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المصدر: Molecules; Volume 27; Issue 1; Pages: 149
Molecules, Vol 27, Iss 149, p 149 (2022)مصطلحات موضوعية: Trypanosoma brucei, natural products, human African trypanosomiasis, Trypanosoma brucei brucei, Pharmaceutical Science, Analytical Chemistry, Lactones, QD241-441, In silico screening, sesquiterpene lactones, parasitic diseases, Drug Discovery, Physical and Theoretical Chemistry, Di-hydrofolate reductase inhibitor, Human African trypanosomiasis, Natural products, Pteridine reductase 1 inhibitor, Sesquiterpene lactones, Folic Acid Antagonists, Molecular Docking Simulation, Oxidoreductases, Protein Binding, Tetrahydrofolate Dehydrogenase, Trypanocidal Agents, pteridine reductase 1 inhibitor, Organic Chemistry, dihydrofolate reductase inhibitor, Chemistry (miscellaneous), Molecular Medicine, in silico screening
وصف الملف: application/pdf
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المؤلفون: Arnold Amusengeri, Özlem Tastan Bishop, Rolland Bantar Tata
المصدر: Molecules
Volume 25
Issue 4
Molecules, Vol 25, Iss 4, p 904 (2020)مصطلحات موضوعية: Plasmodium falciparum, 030303 biophysics, Mutant, malaria, Pharmaceutical Science, Molecular Dynamics Simulation, Ligands, Article, Analytical Chemistry, lcsh:QD241-441, 03 medical and health sciences, lcsh:Organic chemistry, dihydrofolate reductase, Protein Domains, Catalytic Domain, parasitic diseases, Drug Discovery, Dihydrofolate reductase, medicine, Homology modeling, Amino Acids, Physical and Theoretical Chemistry, Binding site, 030304 developmental biology, dynamic residue network, Genetics, 0303 health sciences, drug resistance, biology, Chemistry, Point mutation, Organic Chemistry, Wild type, Active site, MD-TASK, 3. Good health, pyrimethamine, Tetrahydrofolate Dehydrogenase, Pyrimethamine, Chemistry (miscellaneous), Mutation, biology.protein, Thermodynamics, Molecular Medicine, medicine.drug
وصف الملف: application/pdf
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المؤلفون: Soledad Chazarra, María Piedad Fernández-Pérez, Magalí Sáez-Ayala, José Neptuno Rodríguez-López, Nani Mchedlishvili, Alberto Tárraga-Tomás
المصدر: Molecules, Vol 18, Iss 7, Pp 8319-8341 (2013)
Molecules
Volume 18
Issue 7
Pages 8319-8341مصطلحات موضوعية: Stereochemistry, drug design, Serum albumin, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Article, Catechin, Analytical Chemistry, lcsh:QD241-441, 03 medical and health sciences, chemistry.chemical_compound, Folic Acid, 0302 clinical medicine, dihydrofolate reductase, lcsh:Organic chemistry, Cell Line, Tumor, Drug Discovery, Dihydrofolate reductase, antifolates, Humans, Physical and Theoretical Chemistry, Serum Albumin, albumin, Cell Proliferation, 030304 developmental biology, Flavonoids, chemistry.chemical_classification, 0303 health sciences, Tea, biology, tea catechins, Organic Chemistry, Albumin, Polyphenols, Biological activity, Dissociation constant, Tetrahydrofolate Dehydrogenase, Enzyme, chemistry, Biochemistry, Chemistry (miscellaneous), Polyphenol, 030220 oncology & carcinogenesis, biology.protein, Folic Acid Antagonists, Molecular Medicine
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المؤلفون: Amnon Kohen, Kalani Karunaratne, Michael Choi
المصدر: Molecules, Vol 21, Iss 5, p 654 (2016)
Molecules (Basel, Switzerland)مصطلحات موضوعية: 0301 basic medicine, Pharmaceutical Science, mechanism, Flavin group, thymidylate synthase, Biology, 010402 general chemistry, Infections, 01 natural sciences, Thymidylate synthase, Article, Analytical Chemistry, lcsh:QD241-441, 03 medical and health sciences, chemistry.chemical_compound, lcsh:Organic chemistry, Multienzyme Complexes, Flavins, antibiotic, Drug Discovery, Dihydrofolate reductase, Thymidine Monophosphate, Humans, Physical and Theoretical Chemistry, chemistry.chemical_classification, Thymidine monophosphate, Bacteria, Organic Chemistry, biology.organism_classification, flavin, 0104 chemical sciences, 3. Good health, Anti-Bacterial Agents, De novo synthesis, Kinetics, Tetrahydrofolate Dehydrogenase, enzyme, 030104 developmental biology, Enzyme, Biochemistry, chemistry, Chemistry (miscellaneous), biology.protein, Molecular Medicine, DNA