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1دورية أكاديمية
المؤلفون: Lucy O. Ojomoko, Elena V. Kryukova, Natalya S. Egorova, Arthur I. Salikhov, Lyubov A. Epifanova, Daria A. Denisova, Alex R. Khomutov, Dmitry A. Sukhov, Alexander A. Vassilevski, Maxim A. Khomutov, Victor I. Tsetlin, Irina V. Shelukhina
المصدر: Frontiers in Pharmacology, Vol 14 (2023)
مصطلحات موضوعية: nicotinic acetylcholine receptor, oligoarginine, polyamines, acylpolyamine, radioligand analysis, electrophysiology, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Irina V. Shelukhina, Maxim N. Zhmak, Alexander V. Lobanov, Igor A. Ivanov, Alexandra I. Garifulina, Irina N. Kravchenko, Ekaterina A. Rasskazova, Margarita A. Salmova, Elena A. Tukhovskaya, Vladimir A. Rykov, Gulsara A. Slashcheva, Natalya S. Egorova, Inessa S. Muzyka, Victor I. Tsetlin, Yuri N. Utkin
المصدر: Toxins, Vol 10, Iss 1, p 34 (2018)
مصطلحات موضوعية: nicotinic acetylcholine receptor, azemiopsin, preclinical studies, toxicity, pharmacokinetics, myorelaxant, Key Contribution, Investigation of the preclinical profile of azemiopsin demonstrated its high affinity and specificity for muscle type nicotinic acetylcholine receptor as well as good muscle relaxant capacity. Toxicology studies in mice indicated that azemiopsin was well tolerated during chronic dosing and showed no immunotoxicity, allergenic or mutagenic activity, which made it a good candidate for application as a local muscle relaxant., Medicine
وصف الملف: electronic resource
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3
المؤلفون: Natalya S. Egorova, Tr. D. Nguyen, V. I. Tsetlin, Khoa Cuu Nguyen, Anh Ngoc Hoang, T. N. Nguyen, Q. N. Tran, Vladislav G. Starkov, Yu. N. Utkin
المصدر: Doklady Biochemistry and Biophysics. 487:251-255
مصطلحات موضوعية: chemistry.chemical_classification, Drug Carriers, Sulfates, Chemistry, Neurotoxins, Biophysics, Capsules, Venom, Peptide, Nicotinic Antagonists, General Chemistry, General Medicine, Receptors, Nicotinic, Biochemistry, Nanomaterials, Nicotinic acetylcholine receptor, Nicotinic agonist, Polysaccharides, Nanoparticles, Neurotoxin, Particle Size, Receptor, Snake Venoms, Acetylcholine receptor
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4
المؤلفون: V. I. Tsetlin, Igor E. Kasheverov, Natalya S. Egorova, D. A. Senko, Ekaterina N. Spirova, D. S. Lebedev, Igor Ivanov, Elena V. Kryukova
المصدر: Doklady Biochemistry and Biophysics. 483:313-315
مصطلحات موضوعية: 0301 basic medicine, alpha7 Nicotinic Acetylcholine Receptor, Arginine, Biophysics, Peptide, Ligands, Torpedo, complex mixtures, Biochemistry, law.invention, 03 medical and health sciences, chemistry.chemical_compound, law, Peptide synthesis, Animals, Receptor, Acetylcholine receptor, chemistry.chemical_classification, General Chemistry, General Medicine, Radioligand Assay, 030104 developmental biology, Nicotinic agonist, nervous system, chemistry, Peptides
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5
المؤلفون: Igor E. Kasheverov, Oksana V. Nekrasova, Marina V. Serebryakova, Natalya S. Egorova, Maxim N. Zhmak, Victor I. Tsetlin, Andrei M. Gigolaev, Igor Ivanov, Nikita A. Prokopev, Peter B. Oparin, Anh Ngoc Hoang, Denis S. Kudryavtsev, Yuri N. Utkin, Alexander A. Vassilevski
المصدر: FEBS lettersReferences. 593(19)
مصطلحات موضوعية: animal structures, Xenopus, Biophysics, Scorpion Venoms, Nicotinic Antagonists, Receptors, Nicotinic, complex mixtures, Biochemistry, 03 medical and health sciences, Mice, Structural Biology, Genetics, medicine, Neurotoxin, Animals, Molecular Biology, Heterometrus laoticus, Ion channel, 030304 developmental biology, Acetylcholine receptor, 0303 health sciences, biology, Chemistry, 030302 biochemistry & molecular biology, Cell Biology, biology.organism_classification, Nicotinic acetylcholine receptor, Nicotinic agonist, nervous system, Acetylcholine, medicine.drug, Protein Binding
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6
المؤلفون: Margarita A Salmova, A. V. Lobanov, Natalya S. Egorova, G. A. Slashcheva, Victor I. Tsetlin, Maxim N. Zhmak, Elena A Tukhovskaya, Inessa S. Muzyka, Igor Ivanov, I. N. Kravchenko, Irina V. Shelukhina, Alexandra I. Garifulina, Ekaterina A Rasskazova, Yuri N. Utkin, V. A. Rykov
المصدر: Toxins
Toxins; Volume 10; Issue 1; Pages: 34
Toxins, Vol 10, Iss 1, p 34 (2018)مصطلحات موضوعية: 0301 basic medicine, Male, medicine.drug_class, Health, Toxicology and Mutagenesis, Xenopus, lcsh:Medicine, Investigation of the preclinical profile of azemiopsin demonstrated its high affinity and specificity for muscle type nicotinic acetylcholine receptor as well as good muscle relaxant capacity. Toxicology studies in mice indicated that azemiopsin was well tolerated during chronic dosing and showed no immunotoxicity, allergenic or mutagenic activity, which made it a good candidate for application as a local muscle relaxant, CHO Cells, Nicotinic Antagonists, Viper Venoms, Pharmacology, Receptors, Nicotinic, Toxicology, Article, nicotinic acetylcholine receptor, azemiopsin, preclinical studies, toxicity, pharmacokinetics, myorelaxant, Key Contribution, Rats, Sprague-Dawley, 03 medical and health sciences, Cricetulus, Cell Line, Tumor, Toxicity Tests, medicine, Animals, Humans, Receptor, Mice, Inbred ICR, GABAA receptor, Chemistry, lcsh:R, Antagonist, Muscle relaxant, Effective dose (pharmacology), Nicotinic acetylcholine receptor, 030104 developmental biology, Neuromuscular Agents, Toxicity, Oocytes, Female, Peptides, Acetylcholine, medicine.drug
وصف الملف: application/pdf
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7
المؤلفون: Eugene V. Grishin, Peter V. Dubovskii, Olga V. Samsonova, Alexander S. Arseniev, Sergey A. Kozlov, Alexei V. Feofanov, Natalya S. Egorova, Alexander A. Vassilevski
المصدر: FEBS Journal. 278:4382-4393
مصطلحات موضوعية: chemistry.chemical_classification, biology, Spider Venoms, Toxin, Venom, Peptide, Cell Biology, Bioinformatics, medicine.disease_cause, biology.organism_classification, Spider toxin, Biochemistry, chemistry, Lynx spider, medicine, Molecular Biology, Peptide sequence, Frog Skin
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8
المصدر: Biochimie. 93:227-241
مصطلحات موضوعية: Erythrocytes, Dose-Response Relationship, Drug, Membrane permeability, Chemistry, media_common.quotation_subject, Spherocyte, Erythrocyte Membrane, Echinocyte, Spider Venoms, Phosphatidylserines, General Medicine, Mitochondrion, Hemolysis, Biochemistry, Cell biology, Membrane, Humans, K562 Cells, Internalization, Cytotoxicity, Porosity, Antimicrobial Cationic Peptides, media_common, K562 cells
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9
المصدر: Biochimica et Biophysica Acta (BBA) - Biomembranes. 1778(10):2361-2367
مصطلحات موضوعية: Molecular Sequence Data, Biophysics, Biochemistry, Receptor tyrosine kinase, Transmembrane domain, Protein structure, Glycophorin, Humans, Amino Acid Sequence, Receptor, Micelles, biology, Chemistry, Receptor, EphA1, Erythropoietin-producing hepatocellular (Eph) receptor, Cell Biology, EphA1 receptor, Protein Structure, Tertiary, Enzyme Activation, Liposomes, FRET, biology.protein, Signal transduction, Peptides, Tyrosine kinase, Dimerization, SDS-PAGE, Signal Transduction
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10
المؤلفون: Tatiana B. Stoilova, Andrey Y. Surovoy, Vadim T. Ivanov, Natalya S. Egorova, Sergey I. Kovalchuk
المصدر: Biochimica et Biophysica Acta (BBA) - Biomembranes. 1778(10):2026-2031
مصطلحات موضوعية: Amphipathic peptides, Cell Membrane Permeability, Genetic Vectors, Molecular Sequence Data, Biophysics, Peptide, Cell-penetrating peptide, Biochemistry, Cell Line, chemistry.chemical_compound, Transduction (genetics), Mice, Gramicidin A, Drug Delivery Systems, Amphiphile, Animals, Humans, Amino Acid Sequence, chemistry.chemical_classification, Protein delivery, Gramicidin, Biological activity, Cell Biology, beta-Galactosidase, Anti-Bacterial Agents, chemistry, Peptides, Intracellular, Macromolecule