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1
المؤلفون: Gregory R. Ott, Linda Weinberg, Henry J. Breslin, Lisa D. Aimone, Diane E. Gingrich, Kevin J. Wells-Knecht, Mark A. Ator, Gregory J. Wells, Mehran Yazdanian, Eugen F. Mesaros, Zeqi Huang, Kelli S. Zeigler, Bruce D. Dorsey, Mangeng Cheng
المصدر: Chemical Research in Toxicology. 24:1994-2003
مصطلحات موضوعية: Spectrometry, Mass, Electrospray Ionization, Stereochemistry, Chemistry, Pharmaceutical, Toxicology, Mice, Troglitazone, chemistry.chemical_compound, Dogs, Biotransformation, medicine, Animals, Bile, Humans, Pyrroles, Sulfhydryl Compounds, Chromans, Clozapine, Protein Kinase Inhibitors, Chromatography, High Pressure Liquid, chemistry.chemical_classification, Triazines, Kinase, Haplorhini, General Medicine, Glutathione, In vitro, Rats, Biochemistry, chemistry, Toxicity, Microsomes, Liver, Microsome, Thiol, Thiazolidinediones, Protein Kinases, Chromatography, Liquid, medicine.drug
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2
المؤلفون: Deborah Galinis, Sheila J. Miknyoczki, Ted L. Underiner, Damaris Rolon-Steele, Jean Husten, Craig A. Zificsak, Thelma S. Angeles, Torsten Herbertz, Mark S. Albom, Bruce D. Dorsey, Laura S. Kocsis, Kevin J. Wells-Knecht, Jay P. Theroff, Lisa D. Aimone, Kelli S. Zeigler, Candace S. Worrell, Rebecca A. Brown, Christine LoSardo, Seetha Murthy, Jennifer Grobelny
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:660-663
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Metabolite, Clinical Biochemistry, Substituent, Administration, Oral, Mice, Nude, Pharmaceutical Science, Antineoplastic Agents, Carboxamide, Biochemistry, Chemical synthesis, Mice, chemistry.chemical_compound, In vivo, Neoplasms, Drug Discovery, medicine, Animals, Humans, Protein Kinase Inhibitors, Molecular Biology, biology, Bicyclic molecule, Chemistry, Organic Chemistry, Proto-Oncogene Proteins c-met, Xenograft Model Antitumor Assays, Pyrimidines, Diaminopyrimidine, Enzyme inhibitor, biology.protein, Molecular Medicine
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3
المؤلفون: Hong Chang, Jean Husten, Lisa D. Aimone, Thelma S. Angeles, Christine LoSardo, Karen L. Milkiewicz, Damaris Rolon-Steele, Seetha Murthy, Mark S. Albom, Jennifer Grobelny, Candace S. Worrell, Ted L. Underiner, Linda Weinberg, Bruce D. Dorsey, Kelli S. Zeigler, Sheila J. Miknyoczki
المصدر: Bioorganicmedicinal chemistry. 19(21)
مصطلحات موضوعية: Male, Spectrometry, Mass, Electrospray Ionization, C-Met, Magnetic Resonance Spectroscopy, Angiogenesis, Clinical Biochemistry, Pharmaceutical Science, Motility, Biological Availability, Mice, Nude, Antineoplastic Agents, Pharmacology, Biochemistry, Metastasis, Rats, Sprague-Dawley, chemistry.chemical_compound, Inhibitory Concentration 50, Mice, Random Allocation, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Molecular Biology, Protein Kinase Inhibitors, PK/PD models, Molecular Structure, Hepatocyte Growth Factor, Organic Chemistry, Neoplasms, Experimental, Benzazepines, Proto-Oncogene Proteins c-met, medicine.disease, Bioavailability, Rats, Diaminopyrimidine, Pyrimidines, chemistry, Molecular Medicine, Hepatocyte growth factor, Female, medicine.drug
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4
المؤلفون: Kelli S. Zeigler, Joel W. Proksch, Jeanelle E. McSurdy-Freed, Keith W. Ward, Gary J. Stelman, Brian R. Smith, Jayme A. Morgan, Jonathan R Kehler, Leonard M. Azzarano
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 32(2)
مصطلحات موضوعية: Drug, Male, Time Factors, CYP3A, media_common.quotation_subject, Drug Evaluation, Preclinical, Pharmaceutical Science, Administration, Oral, Biological Availability, Pharmacology, Absorption, Xenobiotics, First pass effect, Pharmacokinetics, In vivo, medicine, Animals, Cytochrome P-450 CYP3A, ATP Binding Cassette Transporter, Subfamily B, Member 1, media_common, P-glycoprotein, biology, Dose-Response Relationship, Drug, Oxidoreductases, N-Demethylating, Propranolol, Bioavailability, Erythromycin, Macaca fascicularis, Ketoconazole, Liver, Area Under Curve, Injections, Intravenous, biology.protein, Aryl Hydrocarbon Hydroxylases, medicine.drug, Half-Life
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7b343f51bb773bf547873e0fffa9f799
https://pubmed.ncbi.nlm.nih.gov/14744938