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1دورية أكاديمية
المؤلفون: Chuan Hong, Noel J. Byrne, Beata Zamlynny, Srivanya Tummala, Li Xiao, Jennifer M. Shipman, Andrea T. Partridge, Christina Minnick, Michael J. Breslin, Michael T. Rudd, Shawn J. Stachel, Vanessa L. Rada, Jeffrey C. Kern, Kira A. Armacost, Scott A. Hollingsworth, Julie A. O’Brien, Dawn L. Hall, Terrence P. McDonald, Corey Strickland, Alexei Brooun, Stephen M. Soisson, Kaspar Hollenstein
المصدر: Nature Communications, Vol 12, Iss 1, Pp 1-11 (2021)
مصطلحات موضوعية: Science
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2041-1723
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المؤلفون: Corey Strickland, Christina Minnick, Michael J. Breslin, Srivanya Tummala, Kaspar Hollenstein, Alexei Brooun, Vanessa L. Rada, Shawn J. Stachel, Beata Zamlynny, Kira A. Armacost, Dawn L. Hall, Li Xiao, Terrence P. McDonald, Chuan Hong, Kern Jeffrey, Scott A. Hollingsworth, Stephen M. Soisson, Julie A. O'Brien, Andrea T. Partridge, Jennifer M. Shipman, Michael T. Rudd, Noel Byrne
المصدر: Nature Communications, Vol 12, Iss 1, Pp 1-11 (2021)
Nature Communicationsمصطلحات موضوعية: Agonist, Protein Conformation, alpha-Helical, medicine.drug_class, Science, Genetic Vectors, General Physics and Astronomy, Aminopyridines, Gene Expression, Peptide, Plasma protein binding, Pharmacology, Molecular Dynamics Simulation, General Biochemistry, Genetics and Molecular Biology, Article, G protein-coupled receptors, Cryoelectron microscopy, Orexin Receptors, medicine, Escherichia coli, Humans, Protein Interaction Domains and Motifs, Cloning, Molecular, chemistry.chemical_classification, Sulfonamides, Multidisciplinary, Binding Sites, Chemistry, HEK 293 cells, digestive, oral, and skin physiology, General Chemistry, Azepines, Triazoles, medicine.disease, Small molecule, Orexin receptor, Recombinant Proteins, Orexin, HEK293 Cells, Sleep Aids, Pharmaceutical, Orexin Receptor Antagonists, Protein Conformation, beta-Strand, Peptides, Narcolepsy, Protein Binding
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المؤلفون: Jennifer M. Johnston, Karen O. Akinsanya, Jason E. Imbriglio, Noel Byrne, Hratch J. Zokian, Sookhee Ha, Scott P. Salowe, Hyewon Youm, George H. Addona, JeanMarie Lisnock, Vijayalakshmi Agnani, Deborah L. Zink, Kake Zhao, Gregory C. Adam, Yusheng Xiong, Brian K. Hubbard, Pravien Abeywickrema, John P. Caldwell, Yongcheng Huang, Jen Baysarowich, Peter Orth, Wonsuk Chang, Juncai Meng, Michael Kavana, James R. Tata, Whitney Lane Petrilli, Rui Liang, Gopal Parthasarathy, Xi Ai, Rachael E. Ford, Zhe Feng, Oksana C. Palyha, Edward DiNunzio, Stephen M. Soisson, Alison M. Strack, Jennifer M. Shipman, Roman S. Erdmann, Zhijian Lu, Sujata Sharma, Jun Lu
مصطلحات موضوعية: Models, Molecular, Thermal shift assay, Serine Proteinase Inhibitors, Clinical Biochemistry, Allosteric regulation, Drug Evaluation, Preclinical, Protein degradation, Ligands, 01 natural sciences, Biochemistry, Small Molecule Libraries, Drug Discovery, Humans, Molecular Biology, Pharmacology, Serine protease, biology, Molecular Structure, 010405 organic chemistry, Chemistry, PCSK9, Proprotein convertase, Ligand (biochemistry), Small molecule, 0104 chemical sciences, Proteolysis, biology.protein, Molecular Medicine, Kexin, Proprotein Convertase 9
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::46333ceb2ad6ba949e70430572ed5675
https://doi.org/10.26434/chemrxiv.8800085 -
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المؤلفون: Nathaniel L. Elsen, Zangwei Xu, Peter J. Dandliker, Peter Saradjian, Keith W. Rickert, Berengere Sauvagnat, Nadya Smotrov, Dawn L. Hall, Elliott B. Nickbarg, Yiping Chen, Sujata Sharma, Kevin J. Lumb, Maria Kornienko, Noel Byrne, Chad Chamberlin, Christine Andrews, Samantha J Allen, Ilona Kariv, Jennifer M. Shipman, Patrick J. Curran, Kevin G. Coleman, Beutel Bruce A, Rachael E. Ford, Victoria Kutilek, Andrew Hashke, Rafael Fernandez, Tianxiao Sun, Matthew Richards, Ryan Boinay
المصدر: SLAS Discovery. 21:608-619
مصطلحات موضوعية: 0301 basic medicine, High-throughput screening, Phenotypic screening, Cell, Druggability, Computational biology, Biology, Ligands, Bioinformatics, 01 natural sciences, Biochemistry, Mass Spectrometry, Analytical Chemistry, Structure-Activity Relationship, 03 medical and health sciences, Drug Discovery, medicine, TNF Receptor-Associated Factor 5, Reverse pharmacology, 010405 organic chemistry, Drug discovery, NF-kappa B, Transcription Factor RelA, Ligand (biochemistry), Phenotype, High-Throughput Screening Assays, 0104 chemical sciences, 030104 developmental biology, medicine.anatomical_structure, Molecular Medicine, Protein Binding, Signal Transduction, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::321009edd98ca17a57d26928e293e5e3
https://doi.org/10.1177/1087057116637353 -
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المؤلفون: Kevin J. Lumb, Stephen M. Soisson, Jennifer M. Shipman, Gopal Parthasarathy, Dawn L. Hall, Scott A. Johnson, Keith W. Rickert, Rachael E. Ford, Ronald E. Diehl, Samantha J Allen, Paul Zuck, Paul L. Darke, Sanjeev Munshi, John C. Reid
المصدر: Journal of Biological Chemistry. 290:20360-20373
مصطلحات موضوعية: inorganic chemicals, Models, Molecular, G-Protein-Coupled Receptor Kinase 4, Protein Conformation, Molecular Sequence Data, Mitogen-activated protein kinase kinase, Biology, Crystallography, X-Ray, environment and public health, Biochemistry, Substrate Specificity, MAP2K7, Humans, Amino Acid Sequence, Phosphorylation, Kinase activity, Molecular Biology, Sequence Homology, Amino Acid, MAP kinase kinase kinase, Autophosphorylation, Cyclin-dependent kinase 2, Cyclin-dependent kinase 3, Cell Biology, Cell biology, enzymes and coenzymes (carbohydrates), Protein Structure and Folding, Hypertension, biology.protein, bacteria, Cyclin-dependent kinase 9, biological phenomena, cell phenomena, and immunity
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::206a2a57c447e93465670375d12ebb66
https://doi.org/10.1074/jbc.m115.648907 -
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المؤلفون: Peter A. Lemaire, Chad Chamberlin, Kevin J. Lumb, Daniel Krosky, Alicja Krasowska-Zoladek, Xianshu Yang, Stephen M. Soisson, John M. Sanders, Hua-Poo Su, John C. Reid, Mark T. Bilodeau, Jennifer M. Shipman, Srivanya Tummala, Maria Kornienko, Marina Bukhtiyarova, Abdelghani Achab, Andrew J. Cooke, Christine Burlein, Kartik Narayan, Peter Saradjian, Craig A. Stump, Keith W. Rickert, Danielle M. Hurzy, Berengere Sauvagnat, Amanda Heller, Elliott B. Nickbarg, Xufang Zhang, Darrell A. Henze, Steven S. Carroll, Michael Ziebell
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, animal structures, Protein Conformation, Drug Evaluation, Preclinical, Tropomyosin receptor kinase B, Tropomyosin receptor kinase A, Crystallography, X-Ray, Tropomyosin receptor kinase C, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Humans, Receptor, trkB, Receptor, trkC, Amino Acid Sequence, Binding site, Receptor, trkA, Protein Kinase Inhibitors, Multidisciplinary, Binding Sites, Membrane Glycoproteins, Chemistry, Surface Plasmon Resonance, Ligand (biochemistry), Recombinant Proteins, Cell biology, Kinetics, 030104 developmental biology, nervous system, Biochemistry, Protein kinase domain, PNAS Plus, Trk receptor, Pharmacophore, 030217 neurology & neurosurgery
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d6c57357524723b0ea51de3310b10d9b
https://europepmc.org/articles/PMC5255611/ -
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المؤلفون: Harold G. Selnick, Nathaniel L. Elsen, Sangita B. Patel, Dawn L. Hall, John C. Reid, Fred Hess, Maria Kornienko, Hari Kandula, Daniel J. Klein, Rachael E. Ford, Sujata Sharma, Kevin J. Lumb, Stephen M. Soisson, Jennifer M. Shipman
المصدر: Nature chemical biology. 13(6)
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Dimer, Crystal structure, Calorimetry, Crystallography, X-Ray, 01 natural sciences, Models, Biological, Acetylglucosamine, Substrate Specificity, Serine, 03 medical and health sciences, chemistry.chemical_compound, Protein structure, Catalytic Domain, Hydrolase, Humans, Binding site, Threonine, Enzyme Inhibitors, Molecular Biology, Binding Sites, 010405 organic chemistry, Drug discovery, Chemistry, Cell Biology, beta-N-Acetylhexosaminidases, 0104 chemical sciences, Protein Structure, Tertiary, Enzyme Activation, Crystallography, 030104 developmental biology
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المؤلفون: Rachael E. Ford, Ranabir SinhaRoy, Wayne M. Geissler, Sujata Sharma, Keith W. Rickert, Pravien D. Abeywickrema, Noel Byrne, Kelly Ann D. Pryor, John C. Reid, Dawn L. Hall, Ronald E. Diehl, Kevin J. Lumb, Stephen M. Soisson, Jennifer M. Shipman, Sangita B. Patel
المصدر: Acta Crystallographica Section F Structural Biology and Crystallization Communications. 66:702-705
مصطلحات موضوعية: Glycosylation, genetic structures, Biophysics, Gene Expression, macromolecular substances, CHO Cells, Carboxypeptidases, Crystallography, X-Ray, Biochemistry, law.invention, chemistry.chemical_compound, Cricetulus, Structural Biology, law, Cricetinae, Gene expression, Genetics, Animals, Humans, Proline, Crystallization, chemistry.chemical_classification, biology, Chinese hamster ovary cell, Condensed Matter Physics, biology.organism_classification, Carboxypeptidase, Amino acid, chemistry, Crystallization Communications, biology.protein
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المؤلفون: John C. Reid, Bradley W. Thomas, Paul Kelley, Sanjeev Munshi, Hua-Poo Su, Jennifer M. Shipman, Keith W. Rickert, Noel Byrne, Paul L. Darke, Dawn L. Hall, Ronald E. Diehl, Allison M. Montalvo
المصدر: Journal of Biological Chemistry. 283:34864-34872
مصطلحات موضوعية: Epithelial sodium channel, Protein Folding, Protein Conformation, Proteolysis, Molecular Sequence Data, Protein Renaturation, Molecular Conformation, Crystallography, X-Ray, Guanidines, Biochemistry, Inclusion bodies, Substrate Specificity, Protein structure, Escherichia coli, Extracellular, medicine, Humans, Amino Acid Sequence, Protein precursor, Molecular Biology, Serine protease, Sequence Homology, Amino Acid, biology, medicine.diagnostic_test, Chemistry, Serine Endopeptidases, Cell Biology, Benzamidines, Cell biology, Hypertension, Protein Structure and Folding, biology.protein, Protein folding, Apoproteins
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::af50b945cab45fa758b67de45dd1402b
https://doi.org/10.1074/jbc.m805262200 -
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المؤلفون: John T. Sisko, Christine Fernandes, Bradley K. Wong, Patrice A. Ciecko, Nancy E. Kohl, Mark T. Bilodeau, Keith W. Rickert, Laura Sepp-Lorenzino, Leonard D. Rodman, Timothy J. Koester, Jackson B. Gibbs, Cynthia Miller-Stein, Debra A. McLoughlin, Joseph J. Lynch, Carolyn A. Buser, George D. Hartman, Xianzhi Mao, Kathleen E. Coll, Kenneth A. Thomas, Jennifer M. Shipman, Thomas J. Tucker
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:1146-1150
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Sensitivity and Specificity, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Growth factor receptor, Nitriles, parasitic diseases, Drug Discovery, Animals, Thiazole, Protein Kinase Inhibitors, neoplasms, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Chemistry, Kinase, Organic Chemistry, Macaca mulatta, Vascular Endothelial Growth Factor Receptor-2, Rats, Thiazoles, Pyrimidines, Enzyme, Enzyme inhibitor, cardiovascular system, biology.protein, Molecular Medicine, Amine gas treating, circulatory and respiratory physiology