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1دورية أكاديمية
المؤلفون: Snježana Čužić, Maja Antolić, Anja Ognjenović, Darija Stupin-Polančec, Adriana Petrinić Grba, Boška Hrvačić, Miroslava Dominis Kramarić, Sanja Musladin, Lidija Požgaj, Ivo Zlatar, Denis Polančec, Gorana Aralica, Marko Banić, Marija Urek, Brankica Mijandrušić Sinčić, Aleksandar Čubranić, Ines Glojnarić, Martina Bosnar, Vesna Eraković Haber
المصدر: Frontiers in Pharmacology, Vol 12 (2021)
مصطلحات موضوعية: claudins, inflammatory bowel disease, dextran sodium sulfate colitis model, adoptive transfer colitis model, ulcerative colitis, Crohn’s disease, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2
المؤلفون: Ivaylo Jivkov Elenkov, Simon Feldbaek Nielsen, Kristina Butković, Sanja Koštrun, Dijana Pesic, Dack Kevin Neil, Tine Skak-Nielsen, Dinko Žiher, Martin Stahlhut, Adriana Petrinić Grba, Vlatka Bencetić Mihaljević, Ana Čikoš, Samra Kapić, Andrea Fajdetić, Renata Rupčić, Gordon Saxty, Maja Lambert, Jasna Padovan, Ivana Ozimec Landek, Karmen Brajša, Dubravko Jelić, Haakan Bladh, Ana Grgičević
المصدر: Journal of Medicinal Chemistry. 64:8354-8383
مصطلحات موضوعية: Male, Macrocyclic Compounds, THP-1 Cells, Anti-Inflammatory Agents, 01 natural sciences, Inflammatory bowel disease, Mice, Structure-Activity Relationship, 03 medical and health sciences, Immune system, In vivo, Psoriasis, Drug Discovery, medicine, Animals, Humans, 030304 developmental biology, ADME, 0303 health sciences, Receptors, Interleukin-17, Molecular Structure, Chemistry, Drug discovery, Interleukin-17, medicine.disease, 0104 chemical sciences, Molecular Docking Simulation, proteins, macrocycles, IL 17AM, Il 17RA, chemical structure inhibitors, 010404 medicinal & biomolecular chemistry, Rheumatoid arthritis, Immunology, Molecular Medicine, Interleukin 17, Protein Binding
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3
المصدر: Bioorganicmedicinal chemistry. 28(1)
مصطلحات موضوعية: Jumonji Domain-Containing Histone Demethylases, Epigenetics, KDM4C enzyme, Inhibitor, Drug design, Computational chemistry, Clinical Biochemistry, Pharmaceutical Science, Pyrimidinones, 01 natural sciences, Biochemistry, Madin Darby Canine Kidney Cells, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Dogs, Drug Discovery, Animals, Humans, Viability assay, Epigenetics, Enzyme Inhibitors, Molecular Biology, ADME, chemistry.chemical_classification, Toxoflavin, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Triazines, Organic Chemistry, Rational design, Biological activity, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Enzyme, chemistry, A549 Cells, Drug Design, Microsomes, Liver, Molecular Medicine, Quantum Theory, Histone Demethylases