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1دورية أكاديمية
المؤلفون: Izabella Góral, Tomasz Wichur, Emilia Sługocka, Justyna Godyń, Natalia Szałaj, Paula Zaręba, Monika Głuch-Lutwin, Barbara Mordyl, Dawid Panek, Anna Więckowska
المصدر: Molecules, Vol 29, Iss 11, p 2616 (2024)
مصطلحات موضوعية: GSK-3β, IKK-β, ROCK-1, anti-inflammatory activity, neuroprotective properties Alzheimer’s disease, Organic chemistry, QD241-441
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Barbora Svobodova, Lenka Pulkrabkova, Dawid Panek, Anna Misiachna, Marharyta Kolcheva, Rudolf Andrys, Jiri Handl, Jan Capek, Pavlina Nyvltova, Tomas Rousar, Lukas Prchal, Vendula Hepnarova, Martina Hrabinova, Lubica Muckova, Daniela Tosnerova, Galina Karabanovich, Vladimir Finger, Ondrej Soukup, Martin Horak, Jan Korabecny
المصدر: International Journal of Molecular Sciences, Vol 24, Iss 11, p 9124 (2023)
مصطلحات موضوعية: Alzheimer’s disease, acetylcholinesterase, enzyme inhibition, N-methyl-d-aspartate receptor, monoamine oxidase A/B, multi-target directed ligands, Biology (General), QH301-705.5, Chemistry, QD1-999
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Natalia Szałaj, Justyna Godyń, Jakub Jończyk, Anna Pasieka, Dawid Panek, Tomasz Wichur, Krzysztof Więckowski, Paula Zaręba, Marek Bajda, Anja Pislar, Barbara Malawska, Raimon Sabate, Anna Więckowska
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1944-1952 (2020)
مصطلحات موضوعية: multifunctional ligands, β-secretase, 5-ht6 receptor antagonists, cholinesterase inhibitors, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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4دورية أكاديمية
المؤلفون: Dawid Panek, Anna Więckowska, Anna Pasieka, Justyna Godyń, Jakub Jończyk, Marek Bajda, Damijan Knez, Stanislav Gobec, Barbara Malawska
المصدر: Molecules, Vol 23, Iss 2, p 347 (2018)
مصطلحات موضوعية: isoindoline-1,3-dione derivatives, cholinesterase inhibitors, BACE-1 inhibitors, Aβ-aggregation, molecular modeling, multiple anti-Alzheimer’s ligands, Organic chemistry, QD241-441
وصف الملف: electronic resource
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5دورية أكاديمية
المؤلفون: Michalina Hebda, Marek Bajda, Anna Więckowska, Natalia Szałaj, Anna Pasieka, Dawid Panek, Justyna Godyń, Tomasz Wichur, Damijan Knez, Stanislav Gobec, Barbara Malawska
المصدر: Molecules, Vol 21, Iss 4, p 410 (2016)
مصطلحات موضوعية: cholinesterase inhibitors, molecular modelling, β-amyloid aggregation inhibitors, Alzheimer’s disease, multi-target-directed ligands (MTDL), PAMPA-BBB assay, Organic chemistry, QD241-441
وصف الملف: electronic resource
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6
المؤلفون: Dawid Panek, Alba Espargaró, Marek Bajda, Anna Pasieka, Barbara Malawska, Anna Więckowska, Raimon Sabaté, Natalia Szałaj
المصدر: ACS Chemical Neuroscience
مصطلحات موضوعية: Molecular model, Physiology, Cognitive Neuroscience, In silico, Tau protein, Protein aggregation, aggregation inhibitors, Biochemistry, tau protein, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Alzheimer Disease, Humans, Computer Simulation, IC50, 030304 developmental biology, 0303 health sciences, Amyloid beta-Peptides, biology, molecular modeling, Chemistry, Biological activity, Cell Biology, General Medicine, Peptide Fragments, In vitro, Kinetics, Docking (molecular), Drug Design, biology.protein, Cholinesterase Inhibitors, β-Amyloid, Alzheimer’s disease, 030217 neurology & neurosurgery, Research Article
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7
المؤلفون: Anja Pišlar, Anna Więckowska, Barbara Malawska, Paula Zaręba, Raimon Sabaté, Dawid Panek, Jakub Jończyk, Tomasz Wichur, Natalia Szałaj, Anna Pasieka, Krzysztof Więckowski, Justyna Godyń, Marek Bajda
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1944-1952 (2020)
مصطلحات موضوعية: Pharmacology, cholinesterase inhibitors, 010405 organic chemistry, business.industry, Multifunctional ligands, RM1-950, General Medicine, Disease, Computational biology, multifunctional ligands, 01 natural sciences, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Multi target, Drug Discovery, β secretase, β-secretase, Medicine, Identification (biology), 5-ht6 receptor antagonists, Therapeutics. Pharmacology, business
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8
المؤلفون: Javier Egea, Daniel Diez-Iriepa, Barbara Mordyl, Alejandra Palomino-Antolín, Rim Malek, Lhassane Ismaili, Tereza Kobrlova, Justyna Godyń, Ondrej Soukup, José Marco-Contelles, Agata Siwek, Fakher Chabchoub, Ignacio Moraleda, Cristóbal de los Ríos, Dawid Panek, Céline Demougeot, Perle Totoson, Katarzyna Kieć-Kononowicz, Isabel Iriepa, Monika Głuch-Lutwin, Barbara Malawska, Raquel L Arribas
المصدر: Journal of Medicinal Chemistry. 62:11416-11422
مصطلحات موضوعية: 0303 health sciences, biology, Lipopolysaccharide, Voltage-dependent calcium channel, Pharmacology, 01 natural sciences, 0104 chemical sciences, Blockade, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, Molecular Medicine, Histamine H3 receptor, Receptor, Antagonism, IC50, 030304 developmental biology, Cholinesterase
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9
المؤلفون: Marek Bajda, Dawid Panek, Anna Pasieka, Justyna Godyń, Barbara Malawska, Damijan Knez, Jakub Jończyk, Anna Więckowska, Stanislav Gobec
المصدر: Molecules, vol. 23, no. 2, 347, 2018.
Molecules : A Journal of Synthetic Chemistry and Natural Product Chemistry
Molecules; Volume 23; Issue 2; Pages: 347
Molecules, Vol 23, Iss 2, p 347 (2018)مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Magnetic Resonance Spectroscopy, cholinesterase inhibitors, Molecular model, Pharmaceutical Science, Chemistry Techniques, Synthetic, Isoindoles, 01 natural sciences, isoindoline-1,3-dione derivatives, Analytical Chemistry, chemistry.chemical_compound, Drug Discovery, Aβ-aggregation, Butyrylcholinesterase, media_common, Molecular Structure, biology, BACE-1 inhibitors, molecular modeling, multiple anti-Alzheimer’s ligands, Alzheimerjeva bolezen, Acetylcholinesterase, Molecular Docking Simulation, Chemistry (miscellaneous), udc:616.894:615, Molecular Medicine, Drug, media_common.quotation_subject, Molecular Dynamics Simulation, multiple anti-Alzheimer's ligands, Article, lcsh:QD241-441, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, lcsh:Organic chemistry, Potency, Physical and Theoretical Chemistry, IC50, Cholinesterase, Dose-Response Relationship, Drug, 010405 organic chemistry, Organic Chemistry, Hydrogen Bonding, Isoindoline, Combinatorial chemistry, 0104 chemical sciences, 030104 developmental biology, chemistry, Drug Design, biology.protein, Amyloid Precursor Protein Secretases
وصف الملف: application/pdf; text/url
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10
المؤلفون: Tomasz, Wichur, Anna, Pasieka, Justyna, Godyń, Dawid, Panek, Izabella, Góral, Gniewomir, Latacz, Ewelina, Honkisz-Orzechowska, Adam, Bucki, Agata, Siwek, Monika, Głuch-Lutwin, Damijan, Knez, Xavier, Brazzolotto, Stanislav, Gobec, Marcin, Kołaczkowski, Raimon, Sabate, Barbara, Malawska, Anna, Więckowska
المصدر: European journal of medicinal chemistry. 225
مصطلحات موضوعية: Amyloid beta-Peptides, Indoles, Dose-Response Relationship, Drug, Molecular Structure, tau Proteins, Hep G2 Cells, Ligands, Molecular Docking Simulation, Mice, Protein Aggregates, Structure-Activity Relationship, Butyrylcholinesterase, Receptors, Serotonin, Drug Discovery, Electrophorus, Acetylcholinesterase, Microsomes, Liver, Animals, Humans, Cholinesterase Inhibitors, Horses, Cell Proliferation