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1دورية أكاديمية
المؤلفون: Yibing Shan, Venkatesh P. Mysore, Abba E. Leffler, Eric T. Kim, Shiori Sagawa, David E. Shaw
المصدر: PLoS Computational Biology, Vol 18, Iss 3 (2022)
مصطلحات موضوعية: Biology (General), QH301-705.5
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Dana Katz, Michael A. DiMattia, Dan Sindhikara, Hubert Li, Nikita Abraham, Abba E. Leffler
المصدر: Marine Drugs, Vol 19, Iss 7, p 367 (2021)
مصطلحات موضوعية: conotoxin, nicotinic acetylcholine receptor, selectivity, free-energy perturbation, Biology (General), QH301-705.5
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Dana Katz, Dan Sindhikara, Michael DiMattia, Abba E. Leffler
المصدر: Toxins, Vol 13, Iss 3, p 193 (2021)
مصطلحات موضوعية: gating-modifier toxin, free-energy perturbation, sodium channel, drug discovery, Medicine
وصف الملف: electronic resource
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4دورية أكاديمية
المؤلفون: Binita Shah, Dan Sindhikara, Ken Borrelli, Abba E. Leffler
المصدر: Toxins, Vol 12, Iss 10, p 652 (2020)
مصطلحات موضوعية: peptide toxin, ion channel, WaterMap, cryo-EM, drug discovery, Medicine
وصف الملف: electronic resource
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5
المؤلفون: Pieter H. Bos, Evelyne M. Houang, Fabio Ranalli, Abba E. Leffler, Nicholas A. Boyles, Volker A. Eyrich, Yuval Luria, Dana Katz, Haifeng Tang, Robert Abel, Sathesh Bhat
المصدر: Journal of Chemical Information and Modeling. 62:1905-1915
مصطلحات موضوعية: General Chemical Engineering, General Chemistry, Library and Information Sciences, Computer Science Applications
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6
المؤلفون: Pieter H, Bos, Evelyne M, Houang, Fabio, Ranalli, Abba E, Leffler, Nicholas A, Boyles, Volker A, Eyrich, Yuval, Luria, Dana, Katz, Haifeng, Tang, Robert, Abel, Sathesh, Bhat
المصدر: Journal of chemical information and modeling. 62(8)
مصطلحات موضوعية: Central Nervous System, Drug Design, Drug Discovery, Amino Acids, Algorithms
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7
المؤلفون: Pieter H Bos, Evelyne M. Houang, Fabio Ranalli, Abba E. Leffler, Nicholas A. Boyles, Volker A. Eyrich, Yuval Luria, Dana Katz, Haifeng Tang, Robert Abel, Sathesh Bhat
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::88c2ba821dcd166570c44c7439ae5d47
https://doi.org/10.26434/chemrxiv-2021-m6k5f -
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المؤلفون: Venkat Mysore, Yibing Shan, David E. Shaw, Kim Et, Abba E. Leffler, Shiori Sagawa
مصطلحات موضوعية: Free energy perturbation, Chemistry, Drug discovery, Biophysics, Rational design, Molecule, Binding site, Ligand (biochemistry), Small molecule, Function (biology)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::548996e088ac2a74a60288ac58b3d500
https://doi.org/10.1101/2021.03.31.437917 -
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المؤلفون: Abba E. Leffler, Jingyi Wang, Theodore M. Kamenecka, Alexander Kuryatov, Jon Lindstrom, Christelle Doebelin, Jack Norleans
المصدر: J Biol Chem
مصطلحات موضوعية: 0301 basic medicine, Agonist, Allosteric modulator, Patch-Clamp Techniques, medicine.drug_class, Allosteric regulation, Thiophenes, Receptors, Nicotinic, Biochemistry, 03 medical and health sciences, Xenopus laevis, Allosteric Regulation, Piperidines, medicine, Animals, Humans, Amino Acid Sequence, Nicotinic Agonists, Binding site, Molecular Biology, Binding Sites, 030102 biochemistry & molecular biology, Chemistry, Long-term potentiation, Cell Biology, Recombinant Proteins, Cell biology, Protein Structure, Tertiary, Molecular Docking Simulation, Transmembrane domain, Nicotinic acetylcholine receptor, Kinetics, Protein Subunits, 030104 developmental biology, Docking (molecular), Mutagenesis, Site-Directed, Oocytes, Sequence Alignment, Molecular Biophysics
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f8e8f4a8f34afa413d37f28e4a3bba33
https://pubmed.ncbi.nlm.nih.gov/31221718 -
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المؤلفون: Daniel J. Sindhikara, Dana Katz, Michael A. DiMattia, Abba E. Leffler
المصدر: Toxins
Volume 13
Issue 3
Toxins, Vol 13, Iss 193, p 193 (2021)مصطلحات موضوعية: free-energy perturbation, 0303 health sciences, Health, Toxicology and Mutagenesis, In silico, Sodium channel, lcsh:R, lcsh:Medicine, Gating, Toxicology, drug discovery, Free energy perturbation, 03 medical and health sciences, 0302 clinical medicine, Membrane, Computational chemistry, gating-modifier toxin, Mole, Potency, Molecule, 030217 neurology & neurosurgery, sodium channel, 030304 developmental biology
وصف الملف: application/pdf