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1
المؤلفون: Nicola J. Curtin, Bernard T. Golding, Roger J. Griffin, David R. Newell, Marion Barton, Hannah Barlow, Julian S. Northen, Mei-Ju Lin, Lan-Zhen Wang, Kappusamy Saravanan, Huw D. Thomas
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::77920703b9bfbb55eab67ef3d2666043
https://doi.org/10.1158/1535-7163.c.6532236 -
2
المؤلفون: Nicola J. Curtin, Bernard T. Golding, Roger J. Griffin, David R. Newell, Marion Barton, Hannah Barlow, Julian S. Northen, Mei-Ju Lin, Lan-Zhen Wang, Kappusamy Saravanan, Huw D. Thomas
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4fca8588aa26a79a4189b98acd55ca00
https://doi.org/10.1158/1535-7163.22486086.v1 -
3
المؤلفون: Bernard T. Golding, Mei-Ju Lin, Lan-Zhen Wang, Roger J. Griffin, HC Barlow, Marion Barton, Kappusamy Saravanan, Julian S. Northen, Huw D. Thomas, David R. Newell, Nicola J. Curtin
المصدر: Molecular Cancer Therapeutics. 8:1828-1837
مصطلحات موضوعية: Antimetabolites, Antineoplastic, Cancer Research, Guanine, Lung Neoplasms, Mice, Nude, Pemetrexed, Pharmacology, Thymidylate synthase, Nucleoside salvage, Mice, chemistry.chemical_compound, Glutamates, In vivo, Tumor Cells, Cultured, Animals, Humans, Prodrugs, Tissue Distribution, Phosphorylation, Leukemia L1210, Hypoxanthine, Cell Proliferation, Mice, Inbred BALB C, biology, Drug Synergism, Nucleosides, Dipyridamole, Orosomucoid, Thymidylate Synthase, Prodrug, Xenograft Model Antitumor Assays, Oncology, chemistry, Antifolate, biology.protein, Folic Acid Antagonists, Female, Thymidine, Nucleoside
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8f254167c1691f5608c320d506eaaf8e
https://doi.org/10.1158/1535-7163.mct-08-1208 -
4
المؤلفون: Bernard T. Golding, Claire Hutton, Shafiq U. Ahmed, Rebecca J. Reid, Stefano Norbedo, Stuart J. Kemp, John Lunec, Kappusamy Saravanan, Julian S. Northen, Henriëtte M. G. Willems, Gillian Farnie, Roger J. Griffin, Martin S. Kitching, Helen Atkins, Ian R. Hardcastle, Per Källblad, Sabrina Guyenne, David R. Newell
المصدر: Journal of Medicinal Chemistry. 49:6209-6221
مصطلحات موضوعية: Models, Molecular, Indoles, Transcription, Genetic, Stereochemistry, In silico, Antineoplastic Agents, Stereoisomerism, Plasma protein binding, Chemical synthesis, Protein–protein interaction, Gene product, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, Combinatorial Chemistry Techniques, Humans, Structure–activity relationship, Chemistry, Proto-Oncogene Proteins c-mdm2, Small molecule, Biochemistry, Molecular Medicine, Drug Screening Assays, Antitumor, Tumor Suppressor Protein p53, Protein Binding
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المؤلفون: Shafiq U. Ahmed, Rebecca J. Reid, Roger J. Griffin, Martin S. Kitching, Per Källblad, Stuart J. Kemp, John Lunec, Julian S. Northen, Gillian Farnie, Claire Hutton, Helen Atkins, Ian R. Hardcastle, Bernard T. Golding, Stefano Norbedo, David R. Newell, A. Hilary Calvert, Sabrina Guyenne, Nicola J. Curtin, Henriëtte M. G. Willems, Kappusamy Saravanan
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:1515-1520
مصطلحات موضوعية: Models, Molecular, Indoles, Transcription, Genetic, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Gene product, Structure-Activity Relationship, Transactivation, Transcription (biology), Cell Line, Tumor, Proto-Oncogene Proteins, Drug Discovery, Humans, Structure–activity relationship, Cytotoxicity, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Nuclear Proteins, Proto-Oncogene Proteins c-mdm2, Molecular biology, In vitro, Cell culture, Docking (molecular), Molecular Medicine, Tumor Suppressor Protein p53, Protein Binding
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المؤلفون: Roger J. Griffin, Celine Cano, Bernard T. Golding, Attilla Ting, Mark Frigerio, Keith Allan Menear, Julia Bardos, Christopher M. Bailey, Marc Geoffrey Hummersone, Kappusamy Saravanan, Kerry Shea, Ian R. Hardcastle, Caroline Richardson, Nicola J. Curtin, Pia Thommes, Graeme C. M. Smith, David R. Newell
المصدر: Journal of medicinal chemistry. 56(16)
مصطلحات موضوعية: Chemistry, Stereochemistry, Morpholines, DNA-Activated Protein Kinase, In vitro, chemistry.chemical_compound, In vivo, Morpholine, Drug Discovery, Molecular Medicine, Moiety, Humans, Phosphatidylinositol, Protein kinase A, Cytotoxicity, Protein Kinase Inhibitors, Acetamide, HeLa Cells, Phosphoinositide-3 Kinase Inhibitors
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المؤلفون: HC Barlow, Huw D. Thomas, Julian S. Northen, Bernard T. Golding, Alan Hilary Calvert, Nicola J. Curtin, M Barton, Roger J. Griffin, Kappusamy Saravanan, Newell
المصدر: Journal of medicinal chemistry. 54(6)
مصطلحات موضوعية: Purine, Antimetabolites, Antineoplastic, Guanine, Pyrimidine, Stereochemistry, Antineoplastic Agents, Pemetrexed, chemistry.chemical_compound, Structure-Activity Relationship, Glutamates, Cell Line, Tumor, Drug Discovery, Humans, Prodrugs, Hypoxanthine, Chemistry, Biological Transport, Drug Synergism, Nucleosides, Stereoisomerism, Orosomucoid, Prodrug, Pyrimidines, Biochemistry, Molecular Medicine, Growth inhibition, Thymidine, Nucleoside, Protein Binding
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المؤلفون: Graeme C. M. Smith, Nicola J. Curtin, Kerry Shea, Marc Geoffrey Hummersone, David R. Newell, Celine Cano, Kappusamy Saravanan, Keith Allan Menear, Roger J. Griffin, Bernard T. Golding, Julia Bardos, Mark Frigerio, Ian R. Hardcastle, Christopher M. Bailey
المصدر: Cancer Research. 70:5780-5780
مصطلحات موضوعية: chemistry.chemical_classification, Cancer Research, Kinase, Chemistry, Serine, chemistry.chemical_compound, Enzyme, Oncology, Biochemistry, Phosphatidylinositol, Threonine, Protein kinase A, IC50, DNA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::74e254e6947e0e7fc339e17e26917056
https://doi.org/10.1158/1538-7445.am10-5780 -
9دورية أكاديمية
المؤلفون: Kappusamy Saravanan, Hannah C. Barlow, Marion Barton, A. Hilary Calvert, Bernard T. Golding, David R. Newell, Julian S. Northen, Nicola J. Curtin, Huw D. Thomas, Roger J. Griffin
المصدر: Journal of Medicinal Chemistry; Mar2011, Vol. 54 Issue 6, p1847-1859, 13p