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1
المؤلفون: Deborah Galinis, Sheila J. Miknyoczki, Ted L. Underiner, Damaris Rolon-Steele, Jean Husten, Craig A. Zificsak, Thelma S. Angeles, Torsten Herbertz, Mark S. Albom, Bruce D. Dorsey, Laura S. Kocsis, Kevin J. Wells-Knecht, Jay P. Theroff, Lisa D. Aimone, Kelli S. Zeigler, Candace S. Worrell, Rebecca A. Brown, Christine LoSardo, Seetha Murthy, Jennifer Grobelny
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:660-663
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Metabolite, Clinical Biochemistry, Substituent, Administration, Oral, Mice, Nude, Pharmaceutical Science, Antineoplastic Agents, Carboxamide, Biochemistry, Chemical synthesis, Mice, chemistry.chemical_compound, In vivo, Neoplasms, Drug Discovery, medicine, Animals, Humans, Protein Kinase Inhibitors, Molecular Biology, biology, Bicyclic molecule, Chemistry, Organic Chemistry, Proto-Oncogene Proteins c-met, Xenograft Model Antitumor Assays, Pyrimidines, Diaminopyrimidine, Enzyme inhibitor, biology.protein, Molecular Medicine
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2
المؤلفون: Edward R. Bacon, Robert L. Hudkins, Thelma S. Angeles, Jennifer Grobelny, Mark S. Albom, Reddeppareddy Dandu, Bruce Ruggeri, Sheila J. Miknyoczki, Lisa D. Aimone, Shi Yang, Candy Robinson, Hong Chang, Allison L. Zulli, Ted L. Underiner
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:1916-1921
مصطلحات موضوعية: Umbilical Veins, Hemangiosarcoma, Clinical Biochemistry, Melanoma, Experimental, Administration, Oral, Pharmaceutical Science, Angiogenesis Inhibitors, Biochemistry, Chemical synthesis, Receptor tyrosine kinase, Structure-Activity Relationship, chemistry.chemical_compound, Oximes, Drug Discovery, Animals, Humans, Structure–activity relationship, Receptor, Protein Kinase Inhibitors, Molecular Biology, Cells, Cultured, Cell Proliferation, chemistry.chemical_classification, Molecular Structure, Neovascularization, Pathologic, biology, Organic Chemistry, Oxime, Receptor, TIE-2, Vascular Endothelial Growth Factor Receptor-2, Rats, Enzyme, chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Endothelium, Vascular, Signal transduction
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3
المؤلفون: Hong Chang, Jean Husten, Lisa D. Aimone, Thelma S. Angeles, Christine LoSardo, Karen L. Milkiewicz, Damaris Rolon-Steele, Seetha Murthy, Mark S. Albom, Jennifer Grobelny, Candace S. Worrell, Ted L. Underiner, Linda Weinberg, Bruce D. Dorsey, Kelli S. Zeigler, Sheila J. Miknyoczki
المصدر: Bioorganicmedicinal chemistry. 19(21)
مصطلحات موضوعية: Male, Spectrometry, Mass, Electrospray Ionization, C-Met, Magnetic Resonance Spectroscopy, Angiogenesis, Clinical Biochemistry, Pharmaceutical Science, Motility, Biological Availability, Mice, Nude, Antineoplastic Agents, Pharmacology, Biochemistry, Metastasis, Rats, Sprague-Dawley, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Random Allocation, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Molecular Biology, Protein Kinase Inhibitors, PK/PD models, Molecular Structure, Hepatocyte Growth Factor, Organic Chemistry, Neoplasms, Experimental, Benzazepines, Proto-Oncogene Proteins c-met, medicine.disease, Bioavailability, Rats, Diaminopyrimidine, Pyrimidines, chemistry, Molecular Medicine, Hepatocyte growth factor, Female, medicine.drug
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4
المؤلفون: Bruce Ruggeri, Jean Husten, Robert L. Hudkins, Allison L. Zulli, Candace S. Worrell, Mark A. Ator, Ralph E. Parchment, Natalie McGann, Hong Chang, Jennifer Grobelny, Sonya Pritchard, Sheila J. Miknyoczki, James Deibold
المصدر: Molecular cancer therapeutics. 6(8)
مصطلحات موضوعية: G2 Phase, Cancer Research, Poly Adenosine Diphosphate Ribose, DNA Repair, medicine.medical_treatment, Carbazoles, Antineoplastic Agents, Phthalimides, Pharmacology, Poly(ADP-ribose) Polymerase Inhibitors, Irinotecan, Mice, In vivo, Glioma, Neuroblastoma, Cell Line, Tumor, medicine, Temozolomide, Animals, Humans, Enzyme Inhibitors, Cell Proliferation, Chemotherapy, Cell Death, Chemistry, Drug Synergism, Prodrug, medicine.disease, Xenograft Model Antitumor Assays, Rats, Dacarbazine, Oncology, Drug Resistance, Neoplasm, Topotecan, Camptothecin, Comet Assay, medicine.drug, DNA Damage
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::990d268dbb0f39d13870fa875a5028cd
https://pubmed.ncbi.nlm.nih.gov/17699724 -
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المؤلفون: Mangeng Cheng, Lisa D. Aimone, Sheila J. Miknyoczki, Robert J. Bendesky, Thelma S. Angeles, Jie Qian, Robert L. Hudkins, Bruce D. Dorsey, Jean Husten, Bruce Ruggeri, Thomas Conners, Seetha Murthy, Hong Chang, Amy J. Landis, Jennifer Grobelny, Mark A. Ator
المصدر: Molecular Cancer Therapeutics. 12:C275-C275
مصطلحات موضوعية: Cancer Research, biology, Chemistry, Kinase, Cancer, medicine.disease, Receptor tyrosine kinase, Metastasis, c-Met inhibitor, Therapeutic index, Oncology, Tumor progression, Cancer cell, Immunology, biology.protein, medicine, Cancer research
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::247e348a81300a0bd69b9c09bd262614
https://doi.org/10.1158/1535-7163.targ-13-c275