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المؤلفون: Daniel Grant, Peter Teriete, John C. Reed, Pooi-San Lee, Anna Dembo, Douglas J. Sheffler, Nicholas D. P. Cosford, Haixia Zou, Gavin Magnuson, Allison S. Limpert, Jiwen Zou, Anthony B. Pinkerton, Mark E. Goldman, Robert Ardecky, Juan Rong
المصدر: ACS Chemical Neuroscience
مصطلحات موضوعية: Programmed cell death, Leupeptins, MAP Kinase Signaling System, Physiology, Cognitive Neuroscience, p38 mitogen-activated protein kinases, p38 MAPK, Biology, Biochemistry, Cell Line, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, thapsigargin, medicine, Animals, Homeostasis, Humans, Enzyme Inhibitors, Oleanolic Acid, Progenitor cell, 030304 developmental biology, Neurons, Benzodiazepinones, 0303 health sciences, calcium homeostasis, Cell Death, Dose-Response Relationship, Drug, Kinase, Ionomycin, Endoplasmic reticulum, Neurodegeneration, neurodegeneration, Imidazoles, Benzodiazepinone, Cell Biology, General Medicine, Endoplasmic Reticulum Stress, medicine.disease, Rats, 3. Good health, Cell biology, Mitogen-activated protein kinase, Unfolded protein response, biology.protein, Calcium, ER stress, 030217 neurology & neurosurgery, Research Article
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المؤلفون: Srinivasa Reddy Natala, Shyama Siddique, David Carney, Ann Mladek, Jeffrey Stebbins, Li Yang, Pooi San Lee, Daniel Brimberry, Robert Ardecky, Peter Teriete, Allan Rubenstein, Jann Sarkaria, Nicholas Cosford, Sridhar Prasad
مصطلحات موضوعية: Cancer Research, Abstracts, Oncology, Neurology (clinical)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6a0e79f40065af744033add193aacc19
https://europepmc.org/articles/PMC5475182/ -
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المؤلفون: Manoranjan S. D’Souza, Andre Der-Avakian, Hilary Highfield Nickols, Douglas J. Sheffler, Melinda Davis, Raveendra-Panickar Dhanya, P. Jeffrey Conn, Li Yang, Nicholas D. P. Cosford, Russell Dahl, Pooi San Lee, Layton H. Smith, Athina Markou, Hyekyung P. Cho
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: Male, Allosteric modulator, Allosteric regulation, Pharmacology, Receptors, Metabotropic Glutamate, Article, Cocaine-Related Disorders, 03 medical and health sciences, 0302 clinical medicine, Allosteric Regulation, stomatognathic system, parasitic diseases, Drug Discovery, Animals, Humans, Rats, Wistar, Receptor, 030304 developmental biology, ADME, 0303 health sciences, Dose-Response Relationship, Drug, Metabotropic glutamate receptor 5, Chemistry, Glutamate receptor, Rats, 3. Good health, Disease Models, Animal, HEK293 Cells, Metabotropic receptor, Drug Design, embryonic structures, Molecular Medicine, Metabotropic glutamate receptor 2, 030217 neurology & neurosurgery
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المؤلفون: John C. Reed, Pooi San Lee, Kate Welsh, Kristiina Vuori, Darren Finlay, Nicholas D. P. Cosford, Palaniyandi Ravanan, Peter D. Mace, Marcos González-López, Robert Ardecky, Stefan J. Riedl, Santhi Ganji
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:4253-4257
مصطلحات موضوعية: Cell Survival, Peptidomimetic, Clinical Biochemistry, Pharmaceutical Science, X-Linked Inhibitor of Apoptosis Protein, Plasma protein binding, Inhibitor of apoptosis, Biochemistry, Article, TNF-Related Apoptosis-Inducing Ligand, Structure-Activity Relationship, Biomimetic Materials, Cell Line, Tumor, Drug Discovery, Humans, Structure–activity relationship, Molecular Biology, Binding Sites, Chemistry, Organic Chemistry, Rational design, Ligand (biochemistry), Protein Structure, Tertiary, XIAP, Molecular Docking Simulation, Drug Resistance, Neoplasm, Apoptosis, Drug Design, Cancer research, Molecular Medicine, Oligopeptides, Protein Binding
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المؤلفون: Sridhar G. Prasad, Pooi San Lee, Peter Teriete, Srinivasa Reddy, Robert Ardecky, Jann N. Sarkaria, Li Yang, Nicholas D. P. Cosford, David Carney, Ann C. Mladek, Daniel Brimberry, Shyama Sidique, Jeffrey Stebbins, Allan Rubenstein
المصدر: Neuro-Oncology. 19:vi61-vi61
مصطلحات موضوعية: Cancer Research, biology, business.industry, HSP90 Heat-Shock Proteins, medicine.disease, Hsp90, Molecular conformation, Abstracts, Oncology, Cancer research, biology.protein, Medicine, Neurology (clinical), Primary Brain Tumors, business, Glioblastoma
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dbdcb6eb119211555760769bcec32f42
https://doi.org/10.1093/neuonc/nox168.248 -
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المؤلفون: José Luis Millán, Pooi San Lee, Colin Farquharson, Nicholas D. P. Cosford, Eduard Sergienko, Raveendra Panickar Dhanya, Layton H. Smith, Peter Teriete, Yalda Bravo, Tina Kiffer-Moreira, Russell Dahl, Santhi Ganji
مصطلحات موضوعية: Phosphoric monoester hydrolases, Clinical Biochemistry, Phosphatase, Pharmaceutical Science, Biochemistry, Article, Small Molecule Libraries, Mice, Structure-Activity Relationship, Drug Discovery, High-Throughput Screening Assays, Structure–activity relationship, Animals, Humans, Benzothiazoles, Enzyme Inhibitors, Molecular Biology, ADME, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Hydrogen-Ion Concentration, Small molecule, In vitro, Phosphoric Monoester Hydrolases, Drug Design, Benzamides, Hepatocytes, Molecular Medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::55a28de140d9b826c3f7ff210fda84e1
https://europepmc.org/articles/PMC4170737/ -
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المؤلفون: John C. Reed, Scott J. Snipas, Nicholas D. P. Cosford, Mitchell Vamos, Darren Finlay, Monica L. Gonzalez, Guy S. Salvesen, Kate Welsh, Pooi San Lee, Peter D. Mace, Kristiina Vuori, Santhi Ganji, Stefan J. Riedl, Robert Ardecky
مصطلحات موضوعية: Models, Molecular, Fluorescence Polarization, Inhibitor of apoptosis, Biochemistry, Article, Inhibitor of Apoptosis Proteins, medicine, Fibroblast, Melanoma, Caspase, biology, Cancer, General Medicine, medicine.disease, Caspase Inhibitors, XIAP, body regions, medicine.anatomical_structure, Cell culture, Apoptosis, Drug Design, Cancer cell, biology.protein, Cancer research, Molecular Medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::339df1d3e8e3ef9896e4fd837d1ba780
https://europepmc.org/articles/PMC3953502/