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1
المؤلفون: Deborah Galinis, Sheila J. Miknyoczki, Ted L. Underiner, Damaris Rolon-Steele, Jean Husten, Craig A. Zificsak, Thelma S. Angeles, Torsten Herbertz, Mark S. Albom, Bruce D. Dorsey, Laura S. Kocsis, Kevin J. Wells-Knecht, Jay P. Theroff, Lisa D. Aimone, Kelli S. Zeigler, Candace S. Worrell, Rebecca A. Brown, Christine LoSardo, Seetha Murthy, Jennifer Grobelny
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:660-663
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Metabolite, Clinical Biochemistry, Substituent, Administration, Oral, Mice, Nude, Pharmaceutical Science, Antineoplastic Agents, Carboxamide, Biochemistry, Chemical synthesis, Mice, chemistry.chemical_compound, In vivo, Neoplasms, Drug Discovery, medicine, Animals, Humans, Protein Kinase Inhibitors, Molecular Biology, biology, Bicyclic molecule, Chemistry, Organic Chemistry, Proto-Oncogene Proteins c-met, Xenograft Model Antitumor Assays, Pyrimidines, Diaminopyrimidine, Enzyme inhibitor, biology.protein, Molecular Medicine
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2
المؤلفون: Hong Chang, Jean Husten, Lisa D. Aimone, Thelma S. Angeles, Christine LoSardo, Karen L. Milkiewicz, Damaris Rolon-Steele, Seetha Murthy, Mark S. Albom, Jennifer Grobelny, Candace S. Worrell, Ted L. Underiner, Linda Weinberg, Bruce D. Dorsey, Kelli S. Zeigler, Sheila J. Miknyoczki
المصدر: Bioorganicmedicinal chemistry. 19(21)
مصطلحات موضوعية: Male, Spectrometry, Mass, Electrospray Ionization, C-Met, Magnetic Resonance Spectroscopy, Angiogenesis, Clinical Biochemistry, Pharmaceutical Science, Motility, Biological Availability, Mice, Nude, Antineoplastic Agents, Pharmacology, Biochemistry, Metastasis, Rats, Sprague-Dawley, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Random Allocation, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Molecular Biology, Protein Kinase Inhibitors, PK/PD models, Molecular Structure, Hepatocyte Growth Factor, Organic Chemistry, Neoplasms, Experimental, Benzazepines, Proto-Oncogene Proteins c-met, medicine.disease, Bioavailability, Rats, Diaminopyrimidine, Pyrimidines, chemistry, Molecular Medicine, Hepatocyte growth factor, Female, medicine.drug