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المؤلفون: Pearl S. Huang, David A. Tuveson, Michael M. Morrissey, Meenhard Herlyn, Keiran S.M. Smalley, Rooja G. Contractor, Jerry L. Adams, Ami S. Lakdawala, Lusong Luo, Michael D. Schaber, Cynthia M. Rominger, Earl W. May, Thomas J. Stout, David Chau, Jae Lee, Julie C. Lougheed, Florian Karreth, Lifu Wang, Erin Hugger, David M. Wilson, Andrew K. Takle, David W. Rusnak, Rakesh Kumar, Shu Yun Zhang, Hieu T. Do, Maureen L. Ho, Roberta S. Batorsky, Denis R. Patrick, Alastair J. King
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7b44fc16eeff8bc76ddb0a7cbaf43c3c
https://doi.org/10.1158/0008-5472.22366893 -
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المؤلفون: Pearl S. Huang, David A. Tuveson, Michael M. Morrissey, Meenhard Herlyn, Keiran S.M. Smalley, Rooja G. Contractor, Jerry L. Adams, Ami S. Lakdawala, Lusong Luo, Michael D. Schaber, Cynthia M. Rominger, Earl W. May, Thomas J. Stout, David Chau, Jae Lee, Julie C. Lougheed, Florian Karreth, Lifu Wang, Erin Hugger, David M. Wilson, Andrew K. Takle, David W. Rusnak, Rakesh Kumar, Shu Yun Zhang, Hieu T. Do, Maureen L. Ho, Roberta S. Batorsky, Denis R. Patrick, Alastair J. King
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0381879a2c972a32b228b92d1ab7d021
https://doi.org/10.1158/0008-5472.22366890 -
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المؤلفون: Pearl S. Huang, David A. Tuveson, Michael M. Morrissey, Meenhard Herlyn, Keiran S.M. Smalley, Rooja G. Contractor, Jerry L. Adams, Ami S. Lakdawala, Lusong Luo, Michael D. Schaber, Cynthia M. Rominger, Earl W. May, Thomas J. Stout, David Chau, Jae Lee, Julie C. Lougheed, Florian Karreth, Lifu Wang, Erin Hugger, David M. Wilson, Andrew K. Takle, David W. Rusnak, Rakesh Kumar, Shu Yun Zhang, Hieu T. Do, Maureen L. Ho, Roberta S. Batorsky, Denis R. Patrick, Alastair J. King
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::04a844d6f2ddb9f8350543123fa932bd
https://doi.org/10.1158/0008-5472.22366896.v1 -
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المؤلفون: Pearl S. Huang, David A. Tuveson, Michael M. Morrissey, Meenhard Herlyn, Keiran S.M. Smalley, Rooja G. Contractor, Jerry L. Adams, Ami S. Lakdawala, Lusong Luo, Michael D. Schaber, Cynthia M. Rominger, Earl W. May, Thomas J. Stout, David Chau, Jae Lee, Julie C. Lougheed, Florian Karreth, Lifu Wang, Erin Hugger, David M. Wilson, Andrew K. Takle, David W. Rusnak, Rakesh Kumar, Shu Yun Zhang, Hieu T. Do, Maureen L. Ho, Roberta S. Batorsky, Denis R. Patrick, Alastair J. King
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::25ae9912cc76ff8cd428267b7e6b1596
https://doi.org/10.1158/0008-5472.c.6495336.v1 -
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المؤلفون: Shendong Yuan, Robert G. Wei, Andrea DiMella, Michael Snider, Dewan Zheng, Babu Subramanyam, Imadul Islam, Raju Mohan, Michael M. Morrissey, Brad O. Buckman, Laura Dunning, Wei Xu, Jih-Lie Tseng, Judi Bryant
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:1459-1463
مصطلحات موضوعية: 0301 basic medicine, P2Y receptor, Chemistry, High-throughput screening, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Hit to lead, Plasma levels, 030204 cardiovascular system & hematology, Pharmacology, Metabolic stability, Biochemistry, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, P2Y12, Drug Discovery, Molecular Medicine, Molecular Biology, Liver microsomes
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المؤلفون: Damian Arnaiz, Gary Phillips, Shawn David Erickson, Marc Whitlow, Margaret Kenrick, James J. Devlin, Gonghua Pan, Cecile Santos, William J. Guilford, Robert G. Wei, Marc Adler, Kurt W. Saionz, Bin Ye, Ron Vergona, John Parkinson, Zuchun Spring Zhao, David D. Davey, Michael Ohlmeyer, Babu Subramanyam, Vidyadhar M. Paradkar, Mark A. Polokoff, Keith A. Eagen, Michael M. Morrissey
المصدر: Journal of Medicinal Chemistry. 50:1146-1157
مصطلحات موضوعية: Male, Models, Molecular, Gene isoform, Nitric Oxide Synthase Type II, Crystallography, X-Ray, Chemical synthesis, Cell Line, Nitric oxide, chemistry.chemical_compound, Oxidoreductase, Chlorocebus aethiops, Drug Discovery, Animals, Benzodioxoles, Binding site, chemistry.chemical_classification, biology, Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Imidazoles, Biological activity, Arthritis, Experimental, Rats, Nitric oxide synthase, Pyrimidines, Enzyme, Biochemistry, Rats, Inbred Lew, biology.protein, Molecular Medicine, Dimerization
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المؤلفون: Roberta S. Batorsky, Jerry L. Adams, Shu Yun Zhang, Michael D. Schaber, Rakesh Kumar, Julie Lougheed, Thomas J. Stout, Erin Hugger, Meenhard Herlyn, David Chau, Maureen L. Ho, Ami S. Lakdawala, Earl May, Rooja G. Contractor, Jae Lee, Pearl S. Huang, Andrew K. Takle, Hieu T. Do, Lusong Luo, David M. Wilson, Michael M. Morrissey, Lifu Wang, Cynthia M. Rominger, David A. Tuveson, Alastair J. King, Denis R. Patrick, David W. Rusnak, Keiran S.M. Smalley, Florian A. Karreth
المصدر: Cancer Research. 66:11100-11105
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, Cancer Research, Protein Conformation, Blotting, Western, Mice, Nude, Biology, Crystallography, X-Ray, medicine.disease_cause, Mice, Cell Movement, Mutant protein, Cell Line, Tumor, Neoplasms, Gene expression, medicine, Animals, Humans, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Protein Kinase Inhibitors, Alleles, Cell Proliferation, Molecular Structure, Kinase, Imidazoles, Xenograft Model Antitumor Assays, Molecular biology, Blot, Oncology, Protein kinase domain, Mechanism of action, Cell culture, Mutation, Cancer research, Female, medicine.symptom, Crystallization, Carcinogenesis, HT29 Cells
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a0c07ce13bb3eaa1a428ffcbce4a6d18
https://doi.org/10.1158/0008-5472.can-06-2554 -
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المؤلفون: Guo Ping Wei, Christian Weber, John G. Bauman, H. Daniel Perez, Ghannam Ameen F, Joseph Hesselgesser, Brad O. Buckman, Michael M. Morrissey, Ng Howard P, R. Michael Snider, Zhaohui Wang, Wei Xu, Richard Horuk, Peter J. Nelson, Imadul Islam, Mary Rosser, Kim S. C. Weber, Hermann Josef Gröne, Carol Clayberger, Alan M. Krensky, Monahan Sean D, Laura Dunning, Meina Liang, Karen May
المصدر: Journal of Biological Chemistry. 276:4199-4204
مصطلحات موضوعية: Graft Rejection, Male, Agonist, CCR1, Chemokine, medicine.drug_class, medicine.medical_treatment, Receptors, CCR1, Biology, Biochemistry, Cell Line, Chemokine receptor, Piperidines, medicine, Animals, Humans, Molecular Biology, Heart transplantation, Phenylurea Compounds, Graft Survival, Antagonist, Cell Biology, medicine.disease, Receptor antagonist, Rats, Transplant rejection, Rats, Inbred Lew, Immunology, Cyclosporine, biology.protein, Heart Transplantation, Receptors, Chemokine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::878f551401bcfa7987af8c947333087a
https://doi.org/10.1074/jbc.m007457200 -
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المؤلفون: Ghannam Ameen F, Monahan Sean D, H. Daniel Perez, Susan Harvey, Wei Xu, Laura Dunning, Joseph Hesselgesser, Richard Horuk, Jun Shen, Elena Ho, Ng Howard P, Ron Vergona, Mary Rosser, Karen May, Babu Subramanyam, Imadul Islam, Cornell Mallari, John G. Bauman, Zuchun Zhao, Huynh Oanh, R. Michael Snider, Guo-Ping Wei, Ken Shaw, Meina Liang, Brad O. Buckman, Dennis D. Taub, Michael M. Morrissey
المصدر: Journal of Biological Chemistry. 275:19000-19008
مصطلحات موضوعية: Male, CCR1, Leukocyte migration, DNA, Complementary, Receptors, CCR1, Administration, Oral, Pharmacology, Binding, Competitive, Biochemistry, Cell Line, Chemokine Receptor Antagonist, Dogs, Piperidines, medicine, Animals, Humans, Receptor, Molecular Biology, Chemistry, Phenylurea Compounds, Monocyte, Antagonist, Chemotaxis, Cell Biology, Rats, medicine.anatomical_structure, Rats, Inbred Lew, Receptors, Chemokine, CC chemokine receptors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::96836a4797891eb0ce582451db65d51a
https://doi.org/10.1074/jbc.m001222200 -
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المؤلفون: Joseph Hesselgesser, Mary Rosser, M. Liang, Richard Horuk, R. M. Snider, Ghannam Ameen F, John G. Bauman, P. J. Kretschmer, Ng Howard P, Michael M. Morrissey, H. D. Perez, Imadul Islam, Laura Dunning, Karen May, Haifeng Pu
المصدر: European Journal of Pharmacology. 389:41-49
مصطلحات موضوعية: CCR1, Chemokine, DNA, Complementary, Molecular Sequence Data, Receptors, CCR1, Biology, Piperazines, Mice, Chemokine receptor, Piperidines, Species Specificity, Nitriles, Functional selectivity, medicine, Animals, Humans, Amino Acid Sequence, Cloning, Molecular, Chemokine CCL4, Receptor, Chemokine CCL5, Chemokine CCL3, Pharmacology, Binding Sites, Antagonist, Callithrix, Macrophage Inflammatory Proteins, Molecular biology, Mechanism of action, Biochemistry, Competitive antagonist, biology.protein, Calcium, Receptors, Chemokine, Rabbits, medicine.symptom