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المؤلفون: Julia H Shin, Steven A. Gilbert, Vikram R. Rao, Betsy J. Barnes, Lih-Ling Lin, Ken Dower, Virginia Pascual, Bruce A. Jacobson, Iain Kilty, Jean J Beebe, Tatyana Andreyeva, Bruce L. Homer, Joanne Brodfuehrer, Weiyong Sun, Martin Hegen, Simeon Ramsey, M Nusrat Sharif, Margaret Fleming, Mera Tilley, Heng Liu, Aaron Winkler, Aiping Jiao, Saurav De, Shruti Athale, Peter T. Symanowicz, Ju Wang, Spencer I. Danto
المصدر: Arthritis & Rheumatology. 73:2206-2218
مصطلحات موضوعية: Lactams, Immunology, Arthritis, Inflammation, Peripheral blood mononuclear cell, Mice, Rheumatology, In vivo, Rheumatic Diseases, medicine, Animals, Humans, Immunology and Allergy, Kinase activity, skin and connective tissue diseases, Systemic lupus erythematosus, business.industry, Macrophages, Autoantibody, Dendritic Cells, Isoquinolines, medicine.disease, IRAK4, Arthritis, Experimental, Synoviocytes, Rats, Disease Models, Animal, Interleukin-1 Receptor-Associated Kinases, Leukocytes, Mononuclear, medicine.symptom, business
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2
المؤلفون: Anthony R. Harris, Susan M. Lotarski, Michael Aaron Brodney, Michael Popiolek, Catherine A. Thorn, Stephen Jenkinson, Che Wah Lee, Jennifer E. Davoren, Stefanus J. Steyn, Lei Zhang, Terrence Peter Kenakin, Betty Pettersen, Sarah Grimwood, Damien Webb, Michelle R. Garnsey, Simeon Ramsey, John T. Lazzaro, Steven Victor O'neil, Lisa Nottebaum, Jean-Philippe Fortin, Jeremy R. Edgerton
المصدر: Journal of Medicinal Chemistry. 60:6649-6663
مصطلحات موضوعية: 0301 basic medicine, Agonist, Allosteric modulator, medicine.drug_class, Chemistry, Allosteric regulation, Muscarinic acetylcholine receptor M1, Pharmacology, 03 medical and health sciences, 030104 developmental biology, Drug Discovery, Convulsion, medicine, Molecular Medicine, Cholinergic, Structure–activity relationship, medicine.symptom, Receptor
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المؤلفون: Michael J. Cross, Steven D. Webb, Simeon Ramsey, Swaminathan Sethu, Wai Wong, Naif Alhumeed, Thilipan Thaventhiran, Han Xian Aw Yeang, Amy E. Chadwick, Richard Stebbings, Mohammad A. Aljasir, Laiche Djouhri, Ahmad F. Alghanem, Christina Ball, Jean G. Sathish
المصدر: Monoclonal Antibodies in Immunodiagnosis and Immunotherapy
مصطلحات موضوعية: CD4-Positive T-Lymphocytes, 0301 basic medicine, medicine.drug_class, T cell, Immunology, oxidative phosphorylation, Lymphocyte Activation, Monoclonal antibody, T-Lymphocytes, Regulatory, Article, 03 medical and health sciences, 0302 clinical medicine, Immune system, CD28 Antigens, Acetyl Coenzyme A, Neoplasms, Lipid biosynthesis, CD28 superagonist, Tumor Cells, Cultured, medicine, Humans, Immunology and Allergy, Glycolysis, lipogenesis, Cell Proliferation, 030102 biochemistry & molecular biology, biology, Chemistry, Effector, Lipogenesis, CD4+ effector memory T cells, Antibodies, Monoclonal, CD28, glycolysis, Cell biology, Glucose, medicine.anatomical_structure, 030220 oncology & carcinogenesis, biology.protein, Antibody, Immunologic Memory, Protein Kinases
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3ab47b16601b0af58fa2d2eace6aa33b
https://hdl.handle.net/10576/14207 -
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المؤلفون: Jennifer E, Davoren, Michelle, Garnsey, Betty, Pettersen, Michael A, Brodney, Jeremy R, Edgerton, Jean-Philippe, Fortin, Sarah, Grimwood, Anthony R, Harris, Stephen, Jenkinson, Terry, Kenakin, John T, Lazzaro, Che-Wah, Lee, Susan M, Lotarski, Lisa, Nottebaum, Steven V, O'Neil, Michael, Popiolek, Simeon, Ramsey, Stefanus J, Steyn, Catherine A, Thorn, Lei, Zhang, Damien, Webb
المصدر: Journal of medicinal chemistry. 60(15)
مصطلحات موضوعية: Diarrhea, Male, Lactams, Vomiting, Scopolamine, Isoindoles, Structure-Activity Relationship, Dogs, Allosteric Regulation, Piperidines, Seizures, Thiadiazoles, Animals, Humans, Donepezil, Rats, Wistar, Oxazoles, Sulfonamides, Receptor, Muscarinic M1, Mice, Inbred C57BL, Amphetamine, Drug Design, Indans, Microsomes, Liver, Ataxia, Female
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المؤلفون: Cara M. M. Williams, Bruce Allen Lefker, David C. Limburg, Stephen W. Wright, Julia Shin, Paul D. Bonin, Parag Sahasrabudhe, Simeon Ramsey, Jiang Wu, Kieran F. Geoghegan
المصدر: MedChemComm. 5:1871-1878
مصطلحات موضوعية: Pharmacology, Chemistry, Organic Chemistry, Pharmaceutical Science, Chemical probe, Drug action, Computational biology, Biochemistry, Combinatorial chemistry, law.invention, Bromodomain, law, Drug Discovery, Recombinant DNA, Molecular Medicine, Potency
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4f190a8af45764d22c2e32c175e6988a
https://doi.org/10.1039/c4md00259h -
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المؤلفون: Magnus Ivarsson, Magda Bictash, Nicholas Pullen, Lucy Bateman, Neil Attkins, Rachel Russell, Laura Weibley, Stevie Neal-Morgan, Jamie Turner, Rachel Doyle, Simeon Ramsey
المصدر: European Journal of Pharmacology. 670:347-355
مصطلحات موضوعية: Pharmacology, Agonist, Arginine vasopressin receptor 1B, medicine.medical_specialty, Vasopressin, medicine.drug_class, Chemistry, Receptor antagonist, Oxytocin receptor, Endocrinology, Arginine vasopressin receptor 2, Internal medicine, medicine, hormones, hormone substitutes, and hormone antagonists, Vasopressin Antagonists, Vasopressin receptor
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المؤلفون: Piet H. van der Graaf, Simeon Ramsey, Rebecca L. Fish, Neil Attkins
المصدر: British Journal of Pharmacology. 164:992-1007
مصطلحات موضوعية: Pharmacology, In vivo, Chemistry, Drug discovery, In vitro toxicology, Biophysics, Plasma protein binding, Ligand (biochemistry), Receptor, In vitro, Receptor–ligand kinetics
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المؤلفون: Gareth Jones, Jacques Richard, Simeon Ramsey, Rosalind Walley, Karl Richard Gibson, David C. Howe, Coralie S. Apfeldorfer, Natalie M. Mount, Amy N Brown, Nicholas Pullen, Tony Hawcock, Kirsty Bess, Alison McLeod, Peter M. Bungay, Sarah Tweedy
المصدر: Journal of Pharmacology and Experimental Therapeutics. 339:642-653
مصطلحات موضوعية: Adult, medicine.medical_specialty, Endometriosis, Biology, Pharmacology, Endometrium, Hormone antagonist, Translational Research, Biomedical, Young Adult, Hormone Antagonists, Double-Blind Method, Internal medicine, Follicular phase, Progesterone receptor, medicine, Animals, Humans, Estrogens, Non-Steroidal, Molecular Targeted Therapy, Sulfones, Receptor, Dose-Response Relationship, Drug, Estradiol, Antagonist, Mifepristone, Luteinizing Hormone, medicine.anatomical_structure, Endocrinology, Follicular Phase, Macaca, Pyrazoles, Molecular Medicine, Female, Receptors, Progesterone, Luteinizing hormone, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cf2424928f5d7c154555b10bc8fec040
https://doi.org/10.1124/jpet.111.183848 -
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المؤلفون: Rachel, Russell, Rachel, Doyle, Jamie, Turner, Neil, Attkins, Simeon, Ramsey, Laura, Weibley, Lucy, Bateman, Magda, Bictash, Stevie, Neal-Morgan, Magnus, Ivarsson, Nick, Pullen
المصدر: European journal of pharmacology. 670(2-3)
مصطلحات موضوعية: Male, Receptors, Vasopressin, Administration, Oral, CHO Cells, Triazoles, Models, Biological, Rats, Substrate Specificity, Arginine Vasopressin, Cricetulus, Dogs, Piperidines, Receptors, Oxytocin, Cricetinae, Blood Circulation, Myometrium, Animals, Humans, Female, Capsaicin, Antidiuretic Hormone Receptor Antagonists, Aorta