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1دورية أكاديمية
المؤلفون: Jelena Konstantinović, Andreas M. Kany, Alaa Alhayek, Ahmed S. Abdelsamie, Asfandyar Sikandar, Katrin Voos, Yiwen Yao, Anastasia Andreas, Roya Shafiei, Brigitta Loretz, Esther Schönauer, Robert Bals, Hans Brandstetter, Rolf W. Hartmann, Christian Ducho, Claus-Michael Lehr, Christoph Beisswenger, Rolf Müller, Katharina Rox, Jörg Haupenthal, Anna K.H. Hirsch
المصدر: ACS Central Science, Vol 9, Iss 12, Pp 2205-2215 (2023)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2374-7951
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المؤلفون: Reham A. Mohamed-Ezzat, Mohamed A. Omar, Ahmed Temirak, Ahmed S. Abdelsamie, Marwa M. Abdel-Aziz, Shadia A. Galal, galal elgemeie, Hoda I. El Diwani, Keith J. Flanagan, Mathias O. Senge
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ef70908f8b2acc332bf80588689259fa
https://doi.org/10.2139/ssrn.4446503 -
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المؤلفون: Alaa Alhayek, Ahmed S. Abdelsamie, Esther Schönauer, Virgyl Camberlein, Evelyn Hutterer, Gernot Posselt, Jamil Serwanja, Constantin Blöchl, Christian G. Huber, Jörg Haupenthal, Hans Brandstetter, Silja Wessler, Anna K. H. Hirsch
المصدر: Journal of medicinal chemistry. 65(19)
مصطلحات موضوعية: Microbial Collagenase, Diphosphonates, Drug Discovery, Molecular Medicine, Collagenases, Matrix Metalloproteinase Inhibitors, Clostridium histolyticum
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المؤلفون: Abdelrahman Mohamed, Mohamed Salah, Mariam Tahoun, Manuel Hawner, Ahmed S. Abdelsamie, Martin Frotscher
المصدر: Journal of medicinal chemistry. 65(17)
مصطلحات موضوعية: Structure-Activity Relationship, 17-Hydroxysteroid Dehydrogenases, Phenols, Drug Discovery, Endometriosis, Molecular Medicine, Humans, Female, Prodrugs, Steryl-Sulfatase, Enzyme Inhibitors
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المؤلفون: Mostafa M. Hamed, Ahmed S. Abdelsamie, Katharina Rox, Christian Schütz, Andreas M. Kany, Teresa Röhrig, Stefan Schmelz, Wulf Blankenfeldt, Alejandro Arce‐Rodriguez, José Manuel Borrero‐de Acuña, Dieter Jahn, Jessica Rademacher, Felix C. Ringshausen, Nina Cramer, Burkhard Tümmler, Anna K. H. Hirsch, Rolf W. Hartmann, Martin Empting
المصدر: Advanced Science. 10:2370027
مصطلحات موضوعية: General Chemical Engineering, General Engineering, General Physics and Astronomy, Medicine (miscellaneous), General Materials Science, Biochemistry, Genetics and Molecular Biology (miscellaneous)
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المؤلفون: Rolf W. Hartmann, Chris J. van Koppen, Matthias W. Laschke, Giuseppe Felice Mangiatordi, Ahmed S. Abdelsamie, Martin Frotscher, Orazio Nicolotti, Abdelrahman Mohamed, Angelo Carotti, Arcangela Mazzini, Hanna Drzewiecka, Emanuele M. Gargano, Paweł P. Jagodziński, Sandrine Marchais-Oberwinkler
المساهمون: HIPS, Helmholtz-Institut für Pharmazeutische Forschung Saarland, Universitätscampus E8.1 66123 Saarbrücken, Germany.
المصدر: ACS medicinal chemistry letters
United States
ACS Med Chem Lett
ACS medicinal chemistry letters (2021). doi:10.1021/acsmedchemlett.1c00462
info:cnr-pdr/source/autori:Emanuele M. Gargano, Abdelrahman Mohamed, Ahmed S. Abdelsamie, Giuseppe F. Mangiatordi, Hanna Drzewiecka, Pawe? P. Jagodzi?ski, Arcangela Mazzini, Chris J. van Koppen, Matthias W. Laschke, Orazio Nicolotti, Angelo Carotti, Sandrine Marchais-Oberwinkler, Rolf W. Hartmann, and Martin Frotscher/titolo:17?-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer/doi:10.1021%2Facsmedchemlett.1c00462/rivista:ACS medicinal chemistry letters/anno:2021/pagina_da:/pagina_a:/intervallo_pagine:/volumeمصطلحات موضوعية: business.industry, Organic Chemistry, Treatment options, medicine.disease, Biochemistry, Docking, respiratory tract diseases, Drug Discovery, Cancer research, Medicine, Non small cell, Hydroxysteroid dehydrogenase, business, Lung cancer, hormones, hormone substitutes, and hormone antagonists
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4b72b1eb9a0d3948ea61df325c6e341e
https://hdl.handle.net/10033/623149 -
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المؤلفون: Fatma A.F. Ragab, Ahmed S. Abdelsamie, Sonam Roy, Anna K. H. Hirsch, Mohamed A. Omar, Shadia A. Galal, Imtaiyaz Hassan, Hoda I. El Diwani, Ahmad Abu Turab Naqvi, Sarah H. M. Khairat
المصدر: Archiv der PharmazieREFERENCES. 354(9)
مصطلحات موضوعية: Benzimidazole, Carboxylic acid, Pharmaceutical Science, Antineoplastic Agents, Pyrazole, chemistry.chemical_compound, Structure-Activity Relationship, Adenosine Triphosphate, Cell Line, Tumor, Neoplasms, Drug Discovery, Potency, Humans, Cytotoxicity, IC50, chemistry.chemical_classification, Binding Sites, biology, Hydrogen bond, Combinatorial chemistry, Molecular Docking Simulation, Phosphotransferases (Alcohol Group Acceptor), chemistry, Sphingosine kinase 1, biology.protein, Benzimidazoles
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المؤلفون: Andreas M. Kany, Teresa Röhrig, Wulf Blankenfeldt, Maximilian Bauer, Andrea Scrima, Mostafa M. Hamed, Christian Schütz, Stefan Schmelz, Amir Hodzic, Ahmed S. Abdelsamie, Martin Empting
المصدر: European journal of medicinal chemistry. 226
مصطلحات موضوعية: Pyridines, Sonogashira coupling, Alkyne, Microbial Sensitivity Tests, medicine.disease_cause, chemistry.chemical_compound, Structure-Activity Relationship, Bacterial Proteins, Drug Discovery, medicine, Inverse agonist, Humans, ADME, Pharmacology, chemistry.chemical_classification, Trifluoromethyl, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Pseudomonas aeruginosa, Organic Chemistry, General Medicine, Combinatorial chemistry, Anti-Bacterial Agents, Quorum sensing, Trans-Activators, Divergent synthesis
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المؤلفون: Lorenz Siebenbuerger, Sandrine Marchais-Oberwinkler, Michael D. Menger, Martin Frotscher, Ahmed S. Abdelsamie, Carsten Boerger, Rolf W. Hartmann, Victor Hernandez-Olmos, Claudia Scheuer, Chris J. van Koppen, Matthias W. Laschke
المصدر: Journal of Medicinal Chemistry. 61:10724-10738
مصطلحات موضوعية: 0301 basic medicine, medicine.medical_treatment, Pharmacology, 01 natural sciences, Targeted therapy, Estradiol Dehydrogenases, Mice, 03 medical and health sciences, Pharmacokinetics, Drug Discovery, medicine, Animals, Humans, Potency, Tissue Distribution, Enzyme Inhibitors, Hydroxysteroid dehydrogenase, chemistry.chemical_classification, 010405 organic chemistry, Water, In vitro, 0104 chemical sciences, 030104 developmental biology, Enzyme, Solubility, S9 fraction, chemistry, Drug Design, Osteoporosis, Molecular Medicine, Female, Intracellular
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المؤلفون: Hoda I. El Diwani, Claudiu T. Supuran, Heba T. Abdel-Mohsen, Ahmed S. Abdelsamie, Ahmed M. El Kerdawy, Emanuela Berrino, Mohamed A. Omar
المصدر: Bioorganicmedicinal chemistry. 28(5)
مصطلحات موضوعية: Stereochemistry, Carbonic anhydrase II, Clinical Biochemistry, Pharmaceutical Science, 01 natural sciences, Biochemistry, Carbonic Anhydrase II, Hydrophobic effect, Structure-Activity Relationship, Carbonic anhydrase, Drug Discovery, Moiety, Humans, Carbonic Anhydrase Inhibitors, Molecular Biology, chemistry.chemical_classification, Sulfonamides, biology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Hydrogen bond, Organic Chemistry, Active site, 0104 chemical sciences, Sulfonamide, Amino acid, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Pyrimidines, chemistry, biology.protein, Molecular Medicine