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المؤلفون: John Victor Napoleon, Satish Sagar, Sydney P. Kubica, Lidia Boghean, Smit Kour, Hannah M. King, Yogesh A. Sonawane, Ayrianne J. Crawford, Nagsen Gautam, Smitha Kizhake, Pawel A. Bialk, Eric Kmiec, Jayapal Reddy Mallareddy, Prathamesh P. Patil, Sandeep Rana, Sarbjit Singh, Janani Prahlad, Paul M. Grandgenett, Gloria E. O. Borgstahl, Gargi Ghosal, Yazen Alnouti, Michael A. Hollingsworth, Prakash Radhakrishnan, Amarnath Natarajan
المصدر: Proceedings of the National Academy of Sciences. 119
مصطلحات موضوعية: Pancreatic Neoplasms, Multidisciplinary, Humans, MAP Kinase Kinase Kinase 1, Protein Serine-Threonine Kinases, I-kappa B Kinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6ee2183724df8b2fa739b509626495a6
https://doi.org/10.1073/pnas.2115071119 -
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المؤلفون: Sandeep Rana, Smit Kour, Smitha Kizhake, Hannah M. King, Jayapal Reddy Mallareddy, Adam J. Case, Tom Huxford, Amarnath Natarajan
المصدر: Bioorg Med Chem Lett
مصطلحات موضوعية: Isatin, Organic Chemistry, Clinical Biochemistry, NF-kappa B, Transcription Factor RelA, Pharmaceutical Science, Antineoplastic Agents, Protein Serine-Threonine Kinases, Biochemistry, Article, I-kappa B Kinase, 4-Butyrolactone, Cell Line, Tumor, Drug Discovery, Molecular Medicine, Phosphorylation, Molecular Biology
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المؤلفون: Xu Luo, Michael A. Hollingsworth, Carter J. Barger, Smit Kour, Ayrianne J. Crawford, Smitha Kizhake, Jacob I. Contreras, Hannah M. King, Amarnath Natarajan, Caroline M. Robb, Mourad Bendjennat, Sandeep Rana, Yogesh A. Sonawane
المصدر: Molecular Pharmacology
مصطلحات موضوعية: 0301 basic medicine, Cell Survival, Small Molecule Libraries, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Cyclin-dependent kinase, Cell Line, Tumor, Humans, Protein Kinase Inhibitors, Cell Proliferation, Pharmacology, Sulfonamides, Gene knockdown, Aniline Compounds, Navitoclax, Dose-Response Relationship, Drug, biology, Cell growth, Chemistry, Kinase, Cyclin-dependent kinase 2, Cyclin-Dependent Kinase 5, Drug Synergism, Articles, 3. Good health, Gene Expression Regulation, Neoplastic, Pancreatic Neoplasms, 030104 developmental biology, Apoptosis, Cell culture, Cancer research, biology.protein, Myeloid Cell Leukemia Sequence 1 Protein, Pyrazoles, Molecular Medicine, 030217 neurology & neurosurgery, HeLa Cells
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5cd3ecd3ea09bb8aee6b6189f5a1903a
https://doi.org/10.1124/mol.119.116855 -
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المؤلفون: Smitha Kizhake, Smit Kour, Muhammad Zahid, Hannah M. King, Mourad Bendjennat, Amarnath Natarajan, Sandeep Rana
المصدر: Bioorg Med Chem Lett
مصطلحات موضوعية: Models, Molecular, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Palbociclib, 01 natural sciences, Biochemistry, Article, Piperazines, Structure-Activity Relationship, Drug Discovery, Humans, Binding site, Protein Kinase Inhibitors, Molecular Biology, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, biology, 010405 organic chemistry, Kinase, Organic Chemistry, Cyclin-Dependent Kinase 6, 0104 chemical sciences, Cell biology, 010404 medicinal & biomolecular chemistry, Enzyme, chemistry, Selective degradation, Proteolysis, biology.protein, Molecular Medicine, Cyclin-dependent kinase 6, Function (biology)
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المؤلفون: Meher Rizvi, Mohammad Abid, Bushra Zeya, Sandeep Rana, Farheen Shamsi, Jered C. Garrison, Parvez Khan, Phool Hasan, Muhammad Zahid, Hannah M. King, Mohamed F. Alajmi, Imtaiyaz Hassan, Aarfa Queen, Afzal Hussain
المصدر: Bioorganic chemistry. 98
مصطلحات موضوعية: Drug, Colorectal cancer, media_common.quotation_subject, Oxadiazole, Antineoplastic Agents, 01 natural sciences, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Tumor Cells, Cultured, Potency, Humans, Doxorubicin, Thiazole, Molecular Biology, media_common, Cell Proliferation, Oxadiazoles, Sulfonamides, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Chemistry, Organic Chemistry, Sulfonamide (medicine), medicine.disease, 0104 chemical sciences, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Apoptosis, Cancer research, Drug Screening Assays, Antitumor, Colorectal Neoplasms, medicine.drug
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المؤلفون: Michael A. Hollingsworth, Jared Baxter, Sandeep Rana, Caroline M. Robb, Yogesh A. Sonawane, Smit Kour, Ayrianne J. Crawford, Xu Luo, Smitha Kizhake, Jacob I. Contreras, Amarnath Natarajan, Hannah M. King
المصدر: ACS Chemical Biology. 13:1148-1152
مصطلحات موضوعية: 0301 basic medicine, Cell, Caspase 3, Biochemistry, Article, 03 medical and health sciences, 0302 clinical medicine, Cyclin-dependent kinase, Cell Line, Tumor, Neoplasms, medicine, Humans, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, biology, Chemistry, Kinase, General Medicine, High-Throughput Screening Assays, 030104 developmental biology, medicine.anatomical_structure, Proto-Oncogene Proteins c-bcl-2, Cell culture, Apoptosis, Doxycycline, 030220 oncology & carcinogenesis, biology.protein, Cancer research, Molecular Medicine, Drug Therapy, Combination, Apoptosis Regulatory Proteins, Genetic screen
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المؤلفون: Hannah M. King, Edward L. Ezell, Smitha Kizhake, Muhammad Zahid, Sydney P. Kubica, Michael J. Naldrett, Jayapal Reddy Mallareddy, Amarnath Natarajan, Henry C.-H. Law, Sophie Alvarez, Nicholas T. Woods, Sandeep Rana
المصدر: Bioorg Med Chem Lett
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, 01 natural sciences, Biochemistry, Article, Structure-Activity Relationship, chemistry.chemical_compound, Cyclin-dependent kinase, Drug Discovery, Humans, Kinome, Protein Kinase Inhibitors, Molecular Biology, Cell Proliferation, Sulfonamides, Dose-Response Relationship, Drug, Molecular Structure, biology, 010405 organic chemistry, Venetoclax, Kinase, Organic Chemistry, Proteolysis targeting chimera, Bridged Bicyclo Compounds, Heterocyclic, Cyclin-Dependent Kinase 9, 0104 chemical sciences, Pancreatic Neoplasms, 010404 medicinal & biomolecular chemistry, chemistry, Proteolysis, Cancer research, biology.protein, Pyrazoles, Molecular Medicine, Oncogene MYC, Cyclin-dependent kinase 9, Drug Screening Assays, Antitumor, Growth inhibition