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1
المؤلفون: Nobuyuki Ota, Tetsuya Itoh, Kiyoshi Asakawa, Kazuharu Yamamoto, Akiyoshi Mochizuki, Masashi Aida
المصدر: Japanese Journal of Zoo and Wildlife Medicine. 21:141-144
مصطلحات موضوعية: Ecology, Waterfowl, Leech, Parasitism, Biology, biology.organism_classification
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f8f1c86875f3c5b6d9fa5de2c74463f6
https://doi.org/10.5686/jjzwm.21.141 -
2
المؤلفون: Tsutomu Nagata, Makoto Suzuki, Toshiharu Ohta, Hideyuki Kanno, Masamichi Kishida, Akiyoshi Mochizuki, Daisuke Takano
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:7337-7343
مصطلحات موضوعية: Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Administration, Oral, Pharmaceutical Science, Pharmacology, Inhibitory postsynaptic potential, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Oral administration, Drug Discovery, medicine, Animals, Computer Simulation, Ionic compound, Molecular Biology, Short duration, Ions, Aniline Compounds, Binding Sites, Chemistry, Organic Chemistry, Anticoagulants, Haplorhini, In vitro, Protein Structure, Tertiary, Orally active, Factor Xa, Molecular Medicine, Derivative (chemistry), Factor Xa Inhibitors
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3
المؤلفون: Kenji Yoshikawa, Toshiharu Yoshino, Makoto Takemura, Akiyoshi Mochizuki, Toshiharu Ohta, Tsutomu Nagata, Kouichi Uoto, Yoshihiro Yokomizo, Hiroyuki Naito, Katsuhiro Kawakami, Hideyuki Kanno, Makoto Suzuki
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2133-2140
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, Molecular model, medicine.drug_mechanism_of_action, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Factor Xa Inhibitor, Substituent, Pharmaceutical Science, Ethylenediamine, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Structure–activity relationship, Moiety, Molecular Biology, chemistry.chemical_classification, Organic Chemistry, chemistry, Drug Design, Molecular Medicine, Factor Xa Inhibitors
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4
المؤلفون: Makoto Suzuki, Tsutomu Nagata, Hideyuki Kanno, Toshiharu Yoshino, Satoshi Komoriya, Toshiharu Ohta, Kenji Yoshikawa, Yumi Nakamoto, Shozo Kobayashi, Kengo Watanabe, Noriyasu Haginoya, Akiyoshi Mochizuki
المصدر: Bioorganic & Medicinal Chemistry. 17:8221-8233
مصطلحات موضوعية: medicine.drug_mechanism_of_action, Molecular model, Stereochemistry, medicine.drug_class, Antithrombin III, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Moiety, Molecular Biology, Cyclohexylamines, Binding Sites, Molecular Structure, Bicyclic molecule, Chemistry, Organic Chemistry, Anticoagulants, Drug Design, Lipophilicity, Molecular Medicine, Protein Binding
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5
المؤلفون: Satoshi Komoriya, Yumiko Isobe, Akiyoshi Mochizuki, Noriyasu Haginoya, Haruhiko Horino, Makoto Suzuki, Masanori Suzuki, Tsutomu Nagata, Toshiharu Yoshino, Taketoshi Furugoori, Shozo Kobayashi, Takayasu Nagahara
المصدر: Bioorganic & Medicinal Chemistry. 13:3927-3954
مصطلحات موضوعية: Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Administration, Oral, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Blood Coagulation, Molecular Biology, Active metabolite, Binding Sites, biology, Chemistry, Aryl, Organic Chemistry, Anticoagulants, Biological activity, Rats, Intestinal Absorption, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Blood Coagulation Tests, Lead compound, Factor Xa Inhibitors
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6
المؤلفون: Akinori Tatara, Yoshinori Fujimoto, Noriyuki Hara, Akiyoshi Mochizuki
المصدر: Tetrahedron: Asymmetry. 11:1859-1868
مصطلحات موضوعية: Hydrogen, Stereochemistry, Organic Chemistry, Substituent, chemistry.chemical_element, Optically active, Catalysis, law.invention, Inorganic Chemistry, chemistry.chemical_compound, chemistry, Deuterium, law, Physical and Theoretical Chemistry, Walden inversion, Boron trifluoride
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7
المؤلفون: Shojiro Miyazaki, Kazuhiko Tamaki, Chie Sugita, Yoko Nagai, Teppei Fujimoto, Akiyoshi Mochizuki, Yuji Nakamura, Takahiro Nagayama, Shin-ichi Inoue, Katsuyoshi Chiba, Yutaka Mori, Ogawa Yasuyuki, Takahide Nishi
المصدر: Bioorganicmedicinal chemistry. 21(18)
مصطلحات موضوعية: medicine.medical_specialty, Clinical Biochemistry, hERG, Pharmaceutical Science, High renin, Administration, Oral, Blood Pressure, Pharmacology, Biochemistry, Piperazines, chemistry.chemical_compound, Structure-Activity Relationship, Piperidines, Oral administration, Furosemide, Internal medicine, Drug Discovery, Renin–angiotensin system, Renin, medicine, Animals, Protease Inhibitors, Molecular Biology, biology, Chemistry, Organic Chemistry, Chemical modification, Amides, Rats, Disease Models, Animal, Macaca fascicularis, Endocrinology, Orally active, Hypertension, biology.protein, Molecular Medicine, Piperidine, Rats, Transgenic, medicine.drug, Half-Life
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8
المؤلفون: Kazuhiko Tamaki, Akiyoshi Mochizuki, Kiyoshi Takasuna, Katsuyoshi Chiba, Chie Sugita, Takahide Nishi, Ogawa Yasuyuki, Teppei Fujimoto, Yoko Nagai, Masayoshi Asano, Mikio Kato, Hidenori Namiki, Takahiro Nagayama, Yuji Nakamura, Sayaka Suzuki, Shin-ichi Inoue, Shojiro Miyazaki
المصدر: Bioorganicmedicinal chemistry. 21(11)
مصطلحات موضوعية: Male, medicine.medical_specialty, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Pharmacology, Biochemistry, Renin inhibitor, Plasma renin activity, Piperazines, Structure-Activity Relationship, Organ Culture Techniques, In vivo, Oral administration, Internal medicine, Drug Discovery, Renin–angiotensin system, Renin, medicine, Animals, Humans, Arterial Pressure, Protease Inhibitors, Molecular Biology, Antihypertensive Agents, Chemistry, Organic Chemistry, Furosemide, Arrhythmias, Cardiac, Heart, Rats, Macaca fascicularis, Orally active, Endocrinology, Blood pressure, Hypertension, Molecular Medicine, Female, Rabbits, medicine.drug
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9
المؤلفون: Kenji Yoshikawa, Toshiharu Yoshino, Ryo Muto, Akiyoshi Mochizuki, Toshiharu Ohta, Hideyuki Kanno, Yumi Nakamoto, Tsutomu Nagata, Noriyasu Haginoya
المصدر: ChemInform. 43
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Chemistry, Stereochemistry, Diol, One-Step, Mitsunobu reaction, General Medicine, Ring (chemistry), Thiazole, Pyrrolidine, Sulfonamide
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10
المؤلفون: Takahiro Nagayama, Yumi Matsui, Yutaka Mori, Mizuki Takahashi, Chie Sugita, Yoko Nagai, Shin-ichi Inoue, Takahide Nishi, Akiyoshi Mochizuki, Kazuhiko Tamaki, Ogawa Yasuyuki, Yuji Nakamura, Shojiro Miyazaki
المصدر: Bioorganicmedicinal chemistry letters. 22(24)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Angiotensin-Converting Enzyme Inhibitors, Crystallography, X-Ray, Biochemistry, Molecular conformation, Piperazines, chemistry.chemical_compound, Structure-Activity Relationship, Pharmacokinetics, Piperidines, Renin–angiotensin system, Drug Discovery, Renin, Structure–activity relationship, Animals, Humans, Molecular Biology, Dose-Response Relationship, Drug, Drug discovery, Organic Chemistry, Haplorhini, chemistry, Molecular Medicine, Piperidine