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1
المؤلفون: Nicolas Triballeau, Bertrand Heckmann, Nicolas Houvenaghel, Tanja Poljak, F. Marsais, Adeline Marie Elise Palisse, Emanuelle Wakselman, Mario Smehil, Mia Jans, Kathleen Sonck, Monica Borgonovi, Denis Bucher, Sandy El Bkassiny, Javier Blanc, Beatrice Coornaert, Thierry Christophe, Philippe Pujuguet, Vatroslav Letfus, M. Auberval, Lola Lecru, Laurent Saniere, Inge Duys, Reginald Brys, Line Oste, Brigitte Allart, Alex Jaunet, Maxim De Wachter, Catherine Jagerschmidt, Koen Karel Jansen, Oscar Mammoliti, Ludovic Waeckel, Giovanni Tricarico, Christel Jeanne Marie Menet, Renata Rupčić
المصدر: Journal of medicinal chemistry. 64(19)
مصطلحات موضوعية: Indole test, chemistry.chemical_classification, Benzimidazole, Carboxylic acid, Carboxylic Acids, Administration, Oral, Biological Availability, Transporter, Pharmacology, medicine.disease, In vitro, Idiopathic Pulmonary Fibrosis, chemistry.chemical_compound, Idiopathic pulmonary fibrosis, Disease Models, Animal, Mice, chemistry, Pharmacokinetics, In vivo, Drug Discovery, medicine, Molecular Medicine, Animals, Humans, Sphingosine-1-Phosphate Receptors
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2
المصدر: Bioorganicmedicinal chemistry. 28(1)
مصطلحات موضوعية: Jumonji Domain-Containing Histone Demethylases, Epigenetics, KDM4C enzyme, Inhibitor, Drug design, Computational chemistry, Clinical Biochemistry, Pharmaceutical Science, Pyrimidinones, 01 natural sciences, Biochemistry, Madin Darby Canine Kidney Cells, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Dogs, Drug Discovery, Animals, Humans, Viability assay, Epigenetics, Enzyme Inhibitors, Molecular Biology, ADME, chemistry.chemical_classification, Toxoflavin, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Triazines, Organic Chemistry, Rational design, Biological activity, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Enzyme, chemistry, A549 Cells, Drug Design, Microsomes, Liver, Molecular Medicine, Quantum Theory, Histone Demethylases
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3
المصدر: European journal of drug metabolism and pharmacokinetics. 37(3)
مصطلحات موضوعية: Male, Ketolides, Telithromycin, Erythromycin, Biological Availability, Pharmacology, Rats, Sprague-Dawley, First pass effect, Route of administration, Pharmacokinetics, Clarithromycin, polycyclic compounds, medicine, Animals, Pharmacology (medical), Roxithromycin, Chemistry, Bioavailability, Anti-Bacterial Agents, Rats, Hepatocytes, Microsomes, Liver, Macrolides, medicine.drug