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1دورية أكاديمية
المؤلفون: Lentzas A; Division of Pharmacology, The Netherlands Cancer Institute, Room H3.010, Plesmanlaan 121, Amsterdam, 1066 CX, The Netherlands., de Gooijer MC; Division of Pharmacology, The Netherlands Cancer Institute, Room H3.010, Plesmanlaan 121, Amsterdam, 1066 CX, The Netherlands.; Faculty of Biology, Medicine and Health, University of Manchester, Manchester, M1 3WE, UK.; The Christie NHS Foundation Trust, Manchester, M20 4BX, UK., Zuidema S; Division of Pharmacology, The Netherlands Cancer Institute, Room H3.010, Plesmanlaan 121, Amsterdam, 1066 CX, The Netherlands., Meurs A; Division of Pharmacology, The Netherlands Cancer Institute, Room H3.010, Plesmanlaan 121, Amsterdam, 1066 CX, The Netherlands., Çitirikkaya CH; Division of Pharmacology, The Netherlands Cancer Institute, Room H3.010, Plesmanlaan 121, Amsterdam, 1066 CX, The Netherlands., Venekamp N; Division of Pharmacology, The Netherlands Cancer Institute, Room H3.010, Plesmanlaan 121, Amsterdam, 1066 CX, The Netherlands.; Department of Pharmacy, The Netherlands Cancer Institute, Amsterdam, The Netherlands., Beijnen JH; Department of Pharmacy, The Netherlands Cancer Institute, Amsterdam, The Netherlands.; Division of Pharmacoepidemiology and Clinical Pharmacology, Department of Pharmaceutical Sciences, Faculty of Science, Utrecht University, Universiteitsweg 99, Utrecht, 3584 CG, The Netherlands., van Tellingen O; Division of Pharmacology, The Netherlands Cancer Institute, Room H3.010, Plesmanlaan 121, Amsterdam, 1066 CX, The Netherlands. o.v.tellingen@nki.nl.; Mouse Cancer Clinic, The Netherlands Cancer Institute, Amsterdam, The Netherlands. o.v.tellingen@nki.nl.
المصدر: Fluids and barriers of the CNS [Fluids Barriers CNS] 2024 Aug 05; Vol. 21 (1), pp. 62. Date of Electronic Publication: 2024 Aug 05.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Biomed Central Country of Publication: England NLM ID: 101553157 Publication Model: Electronic Cited Medium: Internet ISSN: 2045-8118 (Electronic) Linking ISSN: 20458118 NLM ISO Abbreviation: Fluids Barriers CNS Subsets: MEDLINE
مواضيع طبية MeSH: Mice, Knockout* , Tetrahydroisoquinolines*/pharmacology , Tetrahydroisoquinolines*/administration & dosage , ATP Binding Cassette Transporter, Subfamily G, Member 2*/metabolism , ATP Binding Cassette Transporter, Subfamily G, Member 2*/antagonists & inhibitors , Brain*/metabolism , Brain*/drug effects , Acridines*/pharmacology , Acridines*/administration & dosage , Blood-Brain Barrier*/metabolism , Blood-Brain Barrier*/drug effects, Animals ; Mice ; Quinolines/pharmacology ; Quinolines/pharmacokinetics ; Quinolines/administration & dosage ; Drug Delivery Systems/methods ; ATP Binding Cassette Transporter, Subfamily B/metabolism ; ATP Binding Cassette Transporter, Subfamily B/antagonists & inhibitors ; ATP Binding Cassette Transporter, Subfamily B/genetics ; Male ; Mice, Inbred C57BL
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2دورية أكاديمية
المؤلفون: El-Khouly ME; Nanoscience Program, Institute of Basic and Applied Sciences, Egypt-Japan University of Science and Technology (E-JUST), New Borg El-Arab City, Alexandria, Egypt. mohamed.elkhouly@ejust.edu.eg., Khatab HA; Pharm D Program, Egypt-Japan University of Science and Technology (E-JUST), New Borg El-Arab City, Alexandria, Egypt., Abdel-Shafi AA; Department of Chemistry, Faculty of Science, Ain Shams University, 11566 Abbassia, Cairo, Egypt., Hammad SF; Pharm D Program, Egypt-Japan University of Science and Technology (E-JUST), New Borg El-Arab City, Alexandria, Egypt.
المصدر: Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology [Photochem Photobiol Sci] 2024 Aug; Vol. 23 (8), pp. 1445-1455. Date of Electronic Publication: 2024 Jun 27.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Springer Country of Publication: England NLM ID: 101124451 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1474-9092 (Electronic) Linking ISSN: 1474905X NLM ISO Abbreviation: Photochem Photobiol Sci Subsets: MEDLINE
مواضيع طبية MeSH: Phthalimides*/chemistry , Phthalimides*/chemical synthesis , Singlet Oxygen*/chemistry , Singlet Oxygen*/metabolism , Photochemotherapy* , Photosensitizing Agents*/chemistry , Photosensitizing Agents*/pharmacology , Photosensitizing Agents*/chemical synthesis , Acridines*/chemistry , Acridines*/pharmacology , Acridines*/chemical synthesis, Electron Transport ; Humans ; Density Functional Theory ; Molecular Structure
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3دورية أكاديمية
المؤلفون: Asadi M; Razi Drug Research Center, Iran University of Medical Sciences, Tehran, Islamic Republic of Iran.; Department of Medicinal Chemistry, School of Pharmacy, Iran University of Medical Sciences, Tehran, Islamic Republic of Iran., Ahangari MM; Department of Medicinal Chemistry, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran., Iraji A; Stem Cells Technology Research Center, Shiraz University of Medical Sciences, Shiraz, Islamic Republic of Iran.; Central Research Laboratory, Shiraz University of Medical Sciences, Shiraz, Islamic Republic of Iran., Azizian H; Razi Drug Research Center, Iran University of Medical Sciences, Tehran, Islamic Republic of Iran.; Department of Medicinal Chemistry, School of Pharmacy, Iran University of Medical Sciences, Tehran, Islamic Republic of Iran., Nokhbehzaim A; Department of Medicinal Chemistry, Faculty of Pharmacy, Alborz University of Medical Sciences, Karaj, Islamic Republic of Iran., Bahadorikhalili S; Department of Electronic Engineering, Universitat Rovira I Virgili, 43007, Tarragona, Spain., Mojtabavi S; Department of Pharmaceutical Biotechnology, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran., Faramarzi MA; Department of Pharmaceutical Biotechnology, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran., Nasli-Esfahani E; Diabetes Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran., Larijani B; Endocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran., Mahdavi M; Endocrinology and Metabolism Research Center, Endocrinology and Metabolism Clinical Sciences Institute, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran. Mahdavi_chem@yahoo.com., Amanlou M; Department of Medicinal Chemistry, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran. amanlou@tums.ac.ir.; Experimental Medicine Research Center, Tehran University of Medical Sciences, Tehran, Islamic Republic of Iran. amanlou@tums.ac.ir.
المصدر: Scientific reports [Sci Rep] 2024 Jul 28; Vol. 14 (1), pp. 17338. Date of Electronic Publication: 2024 Jul 28.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN: 2045-2322 (Electronic) Linking ISSN: 20452322 NLM ISO Abbreviation: Sci Rep Subsets: MEDLINE
مواضيع طبية MeSH: Glycoside Hydrolase Inhibitors*/pharmacology , Glycoside Hydrolase Inhibitors*/chemistry , Glycoside Hydrolase Inhibitors*/chemical synthesis , Triazoles*/chemistry , Triazoles*/pharmacology , Triazoles*/chemical synthesis , Molecular Dynamics Simulation* , alpha-Glucosidases*/metabolism , alpha-Glucosidases*/chemistry , Acridines*/chemistry , Acridines*/pharmacology , Acridines*/chemical synthesis, Kinetics ; Molecular Docking Simulation ; Structure-Activity Relationship ; Humans
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4دورية أكاديمية
المؤلفون: Garberová M; Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University, Moyzesova 11, 040 01 Košice, Slovakia., Kudličková Z; Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University, Moyzesova 11, 040 01 Košice, Slovakia., Michalková R; Department of Pharmacology, Faculty of Medicine, Pavol Jozef Šafárik University, Trieda SNP 1, 040 01 Košice, Slovakia., Tvrdoňová M; Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University, Moyzesova 11, 040 01 Košice, Slovakia., Sabolová D; Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University, Moyzesova 11, 040 01 Košice, Slovakia., Bekešová S; Thermo Fisher Scientific, Mlynské Nivy 5, 821 09 Bratislava, Slovakia., Gramblička M; Thermo Fisher Scientific, Mlynské Nivy 5, 821 09 Bratislava, Slovakia., Mojžiš J; Department of Pharmacology, Faculty of Medicine, Pavol Jozef Šafárik University, Trieda SNP 1, 040 01 Košice, Slovakia., Vilková M; Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University, Moyzesova 11, 040 01 Košice, Slovakia.
المصدر: Molecules (Basel, Switzerland) [Molecules] 2024 Jul 18; Vol. 29 (14). Date of Electronic Publication: 2024 Jul 18.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents*/pharmacology , Antineoplastic Agents*/chemical synthesis , Antineoplastic Agents*/chemistry , Thiazolidinediones*/chemistry , Thiazolidinediones*/pharmacology , Thiazolidinediones*/chemical synthesis , Acridines*/chemistry , Acridines*/pharmacology , Acridines*/chemical synthesis , Drug Design*, Humans ; Cell Line, Tumor ; Structure-Activity Relationship ; Cell Proliferation/drug effects ; Drug Screening Assays, Antitumor ; Molecular Structure
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5دورية أكاديمية
المؤلفون: Wang J; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou University City, Guangzhou, PR China., Wang S; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou University City, Guangzhou, PR China., Zhang J; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou University City, Guangzhou, PR China., Ji D; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou University City, Guangzhou, PR China., Huang ZS; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou University City, Guangzhou, PR China., Li D; School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou University City, Guangzhou, PR China. Electronic address: liding@mail.sysu.edu.cn.
المصدر: Biochimica et biophysica acta. General subjects [Biochim Biophys Acta Gen Subj] 2024 Jul; Vol. 1868 (7), pp. 130631. Date of Electronic Publication: 2024 Apr 27.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 101731726 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-8006 (Electronic) Linking ISSN: 03044165 NLM ISO Abbreviation: Biochim Biophys Acta Gen Subj Subsets: MEDLINE
مواضيع طبية MeSH: Promoter Regions, Genetic*/drug effects , Vascular Endothelial Growth Factor A*/genetics , Vascular Endothelial Growth Factor A*/metabolism , Gene Expression Regulation, Neoplastic*/drug effects , Acridines*/pharmacology , Acridines*/chemistry, Humans ; Animals ; Mice ; Cell Proliferation/drug effects ; Xenograft Model Antitumor Assays ; Neoplasms/drug therapy ; Neoplasms/genetics ; Neoplasms/pathology ; Neoplasms/metabolism ; MCF-7 Cells ; Mice, Nude ; Cell Line, Tumor ; Apoptosis/drug effects ; Female ; Antineoplastic Agents/pharmacology ; Antineoplastic Agents/chemistry
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6دورية أكاديمية
المؤلفون: Jian M; National Key Laboratory of High-efficiency Utilization of Coal and Green Chemical Engineering, Ningxia University, Yinchuan, 750021, PR China; Ningxia Academy of Metrology & Quality Inspection, Yinchuan, 750200, PR China., Xue P; National Key Laboratory of High-efficiency Utilization of Coal and Green Chemical Engineering, Ningxia University, Yinchuan, 750021, PR China. Electronic address: ping@nxu.edu.cn., Zhang X; Ningxia Academy of Metrology & Quality Inspection, Yinchuan, 750200, PR China., Xing Y; Ningxia Academy of Metrology & Quality Inspection, Yinchuan, 750200, PR China., Ma L; National Key Laboratory of High-efficiency Utilization of Coal and Green Chemical Engineering, Ningxia University, Yinchuan, 750021, PR China., Lv X; Ningxia Academy of Metrology & Quality Inspection, Yinchuan, 750200, PR China., Shi K; National Key Laboratory of High-efficiency Utilization of Coal and Green Chemical Engineering, Ningxia University, Yinchuan, 750021, PR China.
المصدر: Chemosphere [Chemosphere] 2024 Aug; Vol. 362, pp. 141752. Date of Electronic Publication: 2024 Mar 18.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 0320657 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1879-1298 (Electronic) Linking ISSN: 00456535 NLM ISO Abbreviation: Chemosphere Subsets: MEDLINE
مواضيع طبية MeSH: Bioelectric Energy Sources* , Electrodes* , Wastewater*/chemistry , Acridines*/chemistry , Aniline Compounds*/chemistry, Waste Disposal, Fluid/methods ; Carbon/chemistry ; Electricity ; Graphite ; Nitrogen Compounds
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7دورية أكاديمية
المؤلفون: de Oliveira Viana J; Bioinformatics Multidisciplinary Environment, Federal University of Rio Grande do Norte, University Campus I-Lagoa Nova, Natal, RN, 59078-970., Sena Mendes M; Department of Pharmacy, Federal University of Bahia, University Campus Ondina - Ondina, Salvador, BA, 40170-110., Santos Castilho M; Department of Pharmacy, Federal University of Bahia, University Campus Ondina - Ondina, Salvador, BA, 40170-110., Olímpio de Moura R; Department of Pharmacy, State University of Paraíba, University Campus I - Universitário, Campina, Grande - PB, 58429-500., Guimarães Barbosa E; Bioinformatics Multidisciplinary Environment, Federal University of Rio Grande do Norte, University Campus I-Lagoa Nova, Natal, RN, 59078-970.; Department of Pharmacy, Federal University of Rio Grande do Norte, University Campus I - Petrópolis, Natal, RN, 59012-570.
المصدر: ChemMedChem [ChemMedChem] 2024 Jun 03; Vol. 19 (11), pp. e202300545. Date of Electronic Publication: 2024 Mar 25.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE
مواضيع طبية MeSH: Oxidoreductases*/antagonists & inhibitors , Oxidoreductases*/metabolism , Acridines*/chemistry , Acridines*/pharmacology , Acridines*/chemical synthesis , Enzyme Inhibitors*/pharmacology , Enzyme Inhibitors*/chemistry , Enzyme Inhibitors*/chemical synthesis, Antiprotozoal Agents/pharmacology ; Antiprotozoal Agents/chemistry ; Antiprotozoal Agents/chemical synthesis ; Molecular Dynamics Simulation ; Spiro Compounds/chemistry ; Spiro Compounds/pharmacology ; Spiro Compounds/chemical synthesis ; Structure-Activity Relationship ; Molecular Structure ; Parasitic Sensitivity Tests ; Dose-Response Relationship, Drug ; Leishmania/drug effects ; Leishmania/enzymology ; Molecular Docking Simulation
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8دورية أكاديمية
المؤلفون: Smith K; School of Chemistry, Cardiff University, Main Building, Park Place, Cardiff, CF10 3AT, United Kingdom.; Chemistry Department, University of Wales Swansea, Singleton Park, Swansea, SA2 8PP, United Kingdom., Holland AM; Chemistry Department, University of Wales Swansea, Singleton Park, Swansea, SA2 8PP, United Kingdom., Woodhead JS; Invitron, Monmouth, United Kingdom., El-Hiti GA; Department of Optometry, College of Applied Medical Sciences, King Saud University, Riyadh, Saudi Arabia.
المصدر: Luminescence : the journal of biological and chemical luminescence [Luminescence] 2024 Jun; Vol. 39 (6), pp. e4794.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Wiley & Sons Country of Publication: England NLM ID: 100889025 Publication Model: Print Cited Medium: Internet ISSN: 1522-7243 (Electronic) Linking ISSN: 15227235 NLM ISO Abbreviation: Luminescence Subsets: MEDLINE
مواضيع طبية MeSH: Acridines*/chemistry , Acridines*/chemical synthesis , Mesylates*/chemistry , Luminescence*, Molecular Structure ; Luminescent Measurements
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9دورية أكاديمية
المؤلفون: Roy R; School of Mathematical and Physical Sciences, Faculty of Science, University of Technology Sydney, Sydney, NSW, 2007, Australia., Chick P; School of Mathematical and Physical Sciences, Faculty of Science, University of Technology Sydney, Sydney, NSW, 2007, Australia., York E; School of Mathematical and Physical Sciences, Faculty of Science, University of Technology Sydney, Sydney, NSW, 2007, Australia., Rawling T; School of Mathematical and Physical Sciences, Faculty of Science, University of Technology Sydney, Sydney, NSW, 2007, Australia. Electronic address: Tristan.Rawling@uts.edu.au.
المصدر: Chemico-biological interactions [Chem Biol Interact] 2024 Jun 01; Vol. 396, pp. 111042. Date of Electronic Publication: 2024 May 10.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Elsevier Country of Publication: Ireland NLM ID: 0227276 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-7786 (Electronic) Linking ISSN: 00092797 NLM ISO Abbreviation: Chem Biol Interact Subsets: MEDLINE
مواضيع طبية MeSH: Ionic Liquids*/chemistry , Ionic Liquids*/pharmacology , Acridines*/chemistry , Acridines*/pharmacology , Reactive Oxygen Species*/metabolism, Humans ; Structure-Activity Relationship ; Cell Line, Tumor ; Cell Survival/drug effects ; Antineoplastic Agents/pharmacology ; Antineoplastic Agents/chemistry ; Oxidative Phosphorylation/drug effects
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10دورية أكاديمية
المؤلفون: Krochtová K; Department of Biochemistry, Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University in Košice, Šrobárova 2, 041 54, Košice, Slovak Republic., Janovec L; Department of Organic Chemistry, Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University in Košice, Šrobárova 2, 041 54, Košice, Slovak Republic., Bogárová V; Department of Biochemistry, Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University in Košice, Šrobárova 2, 041 54, Košice, Slovak Republic., Halečková A; Department of Organic Chemistry, Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University in Košice, Šrobárova 2, 041 54, Košice, Slovak Republic., Kožurková M; Department of Biochemistry, Institute of Chemistry, Faculty of Science, Pavol Jozef Šafárik University in Košice, Šrobárova 2, 041 54, Košice, Slovak Republic. Electronic address: maria.kozurkova@upjs.sk.
المصدر: Chemico-biological interactions [Chem Biol Interact] 2024 May 01; Vol. 394, pp. 110965. Date of Electronic Publication: 2024 Mar 27.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Elsevier Country of Publication: Ireland NLM ID: 0227276 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-7786 (Electronic) Linking ISSN: 00092797 NLM ISO Abbreviation: Chem Biol Interact Subsets: MEDLINE
مواضيع طبية MeSH: Acridines*/chemistry , Acridines*/metabolism , Molecular Docking Simulation* , Poly A*/chemistry , Poly A*/metabolism , Circular Dichroism*, Thermodynamics ; Spectrometry, Fluorescence ; RNA/chemistry ; RNA/metabolism ; Nucleic Acid Conformation