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1دورية أكاديميةCrystal structure of inhibitor-bound P450BM-3 reveals open conformation of substrate access channel.
المؤلفون: Haines DC; Department of Chemistry, The University of Texas at Dallas, Dallas, Texas 75083-0688, USA., Chen B, Tomchick DR, Bondlela M, Hegde A, Machius M, Peterson JA
المصدر: Biochemistry [Biochemistry] 2008 Mar 25; Vol. 47 (12), pp. 3662-70. Date of Electronic Publication: 2008 Feb 26.
نوع المنشور: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.
بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 0370623 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0006-2960 (Print) Linking ISSN: 00062960 NLM ISO Abbreviation: Biochemistry Subsets: MEDLINE
مواضيع طبية MeSH: Cytochrome P-450 Enzyme Inhibitors*, Bacterial Proteins/*antagonists & inhibitors , Bacterial Proteins/*chemistry , Cytochrome P-450 Enzyme System/*chemistry , Enzyme Inhibitors/*chemistry , Fatty Acids/*chemistry , Imidazoles/*chemistry , Leucine/*analogs & derivatives , Leucine/*chemistry , Mixed Function Oxygenases/*antagonists & inhibitors , Mixed Function Oxygenases/*chemistry, Crystallization ; Crystallography, X-Ray ; Fatty Acids/metabolism ; Fatty Acids/pharmacology ; Heme/chemistry ; Imidazoles/pharmacology ; Leucine/pharmacology ; Models, Molecular ; NADP/metabolism ; NADPH-Ferrihemoprotein Reductase ; Oxidation-Reduction/drug effects ; Protein Conformation
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2دورية أكاديمية
المؤلفون: Hegde A; Department of Biochemistry, The University of Texas Southwestern Medical Center at Dallas, Dallas, Texas 75390-9038, USA., Haines DC, Bondlela M, Chen B, Schaffer N, Tomchick DR, Machius M, Nguyen H, Chowdhary PK, Stewart L, Lopez C, Peterson JA
المصدر: Biochemistry [Biochemistry] 2007 Dec 11; Vol. 46 (49), pp. 14010-7. Date of Electronic Publication: 2007 Nov 16.
نوع المنشور: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 0370623 Publication Model: Print-Electronic Cited Medium: Print ISSN: 0006-2960 (Print) Linking ISSN: 00062960 NLM ISO Abbreviation: Biochemistry Subsets: MEDLINE
مواضيع طبية MeSH: Bacterial Proteins/*metabolism , Cytochrome P-450 Enzyme System/*metabolism , Fatty Acids/*metabolism , Mixed Function Oxygenases/*metabolism, Bacterial Proteins/chemistry ; Bacterial Proteins/genetics ; Binding Sites ; Crystallization ; Crystallography, X-Ray ; Cytochrome P-450 Enzyme System/chemistry ; Cytochrome P-450 Enzyme System/genetics ; Leucine/analogs & derivatives ; Leucine/metabolism ; Methionine/analogs & derivatives ; Methionine/metabolism ; Mixed Function Oxygenases/chemistry ; Mixed Function Oxygenases/genetics ; Models, Molecular ; NADPH-Ferrihemoprotein Reductase ; Palmitic Acids/metabolism ; Substrate Specificity
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3دورية أكاديمية
المؤلفون: Haines DC; Department of Biochemistry, The University of Texas Southwestern Medical Center at Dallas, Dallas, Texas 75390-9038, USA., Tomchick DR, Machius M, Peterson JA
المصدر: Biochemistry [Biochemistry] 2001 Nov 13; Vol. 40 (45), pp. 13456-65.
نوع المنشور: Journal Article; Research Support, U.S. Gov't, P.H.S.
بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 0370623 Publication Model: Print Cited Medium: Print ISSN: 0006-2960 (Print) Linking ISSN: 00062960 NLM ISO Abbreviation: Biochemistry Subsets: MEDLINE
مواضيع طبية MeSH: Bacterial Proteins*, Cytochrome P-450 Enzyme System/*chemistry , Glycine/*analogs & derivatives , Mixed Function Oxygenases/*chemistry , Water/*chemistry, Bacillus megaterium/enzymology ; Binding Sites ; Binding, Competitive ; Crystallization ; Crystallography, X-Ray ; Glycine/metabolism ; Heme/metabolism ; Models, Molecular ; NADPH-Ferrihemoprotein Reductase ; Palmitic Acids/metabolism ; Protein Conformation ; Protein Structure, Tertiary ; Substrate Specificity