistry.chemical_classification, Aniline Compounds, biology, CYP1A2, Nitro Compounds, Rats, Inbred F344, Rats, Enzyme Activation, Enzyme, chemistry, Enzyme Induction, Microsomes, Liver, biology.protein, Nitro
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المصدر: Biochemical and Biophysical Research Communications. 244:347-352
مصطلحات موضوعية: Male, Macromolecular Substances, Protein Conformation, Immunoblotting, Sterol O-acyltransferase, Biophysics, Biochemistry, Cyclohexanes, Microsomes, Immunoblot Analysis, Liver enzyme, Adrenal Glands, Animals, Humans, Anilides, Tissue Distribution, Enzyme Inhibitors, Rats, Wistar, Molecular Biology, Aniline Compounds, biology, Phenylurea Compounds, Cell Biology, Rats, Acyl coenzyme A, Molecular Weight, Cross-Linking Reagents, Rat liver, Microsomes, Liver, biology.protein, Microsome, Antibody, Sterol O-Acyltransferase
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المؤلفون: Badger Da, I. G. Sipes, J M Sauer, R. K. Kuester
المصدر: Toxicology. 121:143-153
مصطلحات موضوعية: Male, Kupffer Cells, Beryllium sulfate, Anti-Inflammatory Agents, Aniline Hydroxylase, Gadolinium, Cell Separation, Pharmacology, Cadmium chloride, Hydroxylation, Toxicology, Rats, Sprague-Dawley, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, medicine, Animals, Carbon Tetrachloride, Biotransformation, Cells, Cultured, Analysis of Variance, Aniline Compounds, biology, Kupffer cell, Cytochrome P450, Rats, medicine.anatomical_structure, Liver, chemistry, Biochemistry, Hepatocyte, Injections, Intravenous, Toxicity, Carcinogens, Microsomes, Liver, biology.protein, Microsome, Female
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المؤلفون: Shigeru Ohmori, Kiyoshi Inoue, Sei-ichi Nakamura, Hajime Oda, Tsutomu Shimada, M Mimura, Hiroshi Yamazaki
المصدر: Archives of Toxicology. 71:401-408
مصطلحات موضوعية: Nifedipine, Health, Toxicology and Mutagenesis, Adrenergic beta-Antagonists, Guinea Pigs, Antineoplastic Agents, Pharmacology, Toxicology, chemistry.chemical_compound, Dogs, Cytochrome P-450 Enzyme System, Species Specificity, Coumarins, Oxazines, medicine, Animals, Ethylmorphine, Humans, Mephenytoin, Aniline Compounds, biology, Bufuralol, CYP1A2, Benzphetamine, Phenacetin, Cytochrome P450, General Medicine, Erythromycin, Rats, Macaca fascicularis, chemistry, Ethanolamines, Phenytoin, Carcinogens, Microsomes, Liver, biology.protein, Microsome, Oxidation-Reduction, Drug metabolism, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59acc9014f866424f8d36da545942a22
https://doi.org/10.1007/s002040050403