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1
المؤلفون: Laura Scarone, Gloria Serra, Eduardo Manta, Stella Peña, Lindsay B. Stewart, Vanessa Yardley, Simon L. Croft
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:4994-4997
مصطلحات موضوعية: Cyanobacteria, Microcystis, Stereochemistry, Metabolite, Plasmodium falciparum, Clinical Biochemistry, Pharmaceutical Science, Peptides, Cyclic, Biochemistry, Chemical synthesis, Antimalarials, chemistry.chemical_compound, Drug Discovery, Microcystis aeruginosa, Thiazole, Oxazoles, Molecular Biology, biology, Organic Chemistry, Drug Resistance, Microbial, Biological activity, biology.organism_classification, In vitro, Thiazoles, chemistry, Molecular Medicine, Bacteria
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2
المؤلفون: Peter W. Seale, Peter John Murray, Andrew B. Holmes, Mark Ladlow, Frédéric Berst, Simon L. Croft, Richard J. Upton, Paul Stead, Albert Andrzej Glaxo Wellcome plc Jaxa-Chamiec, William Clegg, Michael Kranz, Kenneth Keavey, Stephen Taylor, Mark R. J. Elsegood
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:773-776
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Trypanosoma brucei brucei, Clinical Biochemistry, Pharmaceutical Science, Trypanosoma brucei, Peptides, Cyclic, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Antiprotozoal Agent, Parasitic Sensitivity Tests, parasitic diseases, Drug Discovery, medicine, Animals, Molecular Biology, chemistry.chemical_classification, Natural product, biology, Chemistry, Organic Chemistry, Biological activity, biology.organism_classification, Trypanocidal Agents, Cyclic peptide, Antiprotozoal, Molecular Medicine, Apicidin
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3
المؤلفون: Junko Ohkanda, Simon L. Croft, Said M. Sebti, Kohei Yokoyama, Maria Isabel Harrell, Jeffrey W. Lockman, Andrew D. Hamilton, Michelle A. Blaskovich, Jean E. Feagin, Howard Kendrick, Michael H. Gelb
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:761-764
مصطلحات موضوعية: Peptidomimetic, Farnesyltransferase, Plasmodium falciparum, Clinical Biochemistry, Drug Resistance, Pharmaceutical Science, Pharmacology, Biochemistry, Antimalarials, Inhibitory Concentration 50, Structure-Activity Relationship, Parasitic Sensitivity Tests, parasitic diseases, Drug Discovery, medicine, Animals, Antimalarial Agent, Enzyme Inhibitors, Molecular Biology, Farnesyl-diphosphate farnesyltransferase, Alkyl and Aryl Transferases, biology, Chemistry, Organic Chemistry, Imidazoles, biology.organism_classification, medicine.disease, In vitro, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Malaria
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4
المؤلفون: Alan H. Fairlamb, Simon L. Croft, Vanessa Yardley, Mark Visser, Kelly Chibale
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:1147-1150
مصطلحات موضوعية: Tertiary amine, Antiparasitic, medicine.drug_class, Trypanosoma cruzi, Trypanosoma brucei brucei, Clinical Biochemistry, Antiprotozoal Agents, Leishmania donovani, Pharmaceutical Science, Trypanosoma brucei, Biochemistry, parasitic diseases, Drug Discovery, medicine, Animals, NADH, NADPH Oxidoreductases, Enzyme Inhibitors, Molecular Biology, biology, Chemistry, Organic Chemistry, Kinetoplastida, Biological activity, Leishmania, biology.organism_classification, Xanthenes, Molecular Medicine
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5
المؤلفون: K. Shirisha, Subhash Padhye, Nikhil H. Gokhale, Howard Kendrick, Simon L. Croft, Vickie McKee
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:430-432
مصطلحات موضوعية: Models, Molecular, Molecular model, Stereochemistry, Plasmodium falciparum, Clinical Biochemistry, Pharmaceutical Science, chemistry.chemical_element, Crystal structure, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Redox, Antimalarials, chemistry.chemical_compound, Parasitic Sensitivity Tests, parasitic diseases, Drug Discovery, Organometallic Compounds, Animals, Molecular Biology, Molecular Structure, Bicyclic molecule, Chemistry, Organic Chemistry, Copper, Quinone, Molecular Medicine, Crystallization, Hydroxynaphthoquinone, Naphthoquinones
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6
المؤلفون: Canio J. Marasco, Diane Snowdon, Simon L. Croft, Arthur J. Spiess, Cyrus J. Bacchi, Vanessa Yardley, Janice R. Sufrin
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:1961-1964
مصطلحات موضوعية: Purine, Antiparasitic, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Periodate, Biochemistry, Redox, Solvent, chemistry.chemical_compound, chemistry, Drug Discovery, medicine, Molecular Medicine, Organic chemistry, Methanol, Molecular Biology