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11
المؤلفون: Vincent P. Alibu, Sylvie Daunes, Claudius D'Silva
المصدر: Bioorganicmedicinal chemistry letters. 23(15)
مصطلحات موضوعية: Clinical Biochemistry, Trypanosoma brucei brucei, Protozoan Proteins, Pharmaceutical Science, Quantitative Structure-Activity Relationship, Drug resistance, Trypanosoma brucei, Biochemistry, chemistry.chemical_compound, parasitic diseases, Drug Discovery, Molecular Biology, biology, Organic Chemistry, Wild type, Membrane Transport Proteins, Transporter, Glutathione, biology.organism_classification, In vitro, Multiple drug resistance, chemistry, Molecular Medicine, Dinitrophenyl, Protein Binding
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12
المصدر: Bioorganic & Medicinal Chemistry Letters; Vol 23
مصطلحات موضوعية: Trypanosoma brucei rhodesiense, medicine.drug_class, Cell Survival, Trypanosoma cruzi, Clinical Biochemistry, Trypanosoma brucei brucei, Antiprotozoal Agents, Pharmaceutical Science, Trypanosoma brucei, 010402 general chemistry, 01 natural sciences, Biochemistry, Cell Line, Structure-Activity Relationship, Parasitic Sensitivity Tests, Amphotericin B, parasitic diseases, Drug Discovery, medicine, Humans, Leishmania infantum, Nifurtimox, Molecular Biology, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, biology.organism_classification, 0104 chemical sciences, 3. Good health, Benznidazole, Nitroimidazoles, Antiprotozoal, Trypanosoma, Quinolines, Molecular Medicine, medicine.drug
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13
المؤلفون: Alden E. Gustafson, Robert K. Campbell, Stefan O. Ochiana, Nicholas D. Bland, Trent D. Ashton, Cuihua Wang, Michael P. Pollastri
المصدر: Bioorganicmedicinal chemistry letters. 22(7)
مصطلحات موضوعية: Sildenafil, Clinical Biochemistry, Trypanosoma brucei brucei, Protozoan Proteins, Pharmaceutical Science, Pharmacology, Trypanosoma brucei, Biochemistry, Article, Tadalafil, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, parasitic diseases, medicine, Structure–activity relationship, Animals, Humans, Molecular Biology, Trypanocidal agent, chemistry.chemical_classification, biology, Phosphoric Diester Hydrolases, Organic Chemistry, Phosphodiesterase, Phosphodiesterase 5 Inhibitors, biology.organism_classification, Trypanocidal Agents, Solutions, Enzyme, chemistry, Drug development, Molecular Medicine, Biological Assay, medicine.drug, Carbolines
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14
المؤلفون: Roberto R. Gil, Shanshan He, Raymond W. Doskotch, Clemens Anklin, Xiaohua Zhu, Trupti Pandharkar, Mark E. Drew, Karl A. Werbovetz, A. Douglas Kinghorn, Armando Navarro-Vázquez, Ye Deng, Mark Bahar
المصدر: Bioorganicmedicinal chemistry letters. 21(9)
مصطلحات موضوعية: Models, Molecular, Berberine, medicine.drug_class, Clinical Biochemistry, Plasmodium falciparum, Trypanosoma brucei brucei, Antiprotozoal Agents, Pharmaceutical Science, Pharmacology, Biochemistry, Antiprotozoal Agent, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, In vivo, Trypanosomiasis, Drug Discovery, Chlorocebus aethiops, medicine, Animals, Parasites, Molecular Biology, Leishmaniasis, Vero Cells, Leishmania, Protozoan Infections, biology, Chemistry, Alkaloid, Organic Chemistry, medicine.disease, biology.organism_classification, Malaria, Disease Models, Animal, Visceral leishmaniasis, Antiprotozoal, Molecular Medicine
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15
المؤلفون: Matthias Leippe, August Stich, Thilo Waag, Tanja Schirmeister, Jennifer Rath, Christoph Gelhaus
المصدر: Bioorganicmedicinal chemistry letters. 20(18)
مصطلحات موضوعية: Proteases, Stereochemistry, Antiparasitic, medicine.drug_class, Clinical Biochemistry, Plasmodium falciparum, Trypanosoma brucei brucei, Pharmaceutical Science, Trypanosoma brucei, Cysteine Proteinase Inhibitors, Biochemistry, Cathepsin B, chemistry.chemical_compound, parasitic diseases, Drug Discovery, medicine, Animals, Humans, Disulfides, Malaria, Falciparum, Garlic, Molecular Biology, Thiosulfinate, biology, Allicin, Antiparasitic Agents, Chemistry, Organic Chemistry, biology.organism_classification, Sulfinic Acids, Cysteine protease, Cysteine Endopeptidases, Trypanosomiasis, African, Molecular Medicine, Cysteine
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16
المؤلفون: Kiplin R. Guy, Michele Connelly, David C. Smithson, Jong Yeon Hwang, Julie Maier, Fangyi Zhu
المصدر: Bioorganicmedicinal chemistry letters. 20(1)
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Trypanosoma brucei brucei, Pharmaceutical Science, Carboxamide, Trypanosoma brucei, Biochemistry, Parasitic Sensitivity Tests, parasitic diseases, Drug Discovery, medicine, Parasite hosting, Humans, African trypanosomiasis, Molecular Biology, biology, Chemistry, Organic Chemistry, Kinetoplastida, medicine.disease, biology.organism_classification, Trypanocidal Agents, In vitro, Trypanosomiasis, African, Benzamides, Molecular Medicine, Protozoa, Trypanosomiasis
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17
المؤلفون: Adam R. Renslo, Linda S. Brinen, Clifford Bryant, James H. McKerrow, Joseline Ratnam, Michelle R. Arkin, Moumita Debnath, Priyadarshini Jaishankar, Kenny K. H. Ang, Rafaela Salgado Ferreira, Iain D. Kerr, Dong-Mei Zhao
المصدر: Bioorganicmedicinal chemistry letters. 19(21)
مصطلحات موضوعية: Proteases, medicine.medical_treatment, Clinical Biochemistry, Trypanosoma brucei brucei, Pharmaceutical Science, Peptide, Trypanosoma brucei, Crystallography, X-Ray, Biochemistry, Article, Jurkat Cells, Cysteine Proteases, parasitic diseases, Drug Discovery, medicine, Humans, Protease Inhibitors, Sulfones, Binding site, Molecular Biology, chemistry.chemical_classification, Protease, Binding Sites, biology, Chemistry, Organic Chemistry, biology.organism_classification, Amides, Trypanocidal Agents, Protein Structure, Tertiary, Enzyme, Enzyme inhibitor, biology.protein, Molecular Medicine, Cysteine
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18Toward a rational design of selective multi-trypanosomatid inhibitors: a computational docking study
المصدر: Bioorganicmedicinal chemistry letters. 16(24)
مصطلحات موضوعية: Models, Molecular, Molecular model, Stereochemistry, Trypanosoma cruzi, Clinical Biochemistry, Plasmodium falciparum, Trypanosoma brucei brucei, Pharmaceutical Science, Trypanosoma brucei, Biochemistry, chemistry.chemical_compound, Entamoeba histolytica, X-Ray Diffraction, parasitic diseases, Drug Discovery, Animals, Humans, Molecular Biology, biology, Organic Chemistry, Rational design, biology.organism_classification, Trypanocidal Agents, Benzothiazole, chemistry, Docking (molecular), Drug Design, Molecular Medicine
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19
المؤلفون: Joshua Howarth, Darragh Wilson
المصدر: Bioorganicmedicinal chemistry letters. 13(12)
مصطلحات موضوعية: Bridged-Ring Compounds, Trypanosoma cruzi, Clinical Biochemistry, Plasmodium falciparum, Trypanosoma brucei brucei, Antiprotozoal Agents, Pharmaceutical Science, Trypanosoma brucei, Biochemistry, Cell Line, Apicomplexa, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Drug Discovery, Alkanes, medicine, Parasite hosting, Animals, Humans, Leishmania infantum, Molecular Biology, Tetradecane, biology, Organic Chemistry, Kinetoplastida, Leishmaniasis, General Medicine, biology.organism_classification, medicine.disease, Virology, In vitro, chemistry, Immunology, Molecular Medicine, Protozoa, Malaria
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20
المؤلفون: Valérie Landry, Louis Maes, Elisabeth Davioud-Charvet, Christian Sergheraert, Régis Millet
المصدر: Bioorganicmedicinal chemistry letters. 12(24)
مصطلحات موضوعية: Stereochemistry, Cell Survival, Trypanosoma cruzi, Clinical Biochemistry, Trypanosoma brucei brucei, Pharmaceutical Science, Trypanosoma brucei, Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Drug Discovery, parasitic diseases, Tumor Cells, Cultured, Animals, Humans, Leishmania infantum, Cytotoxicity, Molecular Biology, biology, Chemistry, Organic Chemistry, General Medicine, biology.organism_classification, Trypanocidal Agents, In vitro, Hydrazines, Nitro, Macrophages, Peritoneal, Molecular Medicine, Protozoa