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المؤلفون: Yan Weng, Kari R. Fonseca, Yi-an Bi, Sumathy Mathialagan, Keith Riccardi, Elaine Tseng, Andrew J. Bessire, Mathew A. Cerny, David A. Tess, A. David Rodrigues, Amit S. Kalgutkar, John Litchfield, Li Di, Manthena V. S. Varma
المصدر: Drug Metabolism and Disposition. 50:1312-1321
مصطلحات موضوعية: Pharmacology, Pharmaceutical Science
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ebf00f47e216d78cc961dc9e84ae92d0
https://doi.org/10.1124/dmd.122.000953 -
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المؤلفون: Andrew J, Bessire, Chakrapani, Subramanyam
المصدر: Methods in molecular biology (Clifton, N.J.). 2078
مصطلحات موضوعية: Immunoconjugates, Humans, Hydrogen-Ion Concentration, Lysosomes, Mass Spectrometry, Chromatography, Liquid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::f2fc14354f0d76e6fac4a6c0dcb1169b
https://pubmed.ncbi.nlm.nih.gov/31643069 -
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المؤلفون: Chakrapani Subramanyam, Andrew J. Bessire
المصدر: Methods in Molecular Biology ISBN: 9781493999286
مصطلحات موضوعية: Cathepsin, chemistry.chemical_classification, 0303 health sciences, General method, Catabolism, 030226 pharmacology & pharmacy, In vitro, body regions, 03 medical and health sciences, 0302 clinical medicine, Enzyme, Biochemistry, chemistry, Liquid chromatography–mass spectrometry, 030304 developmental biology, Conjugate
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::bf0c6ba753d6127332cd4ab86d5473e3
https://doi.org/10.1007/978-1-4939-9929-3_24 -
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المؤلفون: Judy Lucas, Guoyun Bai, Christopher J. O’Donnell, Sai Chetan K. Sukuru, Brian Rago, Sarah P. Hudson, Carolyn A. Leverett, Lioudmila Tchistiakova, Edmund I. Graziani, Anokha S. Ratnayake, Sylvia Musto, Jeffrey M. Casavant, Joseph Stock, Frank Loganzo, Christine Hosselet, Sujiet Puthenveetil, Andrew J. Bessire, Fengping Li, Xiaogang Han, Tracey Clark, Venkata Doppalapudi, Kimberly Ann Marquette, Beth C. Vetelino, Chakrapani Subramanyam, L. Nathan Tumey
المصدر: ACS Medicinal Chemistry Letters. 7:977-982
مصطلحات موضوعية: 0301 basic medicine, Drug, Heavy chain, biology, Chemistry, media_common.quotation_subject, Organic Chemistry, Metabolism, Biochemistry, body regions, 03 medical and health sciences, 030104 developmental biology, Drug Discovery, biology.protein, Antibody, media_common, Conjugate
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المؤلفون: Alfin D. N. Vaz, T. Eric Ballard, Upendra P. Dahal, Andrew J. Bessire, Kieran F. Geoghegan, Richard P. Schneider
المصدر: Rapid Communications in Mass Spectrometry. 29:2175-2183
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Mass spectrometry, Combinatorial chemistry, Small molecule, Dissociation (chemistry), Analytical Chemistry, Adduct, Ion, Fragmentation (mass spectrometry), Molecule, Spectroscopy, Macromolecule
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المؤلفون: Edmund I. Graziani, Xiaotian Zhong, Chethana Kulkarni, Andrew J. Bessire, James E. Finley, Sylvia Musto
المصدر: Bioconjugate chemistry. 28(4)
مصطلحات موضوعية: 0301 basic medicine, Drug, Azides, Fluorophore, Immunoconjugates, Stereochemistry, media_common.quotation_subject, Biomedical Engineering, Pharmaceutical Science, Bioengineering, 010402 general chemistry, Antibodies, Monoclonal, Humanized, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Molecular level, Cell Line, Tumor, Humans, media_common, Fluorescent Dyes, Pyrans, Pharmacology, Microscopy, Confocal, biology, Chemistry, Organic Chemistry, Biological Transport, 0104 chemical sciences, body regions, 030104 developmental biology, Transcytosis, Pharmaceutical Preparations, biology.protein, Biophysics, Click chemistry, Click Chemistry, Azide, Antibody, Biotechnology, Conjugate
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المؤلفون: Frank Loganzo, Klaas Schildknegt, Sujiet Puthenveetil, Birte Nolting, Andrew J. Bessire, T. Eric Ballard, Lee R. Roberts, My-Hanh Lam, Chakrapani Subramanyam, Michael Eric Green, Betsy Pierce, Manoj Charati, Justin Cohen
المصدر: Bioconjugate chemistry. 27(7)
مصطلحات موضوعية: 0301 basic medicine, Antibody-drug conjugate, Immunoconjugates, Biomedical Engineering, Pharmaceutical Science, Bioengineering, Nanotechnology, Mass Spectrometry, Cathepsin B, 03 medical and health sciences, Mice, 0302 clinical medicine, Cell Line, Tumor, Animals, Humans, Pharmacology, chemistry.chemical_classification, Drug Carriers, Organic Chemistry, In vitro toxicology, In vitro, Rats, Drug Liberation, 030104 developmental biology, Enzyme, chemistry, S9 fraction, Biochemistry, Targeted drug delivery, Liver, 030220 oncology & carcinogenesis, Lysosomes, Linker, Biotechnology, Conjugate
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المؤلفون: Kay Ahn, Steven J. Conrad, Alison H. Varghese, Roger B. Ruggeri, Felix Vajdos, Andrew J. Bessire, Philip A. Carpino, Xidong Feng, James J. Conboy, Samantha N. Spath, Sergey V. Filippov, Cristiano Ruch Werneck Guimarães, Kieran F. Geoghegan
المصدر: Biochemistry. 51:2065-2077
مصطلحات موضوعية: Models, Molecular, Protein mass spectrometry, Neutrophils, Molecular Sequence Data, Heme, Crystallography, X-Ray, Mass spectrometry, Tandem mass spectrometry, Orbitrap, Peptide Mapping, Biochemistry, Sample preparation in mass spectrometry, law.invention, chemistry.chemical_compound, Tandem Mass Spectrometry, law, Catalytic Domain, Humans, Amino Acid Sequence, Peroxidase, Chromatography, biology, Peptide Fragments, Molecular Weight, Models, Chemical, chemistry, Myeloperoxidase, biology.protein, Ion trap, Oxidation-Reduction, Chromatography, Liquid
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المؤلفون: Alfin D. N. Vaz, Hao Sun, Andrew J. Bessire
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:371-376
مصطلحات موضوعية: Models, Molecular, Drug, Conformational change, Indoles, Protein Conformation, Stereochemistry, Chemistry, Pharmaceutical, media_common.quotation_subject, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Crystallography, X-Ray, Ligands, Biochemistry, Catalysis, Mass Spectrometry, Computational chemistry, Catalytic Domain, Drug Discovery, Cytochrome P-450 CYP3A, Computer Simulation, Molecular Biology, media_common, Computational model, biology, Chemistry, Organic Chemistry, Temperature, Active site, Template, Models, Chemical, Docking (molecular), Drug Design, Microsomes, Liver, biology.protein, Molecular Medicine, Structure based, Carbamates, Crystallization
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المؤلفون: Weiwei Wang, Raman Sharma, Anne E. Hagen, Alfin D. N. Vaz, Andrew J. Bessire
المصدر: Rapid Communications in Mass Spectrometry. 24:2109-2121
مصطلحات موضوعية: Reaction conditions, chemistry.chemical_classification, Chromatography, Hydroxamic acid, Organic Chemistry, Mass spectrometry, Analytical Chemistry, chemistry.chemical_compound, Hydroxylamine, chemistry, Organic chemistry, lipids (amino acids, peptides, and proteins), Derivatization, Spectroscopy, Derivative (chemistry), Alkyl