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1
المؤلفون: Samuel J. Tremont, Rick L. Fenton, Alan F. Gasiecki, William E. Perkins, Peter H. Jones, Paul W. Collins, Denis Forster, Grace M. Wagner, Martin P. Mcgrath
المصدر: Catalysis of Organic Reactions
مصطلحات موضوعية: chemistry.chemical_classification, Materials science, chemistry, Nanotechnology, Polymer, Designing drug, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a3b7d8aca6d9db697d10afd6b25203de
https://doi.org/10.1201/9781315138855-21 -
2
المؤلفون: Alan F. Gasiecki, Douglas Kalvin, Eric F. Johnson, Irini Akritopoulou-Zanze, Stevan W. Djuric, Brian D. Wakefield, Peter Kovar
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:1480-1483
مصطلحات موضوعية: Indazoles, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Protein Kinase Inhibitors, Molecular Biology, EGFR inhibitors, chemistry.chemical_classification, Molecular Structure, biology, Bicyclic molecule, Chemistry, Kinase, Organic Chemistry, Enzyme, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Tau-protein kinase, Signal transduction
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3
المؤلفون: Srinivasan Nagarajan, Ish K. Libertyville Khanna, Tiffany Duffin, Alan F. Gasiecki, Jeffery L. Keene, Mihir D. Parikh, Michael Clare, Marisa M. Westlin, Maureen A. Nickols, Christina A. Steininger, Melanie L. Williams, Hwang-Fun Lu, Thomas Rogers, Jon A. Klover, Mary Beth Finn, V. Wayne Engleman, Sandra K. Freeman, William F. Westlin, Barbara B. Chen, G. Alan Nickols, Kristen E. Shannon, Mark A. Russell, Bipinchandra N. Desai
المصدر: Bioorganic & Medicinal Chemistry. 15:3390-3412
مصطلحات موضوعية: Male, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Tripeptide, Acetates, Crystallography, X-Ray, Transfection, Biochemistry, Chemical synthesis, Cell Line, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Structure–activity relationship, Peptide bond, Naphthyridines, Molecular Biology, Chromatography, High Pressure Liquid, Integrin alphaVbeta3, Organic Chemistry, Biological activity, Small molecule, Rats, chemistry, Area Under Curve, Drug Design, Molecular Medicine, Indicators and Reagents, Spectrophotometry, Ultraviolet, Lead compound, Half-Life
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المؤلفون: Peter F. Bousquet, Daniel H. Albert, Gary A. Gintant, Patrick A. Marcotte, Gilbert Diaz, George A. Cunha, Ruth L. Martin, Kathryn Houseman, Stevan W. Djuric, Jürgen Dinges, Jennifer J. Bouska, Thomas J. Sowin, Paul Tapang, Charles W. Hutchins, Michael R. Michaelides, Kimba L. Ashworth, Eric F. Johnson, Henry Q. Zhang, Irini Akritopoulou-Zanze, Michelle Nyein, Arnold Lee D, Hu Li, Steven K. Davidsen, Alan F. Gasiecki, Christopher M. Harris, Vijaya Gracias, Zhi Su, Zhiren Xia
المصدر: Journal of Medicinal Chemistry. 50:2011-2029
مصطلحات موضوعية: Models, Molecular, ERG1 Potassium Channel, Patch-Clamp Techniques, Platelet-derived growth factor, hERG, Antineoplastic Agents, Thiophenes, Binding, Competitive, Cell Line, Mice, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Growth factor receptor, Drug Discovery, Animals, Edema, Humans, Receptors, Platelet-Derived Growth Factor, Uterine Diseases, Mice, Inbred BALB C, Estradiol, biology, Kinase, Stereoisomerism, Vascular Endothelial Growth Factor Receptor-2, Xenograft Model Antitumor Assays, Ether-A-Go-Go Potassium Channels, Potassium channel, Receptors, Vascular Endothelial Growth Factor, Indenes, Biochemistry, chemistry, Enzyme inhibitor, Alkynes, biology.protein, Pyrazoles, Molecular Medicine, Female, Signal transduction, Platelet-derived growth factor receptor, Protein Binding
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5
المؤلفون: Thomas G. Pagano, Vijaya Gracias, Stevan W. Djuric, Alan F. Gasiecki
المصدر: Tetrahedron Letters. 47:8873-8876
مصطلحات موضوعية: C h bond, Chemistry, Stereochemistry, education, Organic Chemistry, General Medicine, Biochemistry, Medicinal chemistry, humanities, Catalysis, chemistry.chemical_compound, Reaction sequence, Intramolecular force, Drug Discovery, Imidazole
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6
المؤلفون: Alan F. Gasiecki, Vijaya Gracias, Stevan W. Djuric
المصدر: Tetrahedron Letters. 46:9049-9052
مصطلحات موضوعية: Molecular complexity, chemistry.chemical_compound, Reaction sequence, Chemistry, Stereochemistry, Intramolecular force, Organic Chemistry, Drug Discovery, General Medicine, Azepine, Enyne metathesis, Combinatorial chemistry, Biochemistry
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7
المؤلفون: Vijaya Gracias, Alan F. Gasiecki, Stevan W. Djuric
المصدر: Organic Letters. 7:3183-3186
مصطلحات موضوعية: Molecular complexity, chemistry.chemical_compound, Ring-closing metathesis, Bicyclic molecule, Chemistry, Stereochemistry, Organic Chemistry, Salt metathesis reaction, Imidazole, General Medicine, Physical and Theoretical Chemistry, Combinatorial chemistry, Biochemistry
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المؤلفون: Thomas D. Penning, Nizal S. Chandrakumar, Barbara B. Chen, Helen Y. Chen, Bipin N. Desai, Stevan W. Djuric, Stephen H. Docter, Alan F. Gasiecki, Richard A. Haack, Julie M. Miyashiro, Mark A. Russell, Stella S. Yu, David G. Corley, Richard C. Durley, Brian F. Kilpatrick, Barry L. Parnas, Leslie J. Askonas, James K. Gierse, Elizabeth I. Harding, Maureen K. Highkin, James F. Kachur, Suzanne H. Kim, Gwen G. Krivi, Doreen Villani-Price, E. Yvonne Pyla, Walter G. Smith, Nayereh S. Ghoreishi-Haack
المصدر: Journal of Medicinal Chemistry. 43:721-735
مصطلحات موضوعية: Male, Pyrrolidines, Tertiary amine, Administration, Oral, In Vitro Techniques, Pharmacology, Leukotriene B4, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Drug Discovery, Hydrolase, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Epoxide Hydrolases, chemistry.chemical_classification, biology, In vitro, Enzyme, Biochemistry, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Ex vivo
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9
المصدر: Tetrahedron Letters. 49:6286-6288
مصطلحات موضوعية: chemistry.chemical_compound, Ring-closing metathesis, Chemistry, Stereochemistry, Organic Chemistry, Drug Discovery, Ammonium, Structural motif, Biochemistry, Combinatorial chemistry
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المؤلفون: Doreen Villani-Price, Suzanne H Kim, Walter G. Smith, Leslie J Askonas, Elizabeth I Harding, Maureen K Highkin, Thomas D. Penning, Alan F. Gasiecki, Nayereh S Ghoreishi-Haack, Nizal S Chandrakumar, E.Yvonne Pyla, Bipin N Desai, James F Kachur, Mark A Russell, Stevan W Djuric, James W. Malecha, James K. Gierse, Julie M Miyashiro
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:1137-1139
مصطلحات موضوعية: Imidazopyridine, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Purine analogue, In Vitro Techniques, Biochemistry, Chemical synthesis, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Purine metabolism, Molecular Biology, Epoxide Hydrolases, biology, Chemistry, Organic Chemistry, Recombinant Proteins, stomatognathic diseases, Purines, Enzyme inhibitor, biology.protein, Molecular Medicine, Indicators and Reagents, Ex vivo