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المؤلفون: Christopher P. Regan, Elizabeth Cauchon, Bruce Mackay, Yves Ducharme, Sylvie Toulmond, Sebastien Laliberte, Patrick Lacombe, Sébastien Gagné, M. David Percival, Daniel Dube, Jean-Pierre Falgueyret, JingQi Huang, Jean-François Lévesque, Dan McKay, Yongxin Han, René St-Jacques, Louis-Charles Campeau, Austin Chen, Hillary K. Regan, Pierre-André Fournier, Amandine Chefson, Erich L. Grimm, Robert Houle, Dwight Macdonald, Susana Liu
المصدر: Bioorganicmedicinal chemistry letters. 21(13)
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, Stereochemistry, Pyridones, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Renin inhibitor, Chemical synthesis, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, Dogs, Piperidines, In vivo, Drug Discovery, Renin–angiotensin system, Renin, medicine, Structure–activity relationship, Animals, Enzyme Inhibitors, Molecular Biology, biology, Molecular Structure, Organic Chemistry, Rats, chemistry, Enzyme inhibitor, Drug Design, Lipophilicity, Hypertension, Lactam, biology.protein, Molecular Medicine
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2
المؤلفون: Laurence Dube, David Martin, Daniel Dube, Dan McKay, Michel Gallant, Robert Houle, Austin Chen, Dwight Macdonald, Bruce Mackay, Erich L. Grimm, Suzanna Liu, Sebastien Laliberte, Patrick Lacombe, Sébastien Gagné, David A. Powell, Mireille Gaudreault, Jean-François Lévesque
المصدر: Bioorganicmedicinal chemistry letters. 20(17)
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Isozyme, chemistry.chemical_compound, Inhibitory Concentration 50, Drug Discovery, Renin–angiotensin system, Renin, Cytochrome P-450 CYP3A, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, CYP3A4, biology, Organic Chemistry, Cytochrome P450, Propanamide, Amides, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Microsomes, Liver, Molecular Medicine, Cytochrome P-450 CYP3A Inhibitors, Propionates