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1
المؤلفون: Alexandra E. Gould, Courtney Cullis, Lee Hong Myung, David Lok, Rachel E. Gershman, Scott R. Rowland, Miho Mizutani, Dave Janowick, Gipson Krista E, Vihren Kolev, Robert J. Griffin, Joe Conlon, Steve Stroud, Akito Hata, Jeffrey Ciavarri, Dylan Bradley England, Cardin David P, Sandeep Pusalkar, Paul D. Greenspan, Adnan O Abu-Yousif, Jenna Malley, Doanh Mai, Michael Shaw, Ji Zhang, Robert J. Skene, Hu Zhigen, Matthew A. Jones, Atsushi Matsuda, Shih-Chung Huang, Nina Molchanova, Xu Tianlin, Jian Huang, He Xu, Stepan Vyskocil, Nanda Gulavita, Francois Soucy, Gang Li, Yongbo Hu, Liting Ma, Steven P. Langston, Zhan Shi, Christelle C. Renou, Luhua Shen, Sean Harrison, Elise Nunes, Kenneth M. Gigstad, Yosuke Sato, Hirotake Mizutani
المصدر: Journal of Medicinal Chemistry. 64:6902-6923
مصطلحات موضوعية: Transplantation, Heterologous, Inflammation, 01 natural sciences, Phosphates, Mice, Structure-Activity Relationship, 03 medical and health sciences, Cell Line, Tumor, Neoplasms, Drug Discovery, medicine, Animals, Humans, 030304 developmental biology, 0303 health sciences, Tumor microenvironment, Binding Sites, Innate immune system, Chemistry, Membrane Proteins, Type I interferon production, Acquired immune system, eye diseases, Rats, 0104 chemical sciences, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Sting, Pyrimidines, Stimulator of interferon genes, Cancer research, Molecular Medicine, Administration, Intravenous, Cytokine secretion, Immunotherapy, Nucleotides, Cyclic, medicine.symptom, Half-Life
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2
المؤلفون: Xingyue He, Mark G. Qian, Matthew O. Duffey, Larry Cohen, Michael D. Sintchak, Mi-Sook Kim, Jessica Riceberg, Vaishali Shindi, Kelly Connolly, Jianping Guo, Agatha Zawadzka, Rachel E. Gershman, Teresa A. Soucy, Neil Bence, Zhigen Hu, Xiaofeng Yang, Shumet A. Hailu, Nina Molchinova, Nanda Gulavita, Ji Zhang, Hirotake Mizutani, Keli Song, A D Patil, Scott Freeze, Jessica Grieves, Dylan Bradley England, Roushan Afroze, James J. Minissale, Anya Lublinsky, Mitsuhiro Ito, David Lok, Scott Weston Lane, William D. Mallender, Stephen Grossman, Kara Hoar, Nitya Durvasula, Bei-Ching Chuang, Yongbo Hu, Steven P. Langston, Sai M. Pulukuri, Miho Mizutani, Ryan Chau, Nancy Bump, Katherine M. Galvin, Christopher F. Claiborne, Paul D. Greenspan, He Xu, Gaulin Jeffrey L, Melissa Gallery, Douglas Bowman, Yana Wang, Koji Ono, Mcintyre Charles
المصدر: Journal of medicinal chemistry. 64(5)
مصطلحات موضوعية: Adenosine, SUMO protein, Antineoplastic Agents, Plasma protein binding, Ubiquitin-Activating Enzymes, 01 natural sciences, Adduct, 03 medical and health sciences, Mice, Structure-Activity Relationship, Cell Line, Tumor, Neoplasms, Drug Discovery, medicine, Structure–activity relationship, Animals, Humans, Enzyme Inhibitors, 030304 developmental biology, chemistry.chemical_classification, 0303 health sciences, Molecular Structure, Chemistry, Cancer, Sumoylation, medicine.disease, Xenograft Model Antitumor Assays, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Enzyme, Biochemistry, Cell culture, Covalent bond, Molecular Medicine, Sulfonic Acids, Protein Processing, Post-Translational, Protein Binding
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3
المؤلفون: Emily F. Calderwood, Kathleen Aertgeerts, Michael D. Smith, Dylan Bradley England, Roushan Afroze, Ryan Chau, Stepan Vyskocil, Nancy E. Forsyth, Dong Mei Zhang, Ruth Adams, Stephen G. Stroud, O. P. Veiby, Christelle C. Renou, R. Scott Rowland, Erin Paske, Jane X. Liu, Ming Tregay, Michael D. Sintchak, Juliet A Williams, Shih-Chung Huang, Xu Tianlin, Bheemashankar Kulkarni, Sharmila Adhikari, Yuan Tian, Jason Yano, Christopher Blackburn, Paul D. Greenspan, Cheryl A. Farrer, Matthew O. Duffey, Liting Ma, Mi-Sook Kim, Qin Zhang, Sean Harrison, Hirotake Mizutani, Katherine M. Galvin, Alexandra E. Gould, Johnny J. Yang, Steven P. Langston, Dave Janowick, Natalia Iartchouk, Mansoureh Rezaei, Jeffery Gaulin, Khristofer Garcia, Hongbo Zeng, Ribo Guo, Tricia J. Vos, Jouhara Chouitar, Saurabh Menon
المصدر: Journal of Medicinal Chemistry. 54:1836-1846
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, Tetrahydronaphthalenes, Mutant, Melanoma, Experimental, Administration, Oral, Biological Availability, Mice, Nude, Antineoplastic Agents, Pharmacology, Crystallography, X-Ray, Mice, Structure-Activity Relationship, Pharmacokinetics, Mouse xenograft, In vivo, Drug Discovery, medicine, Animals, chemistry.chemical_classification, Chemistry, Melanoma, Stereoisomerism, medicine.disease, Xenograft Model Antitumor Assays, In vitro, Bioavailability, Enzyme, Drug Design, Mutation, Molecular Medicine