المؤلفون: Masci D; Department of Basic Biotechnological Sciences, Intensivological and Perioperative Clinics, Catholic University of the Sacred Heart, Largo Francesco Vito 1, Rome 00168, Italy., Puxeddu M; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy., Di Magno L; Laboratory Affiliated to Istituto Pasteur Italia─Fondazione Cenci Bolognetti, Department of Molecular Medicine, Sapienza University of Rome, Viale Regina Elena 291, Rome 00161, Italy., D'Ambrosio M; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy., Parisi A; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy., Nalli M; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy., Bai R; Molecular Pharmacology Branch, Developmental Therapeutics Program, Division of Cancer Treatment and Diagnosis, Frederick National Laboratory for Cancer Research, National Cancer Institute, National Institutes of Health, Frederick, Maryland 21702, United States., Coluccia A; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy., Sciò P; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy., Orlando V; Department of Biology and Biotechnologies 'Charles Darwin', Sapienza University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy., D'Angelo S; Department of Biology and Biotechnologies 'Charles Darwin', Sapienza University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy., Biagioni S; Department of Biology and Biotechnologies 'Charles Darwin', Sapienza University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy., Urbani A; Department of Basic Biotechnological Sciences, Intensivological and Perioperative Clinics, Catholic University of the Sacred Heart, Largo Francesco Vito 1, Rome 00168, Italy., Hamel E; Molecular Pharmacology Branch, Developmental Therapeutics Program, Division of Cancer Treatment and Diagnosis, Frederick National Laboratory for Cancer Research, National Cancer Institute, National Institutes of Health, Frederick, Maryland 21702, United States., Nocentini A; Dipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Universitá degli Studi di Firenze, Via Ugo Schiff 6, Sesto Fiorentino I-50019, Firenze, Italy., Filiberti S; Experimental Oncology and Immunology Unit, Department of Molecular and Translational Medicine, University of Brescia, Via Branze 39, Brescia 25123, Italy., Turati M; Experimental Oncology and Immunology Unit, Department of Molecular and Translational Medicine, University of Brescia, Via Branze 39, Brescia 25123, Italy., Ronca R; Experimental Oncology and Immunology Unit, Department of Molecular and Translational Medicine, University of Brescia, Via Branze 39, Brescia 25123, Italy., Kopecka J; Department of Oncology and Molecular Biotecnology Center 'Guido Tarone″, Oncological Pharmacology Unit, Via Nizza 44, Torino 10126, Italy., Riganti C; Department of Oncology and Molecular Biotecnology Center 'Guido Tarone″, Oncological Pharmacology Unit, Via Nizza 44, Torino 10126, Italy., Fionda C; Laboratory Affiliated to Istituto Pasteur Italia─Fondazione Cenci Bolognetti, Department of Molecular Medicine, Sapienza University of Rome, Viale Regina Elena 291, Rome 00161, Italy., Bordone R; Laboratory Affiliated to Istituto Pasteur Italia─Fondazione Cenci Bolognetti, Department of Molecular Medicine, Sapienza University of Rome, Viale Regina Elena 291, Rome 00161, Italy., Della Rocca G; Laboratory Affiliated to Istituto Pasteur Italia─Fondazione Cenci Bolognetti, Department of Molecular Medicine, Sapienza University of Rome, Viale Regina Elena 291, Rome 00161, Italy., Canettieri G; Laboratory Affiliated to Istituto Pasteur Italia─Fondazione Cenci Bolognetti, Department of Molecular Medicine, Sapienza University of Rome, Viale Regina Elena 291, Rome 00161, Italy., Supuran CT; Dipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Universitá degli Studi di Firenze, Via Ugo Schiff 6, Sesto Fiorentino I-50019, Firenze, Italy., Silvestri R; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy., La Regina G; Laboratory Affiliated with the Institute Pasteur Italy─Cenci Bolognetti Foundation, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Piazzale Aldo Moro 5, Roma 00185, Italy.

المصدر: Journal of medicinal chemistry [J Med Chem] 2023 Nov 09; Vol. 66 (21), pp. 14824-14842. Date of Electronic Publication: 2023 Oct 30.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't; Research Support, N.I.H., Extramural

بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrases*/metabolism , Neoplasms*, Humans ; Structure-Activity Relationship ; Drug Resistance, Multiple ; Wnt Signaling Pathway ; Drug Resistance, Neoplasm ; Carbonic Anhydrase Inhibitors/pharmacology ; Carbonic Anhydrase IX ; Molecular Structure ; Benzenesulfonamides

المؤلفون: Saied S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, P.O. Box 33516, Egypt., Shaldam M; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, P.O. Box 33516, Egypt., Elbadawi MM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, P.O. Box 33516, Egypt., Giovannuzzi S; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Via U. Schiff 6, 50019, Sesto Fiorentino, Firenze, Italy., Nocentini A; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Via U. Schiff 6, 50019, Sesto Fiorentino, Firenze, Italy., Almahli H; Department of Chemistry, University of Cambridge, CB2 1EW, Cambridge, United Kingdom., Salem R; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, P.O. Box 33516, Egypt., Ibrahim TM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, P.O. Box 33516, Egypt., Supuran CT; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Via U. Schiff 6, 50019, Sesto Fiorentino, Firenze, Italy. Electronic address: claudiu.supuran@unifi.it., Eldehna WM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, P.O. Box 33516, Egypt. Electronic address: wagdy2000@gmail.com.

المصدر: European journal of medicinal chemistry [Eur J Med Chem] 2023 Nov 05; Vol. 259, pp. 115707. Date of Electronic Publication: 2023 Aug 02.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrases*/metabolism , Antineoplastic Agents*/chemistry, Humans ; Molecular Structure ; Structure-Activity Relationship ; Oxindoles ; Molecular Docking Simulation ; Vascular Endothelial Growth Factor Receptor-2/metabolism ; Sulfonamides/chemistry ; Carbonic Anhydrase Inhibitors/chemistry ; Carbonic Anhydrase IX/metabolism ; Benzenesulfonamides

المؤلفون: Akocak S; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Adıyaman University, 02040 Adıyaman, Turkey. Electronic address: sakocak@adiyaman.edu.tr., Lolak N; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Adıyaman University, 02040 Adıyaman, Turkey., Giovannuzzi S; Università degli Studi di Firenze, Dipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Via U. Schiff 6, 50019 Sesto Fiorentino (Florence), Italy., Supuran CT; Università degli Studi di Firenze, Dipartimento Neurofarba, Sezione di Scienze Farmaceutiche e Nutraceutiche, Via U. Schiff 6, 50019 Sesto Fiorentino (Florence), Italy. Electronic address: claudiu.supuran@unifi.it.

المصدر: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2023 Oct 15; Vol. 95, pp. 129479. Date of Electronic Publication: 2023 Sep 12.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrases*/metabolism , Pyrazolones*/pharmacology , Neoplasms*, Humans ; Carbonic Anhydrase IX/metabolism ; Carbonic Anhydrase Inhibitors/pharmacology ; Isoenzymes ; Structure-Activity Relationship ; Sulfonamides/pharmacology ; Molecular Structure ; Benzenesulfonamides

المؤلفون: Benito G; Neurofarba Department, University of Florence, Sesto Fiorentino, Florence, 50019, Italy., D'Agostino I; Department of Pharmacy, University of Pisa, Pisa, 56126, Italy., Carradori S; Department of Pharmacy, 'G. d'Annunzio' University of Chieti - Pescara, Chieti, 66100, Italy., Fantacuzzi M; Department of Pharmacy, 'G. d'Annunzio' University of Chieti - Pescara, Chieti, 66100, Italy., Agamennone M; Department of Pharmacy, 'G. d'Annunzio' University of Chieti - Pescara, Chieti, 66100, Italy., Puca V; Department of Pharmacy, 'G. d'Annunzio' University of Chieti - Pescara, Chieti, 66100, Italy., Grande R; Department of Pharmacy, 'G. d'Annunzio' University of Chieti - Pescara, Chieti, 66100, Italy.; Center for Advanced Studies & Technology, 'G. d'Annunzio' University of Chieti - Pescara, Chieti, 66100, Italy., Capasso C; Department of Biology, Agriculture & Food Sciences, National Research Council, Institute of Biosciences & Bioresources, Naples, 80131, Italy., Carta F; Neurofarba Department, University of Florence, Sesto Fiorentino, Florence, 50019, Italy., Supuran CT; Neurofarba Department, University of Florence, Sesto Fiorentino, Florence, 50019, Italy.

المصدر: Future medicinal chemistry [Future Med Chem] 2023 Oct; Vol. 15 (20), pp. 1865-1883. Date of Electronic Publication: 2023 Oct 27.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: Future Science Country of Publication: England NLM ID: 101511162 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1756-8927 (Electronic) Linking ISSN: 17568919 NLM ISO Abbreviation: Future Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrases*/metabolism , Helicobacter pylori*/metabolism, Erlotinib Hydrochloride/pharmacology ; Carbonic Anhydrase Inhibitors/pharmacology ; Carbonic Anhydrase Inhibitors/chemistry ; ErbB Receptors/metabolism ; Structure-Activity Relationship ; Molecular Structure ; Carbonic Anhydrase IX ; Benzenesulfonamides

المؤلفون: Vats L; Department of Chemistry, Kurukshetra University, Kurukshetra, Haryana, 136119, India.; Department of Chemistry, Government College Bherian, Pehowa, Kurukshetra, Haryana, 136128, India., Arya P; Department of Chemistry, Kurukshetra University, Kurukshetra, Haryana, 136119, India., Kumar R; Ch. Mani Ram Godara Government College for Women, Bhodia Khera, Fatehabad, Haryana, 125050, India., Giovannuzzi S; Neurofarba Department, Pharmaceutical & Nutraceutical Section, University of Florence, Florence, Italy., Raghav N; Department of Chemistry, Kurukshetra University, Kurukshetra, Haryana, 136119, India., Supuran CT; Neurofarba Department, Pharmaceutical & Nutraceutical Section, University of Florence, Florence, Italy., Sharma PK; Department of Chemistry, Kurukshetra University, Kurukshetra, Haryana, 136119, India.; Department of Chemistry, Central University of Haryana, Mahendergarh, 123031, India.

المصدر: Future medicinal chemistry [Future Med Chem] 2023 Oct; Vol. 15 (20), pp. 1843-1863. Date of Electronic Publication: 2023 Oct 25.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: Future Science Country of Publication: England NLM ID: 101511162 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1756-8927 (Electronic) Linking ISSN: 17568919 NLM ISO Abbreviation: Future Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrases*/metabolism , Neoplasms*, Humans ; Structure-Activity Relationship ; Molecular Docking Simulation ; Triazoles/pharmacology ; Cathepsin B ; Carbonic Anhydrase Inhibitors/pharmacology ; Protein Isoforms ; Benzenesulfonamides

المؤلفون: Abdoli M; Institute of Technology of Organic Chemistry, Faculty of Materials Science and Applied Chemistry, Riga Technical University, Riga, Latvia., Krasniqi V; Pharmaceutical Institute, Pharmaceutical & Medicinal Chemistry University of Bonn, An der Immenburg 4, 53121 Bonn, Germany., Bonardi A; Neurofarba Department, Universita Degli Studi di Firenze, Florence, Italy., Gütschow M; Pharmaceutical Institute, Pharmaceutical & Medicinal Chemistry University of Bonn, An der Immenburg 4, 53121 Bonn, Germany. Electronic address: guetschow@uni-bonn.de., Supuran CT; Neurofarba Department, Universita Degli Studi di Firenze, Florence, Italy. Electronic address: claudiu.supuran@unifi.it., Žalubovskis R; Institute of Technology of Organic Chemistry, Faculty of Materials Science and Applied Chemistry, Riga Technical University, Riga, Latvia; Latvian Institute of Organic Synthesis, Riga, Latvia. Electronic address: raivis@osi.lv.

المصدر: Bioorganic chemistry [Bioorg Chem] 2023 Oct; Vol. 139, pp. 106725. Date of Electronic Publication: 2023 Jul 08.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrases*/metabolism, Structure-Activity Relationship ; Carbonic Anhydrase Inhibitors/pharmacology ; Carbonic Anhydrase Inhibitors/chemistry ; Cathepsins ; Benzenesulfonamides

المؤلفون: Hesar Shourkabi M; Department of Biology, Science and Research Branch, Islamic Azad University, Tehran, Iran., Ghobeh M; Department of Biology, Science and Research Branch, Islamic Azad University, Tehran, Iran. Electronic address: ghobeh@srbiau.ac.ir., Jafary H; Department of Biology, Science and Research Branch, Islamic Azad University, Tehran, Iran.

المصدر: Biochemical and biophysical research communications [Biochem Biophys Res Commun] 2023 Sep 24; Vol. 674, pp. 154-161. Date of Electronic Publication: 2023 Jun 19.

نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't

بيانات الدورية: Publisher: Elsevier Country of Publication: United States NLM ID: 0372516 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2104 (Electronic) Linking ISSN: 0006291X NLM ISO Abbreviation: Biochem Biophys Res Commun Subsets: MEDLINE

مواضيع طبية MeSH: Alzheimer Disease*/drug therapy , Alzheimer Disease*/genetics , Alzheimer Disease*/metabolism , Neurodegenerative Diseases* , Sulfonamides*/pharmacology, Animals ; Rats ; Amyloid beta-Peptides/metabolism ; Biomarkers/metabolism ; Gene Expression ; Oxidative Stress ; Peptide Fragments/metabolism ; Rats, Wistar ; Reactive Oxygen Species/metabolism ; Benzenesulfonamides

المؤلفون: Murugesan A; Department of Biotechnology, Lady Doak College, Madurai Kamaraj University, Thallakulam, Madurai 625002, India.; Molecular Signaling Group, Faculty of Medicine and Health Technology, Tampere University and BioMediTech, P.O. Box 553, 33101 Tampere, Finland., Konda Mani S; Department of Biotechnology, Bharath Institute of Higher Education & Research, Chennai 600073, India., Thiyagarajan R; Department of Basic Medical Sciences, College of Medicine, Prince Sattam Bin Abdulaziz University, Al-Kharj 11942, Saudi Arabia., Palanivel S; Molecular Signaling Group, Faculty of Medicine and Health Technology, Tampere University and BioMediTech, P.O. Box 553, 33101 Tampere, Finland., Gurbanov AV; Centro de Química Estrutural, Institute of Molecular Sciences, Instituto Superior Técnico, Universidade de Lisboa, Av. Rovisco Pais, 1049-001 Lisboa, Portugal.; Excellence Center, Baku State University, Z. Xalilov Str. 23, Az 1148 Baku, Azerbaijan., Zubkov FI; Organic Chemistry Department, Faculty of Science, RUDN University, 6 Miklukho-Maklaya St., 117198 Moscow, Russia., Kandhavelu M; Molecular Signaling Group, Faculty of Medicine and Health Technology, Tampere University and BioMediTech, P.O. Box 553, 33101 Tampere, Finland.

المصدر: International journal of molecular sciences [Int J Mol Sci] 2023 Jul 31; Vol. 24 (15). Date of Electronic Publication: 2023 Jul 31.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

مواضيع طبية MeSH: Glioblastoma*/drug therapy , Antineoplastic Agents*/chemistry, Humans ; Cisplatin/pharmacology ; Structure-Activity Relationship ; Molecular Docking Simulation ; Cell Proliferation ; Molecular Structure ; Drug Screening Assays, Antitumor ; Benzenesulfonamides

المؤلفون: Cysewski P; Department of Physical Chemistry, Pharmacy Faculty, Collegium Medicum of Bydgoszcz, Nicolaus Copernicus University in Toruń, Kurpińskiego 5, 85-096 Bydgoszcz, Poland., Jeliński T; Department of Physical Chemistry, Pharmacy Faculty, Collegium Medicum of Bydgoszcz, Nicolaus Copernicus University in Toruń, Kurpińskiego 5, 85-096 Bydgoszcz, Poland., Przybyłek M; Department of Physical Chemistry, Pharmacy Faculty, Collegium Medicum of Bydgoszcz, Nicolaus Copernicus University in Toruń, Kurpińskiego 5, 85-096 Bydgoszcz, Poland.

المصدر: Molecules (Basel, Switzerland) [Molecules] 2023 Jun 26; Vol. 28 (13). Date of Electronic Publication: 2023 Jun 26.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: PubMed not MEDLINE; MEDLINE

مواضيع طبية MeSH: Models, Chemical* , Water*, Solvents ; Cost-Benefit Analysis ; Solubility ; Benzenesulfonamides

المؤلفون: Żołnowska B; Department of Organic Chemistry, Medical University of Gdańsk, Al. Gen. J. Hallera 107, 80-416 Gdańsk, Poland., Sławiński J; Department of Organic Chemistry, Medical University of Gdańsk, Al. Gen. J. Hallera 107, 80-416 Gdańsk, Poland., Belka M; Department of Pharmaceutical Chemistry, Medical University of Gdańsk, Al. Gen. J. Hallera 107, 80-416 Gdańsk, Poland., Bączek T; Department of Pharmaceutical Chemistry, Medical University of Gdańsk, Al. Gen. J. Hallera 107, 80-416 Gdańsk, Poland., Chojnacki J; Department of Inorganic Chemistry, Gdańsk University of Technology, ul. Narutowicza 11/12, 80-233 Gdańsk, Poland., Kawiak A; Department of Biotechnology, Intercollegiate Faculty of Biotechnology, University of Gdańsk and Medical University of Gdańsk, ul. Abrahama 58, 80-307 Gdańsk, Poland.

المصدر: International journal of molecular sciences [Int J Mol Sci] 2023 Jun 05; Vol. 24 (11). Date of Electronic Publication: 2023 Jun 05.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

مواضيع طبية MeSH: Antineoplastic Agents*/chemistry, Humans ; Molecular Structure ; Structure-Activity Relationship ; HeLa Cells ; Cell Proliferation ; Drug Screening Assays, Antitumor ; Cell Line, Tumor ; Apoptosis ; Dose-Response Relationship, Drug ; Benzenesulfonamides