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1
المؤلفون: Na Li, Hong Yang, Ke Liu, Liwei Zhou, Yuting Huang, Danyan Cao, Yanlian Li, Yaoliang Sun, Aisong Yu, Zhiyan Du, Feng Yu, Ying Zhang, Bingyang Wang, Meiyu Geng, Jian Li, Bing Xiong, Shilin Xu, Xun Huang, Tongchao Liu
المصدر: Journal of medicinal chemistry. 65(13)
مصطلحات موضوعية: Histones, Protein Domains, Catalytic Domain, Drug Discovery, Molecular Medicine, Histone-Lysine N-Methyltransferase
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2
المؤلفون: Zhaomin Liu, Shaomeng Wang, Jeanne A. Stuckey, Caroline Foster, Krishnapriya Chinnaswamy, Liyue Huang, Kaitlin P Zawacki, Sally Przybranowski, Donna McEachern, Angelo Aguilar, Ke Zheng, Shilin Xu, Tianfeng Xu
المصدر: Journal of Medicinal Chemistry. 63:4997-5010
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, endocrine system, Acute leukemia, Myeloid, endocrine system diseases, Cell growth, Chemistry, medicine.disease, Small molecule, Leukemia, medicine.anatomical_structure, In vivo, Cell culture, Covalent bond, hemic and lymphatic diseases, Drug Discovery, medicine, Cancer research, Molecular Medicine, neoplasms
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3
المؤلفون: Shilin, Xu, Angelo, Aguilar, Liyue, Huang, Tianfeng, Xu, Ke, Zheng, Donna, McEachern, Sally, Przybranowski, Caroline, Foster, Kaitlin, Zawacki, Zhaomin, Liu, Krishnapriya, Chinnaswamy, Jeanne, Stuckey, Shaomeng, Wang
المصدر: J Med Chem
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, endocrine system, endocrine system diseases, Molecular Structure, Antineoplastic Agents, Histone-Lysine N-Methyltransferase, Mice, SCID, Crystallography, X-Ray, Xenograft Model Antitumor Assays, Article, Leukemia, Myeloid, Acute, hemic and lymphatic diseases, Cell Line, Tumor, Proto-Oncogene Proteins, Animals, Azetidines, Humans, Female, Drug Screening Assays, Antitumor, neoplasms, Myeloid-Lymphoid Leukemia Protein, Protein Binding
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4
المصدر: Journal of medicinal chemistry. 62(20)
مصطلحات موضوعية: Allosteric regulation, 01 natural sciences, Autoimmune Diseases, 03 medical and health sciences, TYK2 Kinase, Heterocyclic Compounds, Psoriasis, Drug Discovery, medicine, Humans, 030304 developmental biology, Janus Kinases, 0303 health sciences, biology, Janus kinase 1, Chemistry, Active site, JAK Family, Janus Kinase 1, medicine.disease, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Tyrosine kinase 2, Cancer research, biology.protein, Molecular Medicine, Janus kinase
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5
المؤلفون: Shaomeng Wang, Denzil Bernard, Shilin Xu, James Delproposto, Ester Fernandez-Salas, Liyue Huang, Kaitlin Harvey, Jeff W. Kampf, Liu Liu, Angelo Aguilar, Jeanne A. Stuckey, Tianfeng Xu, Caroline Foster, Donna McEachern, Ke Zheng, Krishnapriya Chinnaswamy
المصدر: J Med Chem
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, endocrine system, Lineage (genetic), endocrine system diseases, HL-60 Cells, Plasma protein binding, Crystallography, X-Ray, 01 natural sciences, Article, Small Molecule Libraries, 03 medical and health sciences, Structure-Activity Relationship, MIXED LINEAGE LEUKEMIA, hemic and lymphatic diseases, Cell Line, Tumor, Proto-Oncogene Proteins, Drug Discovery, medicine, Structure–activity relationship, Humans, neoplasms, 030304 developmental biology, Cell Proliferation, 0303 health sciences, Acute leukemia, Molecular Structure, Chemistry, Cell growth, medicine.disease, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Leukemia, Models, Chemical, Cell culture, Leukemia, Myeloid, Acute Disease, Cancer research, Molecular Medicine, Myeloid-Lymphoid Leukemia Protein, Protein Binding
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6
المؤلفون: Xiaofen Pan, Zhang Zhang, Shilin Xu, Lianwen Zhang, Lei Duan, Yingxue Liu, Xiaomei Ren, Xiaoxi Zhuang, Ke Ding
المصدر: Journal of Medicinal Chemistry. 56:4631-4640
مصطلحات موضوعية: Male, Transcription, Genetic, Cell, Administration, Oral, Biological Availability, Antineoplastic Agents, Breast Neoplasms, Pharmacology, Cell Line, Rats, Sprague-Dawley, Structure-Activity Relationship, Estrogen-related receptor alpha, Estrogen-related receptor, Genes, Reporter, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, RNA, Messenger, Luciferases, Receptor, Reporter gene, Aniline Compounds, Chemistry, Triazoles, Small molecule, Rats, medicine.anatomical_structure, Receptors, Estrogen, Cell culture, Molecular Medicine, Female, Drug Screening Assays, Antitumor
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7
المؤلفون: Meiyu Geng, Yong Xu, Duanqing Pei, Xiaomei Ren, Lianwen Zhang, Tianfeng Xu, Xiaoyun Lu, Zhang Zhang, Ke Ding, Chang Shaohua, Shilin Xu, Jian Ding, Zhengchao Tu, Jinfeng Luo, Yingxue Liu
المصدر: Journal of Medicinal Chemistry. 55:2711-2723
مصطلحات موضوعية: biology, Chemistry, Kinase, Mutant, Pharmacology, respiratory tract diseases, T790M, Gefitinib, Drug Discovery, Cancer cell, Cancer research, medicine, biology.protein, Molecular Medicine, Epidermal growth factor receptor, Erlotinib, medicine.drug, EGFR inhibitors
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8
المؤلفون: Shaohua, Chang, Lianwen, Zhang, Shilin, Xu, Jinfeng, Luo, Xiaoyun, Lu, Zhang, Zhang, Tianfeng, Xu, Yingxue, Liu, Zhengchao, Tu, Yong, Xu, Xiaomei, Ren, Meiyu, Geng, Jian, Ding, Duanqing, Pei, Ke, Ding
المصدر: Journal of medicinal chemistry. 55(6)
مصطلحات موضوعية: Threonine, Lung Neoplasms, Transplantation, Heterologous, Molecular Conformation, Mice, Nude, Antineoplastic Agents, Gefitinib, Mice, SCID, ErbB Receptors, Erlotinib Hydrochloride, Mice, Structure-Activity Relationship, Methionine, Pyrimidines, Drug Resistance, Neoplasm, Carcinoma, Non-Small-Cell Lung, Drug Design, Mutation, Quinazolines, Animals, Humans, Drug Screening Assays, Antitumor, Neoplasm Transplantation, Cell Proliferation