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1
المؤلفون: Christopher I. Bayly, Dan McKay, Tom Y.-H. Wu, Patrick Roy, Suzanna Liu, Michel Gallant, Austin Chen, Helene Juteau, Rejean Fortin, Daniel Dube, Renee Aspiotis, Patrick Lacombe
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5822-5826
مصطلحات موضوعية: Molecular model, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Bibenzyls, Renin, Drug Discovery, Renin–angiotensin system, medicine, Animals, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, fungi, Organic Chemistry, Amides, In vitro, Rats, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Amine gas treating
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2
المؤلفون: Mélissa Arbour, Gavin Chit Tsui, Jean-Pierre Falgueyret, Pierre-André Fournier, Yongxin Han, Michel Gallant, Patrick Lacombe, Daniel Dube, Daniel Simard, Elizabeth Cauchon, Austin Chen, Renee Aspiotis, Suzanna Liu, René St-Jacques, Christophe Mellon, Erich L. Grimm, Yeeman K. Ramtohul, Helene Juteau
المصدر: Bioorganicmedicinal chemistry letters. 22(5)
مصطلحات موضوعية: Transgene, Clinical Biochemistry, hERG, Pharmaceutical Science, Biological Availability, Pharmacology, Biochemistry, Plasma renin activity, Rats, Sprague-Dawley, Structure-Activity Relationship, Dogs, Piperidines, Drug Discovery, Renin–angiotensin system, Renin, Structure–activity relationship, Animals, Cytochrome P-450 CYP3A, Humans, Animal species, Molecular Biology, Antihypertensive Agents, Cytochrome P-450 CYP3A Inhibitors, biology, Chemistry, Organic Chemistry, Ether-A-Go-Go Potassium Channels, Bioavailability, Rats, Hypertension, biology.protein, Molecular Medicine, Rats, Transgenic
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3
المؤلفون: Laurence Dube, David Martin, Daniel Dube, Dan McKay, Michel Gallant, Robert Houle, Austin Chen, Dwight Macdonald, Bruce Mackay, Erich L. Grimm, Suzanna Liu, Sebastien Laliberte, Patrick Lacombe, Sébastien Gagné, David A. Powell, Mireille Gaudreault, Jean-François Lévesque
المصدر: Bioorganicmedicinal chemistry letters. 20(17)
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Isozyme, chemistry.chemical_compound, Inhibitory Concentration 50, Drug Discovery, Renin–angiotensin system, Renin, Cytochrome P-450 CYP3A, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, CYP3A4, biology, Organic Chemistry, Cytochrome P450, Propanamide, Amides, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Microsomes, Liver, Molecular Medicine, Cytochrome P-450 CYP3A Inhibitors, Propionates