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1
المؤلفون: Shaker A. Mousa, Alexander L. Johnson, Anju Parthasarathy, Gregory James Wells, John M. Fevig, Ruth R. Wexler, William F. DeGrado, John Wityak, Sharon A. Jackson
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:2097-2100
مصطلحات موضوعية: chemistry.chemical_classification, Quantitative structure–activity relationship, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Molecular Biology, Biochemistry, Combinatorial chemistry, Cyclic peptide
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2
المؤلفون: Peter J. Gillies, C. Anne Higley, Pennio Pennev, Alexander L. Johnson, Candy S. Robinson, Richard G. Wilde, Thomas P. Maduskuie, Jeffrey T. Billheimer, Ruth R. Wexler
المصدر: Journal of Medicinal Chemistry. 37:3511-3522
مصطلحات موضوعية: Male, Stereochemistry, Sterol O-acyltransferase, Thio, Structure-Activity Relationship, In vivo, Cricetinae, Drug Discovery, Animals, Urea, Structure–activity relationship, IC50, chemistry.chemical_classification, Mesocricetus, Molecular Structure, biology, Anticholesteremic Agents, Imidazoles, In vitro, Rats, Cholesterol, Enzyme, Biochemistry, chemistry, Enzyme inhibitor, Microsomes, Liver, biology.protein, Molecular Medicine, Sterol O-Acyltransferase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::384606c84f7d1f655086b272c98237d8
https://doi.org/10.1021/jm00047a009 -
3
المؤلفون: Thomas E. Christos, Alexander L. Johnson, Gary A. Cain, William K. Schmidt, S. William Tam
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:2347-2352
مصطلحات موضوعية: chemistry.chemical_classification, 5-HT2 receptor, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Sigma, Ether, Biochemistry, Combinatorial chemistry, Propargyl ether, chemistry.chemical_compound, chemistry, In vivo, Drug Discovery, Molecular Medicine, Receptor, Molecular Biology, Alkyl, 5-HT receptor
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4
المؤلفون: D. E. Grigoriadis, Paul J. Gilligan, Alexander L. Johnson, Gary A. Cain, S. William Tam, Charles J. Eyermann, Thomas E. Christos
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:329-334
مصطلحات موضوعية: Ligand, Stereochemistry, Chemistry, fungi, Organic Chemistry, Clinical Biochemistry, Sigma receptor, Pharmaceutical Science, Sigma, Conjugated system, Biochemistry, Drug Discovery, bacteria, Molecular Medicine, Receptor, Molecular Biology
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5
المؤلفون: Gary A. Cain, Alexander L. Johnson, Pat N. Confalone, Richard S. Pottorf, S. William Tam, William K. Schmidt, Thomas E. Christos
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:2055-2060
مصطلحات موضوعية: Stereochemistry, Chemistry, digestive, oral, and skin physiology, Organic Chemistry, Clinical Biochemistry, Analgesic, Pharmaceutical Science, Neuropeptide, Peptide hormone, complex mixtures, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Nociception, In vivo, Drug Discovery, Molecular Medicine, Molecular Biology, hormones, hormone substitutes, and hormone antagonists, Neurotensin, Neurotensin receptor binding
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6
المؤلفون: S.William Tam, Alexander L. Johnson, Richard S. Pottorf, Gary Avonn Cain, Thomas Eugene Christos, William K. Schmidt
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:1767-1772
مصطلحات موضوعية: chemistry.chemical_classification, Tetrapeptide, Chemistry, Stereochemistry, musculoskeletal, neural, and ocular physiology, digestive, oral, and skin physiology, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Neuropeptide, Biological activity, digestive system, complex mixtures, Biochemistry, Pentapeptide repeat, Amino acid, chemistry.chemical_compound, In vivo, Drug Discovery, Molecular Medicine, Molecular Biology, hormones, hormone substitutes, and hormone antagonists, Neurotensin receptor binding, Neurotensin
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7
المؤلفون: Alexander L. Johnson, William K. Schmidt, S. William Tam, Thomas E. Christos, Argyrios G. Arvanitis, Richard S. Pottorf, Gary A. Cain
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:1035-1040
مصطلحات موضوعية: chemistry.chemical_classification, Double bond, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Combinatorial chemistry, chemistry.chemical_compound, chemistry, In vivo, Amide, Drug Discovery, Molecular Medicine, Peptide bond, Molecular Biology, Function (biology), Neurotensin
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8
المؤلفون: Andrew T. Chiu, Pieter B.M.W.M. Timmermans, Alexander L. Johnson, Pancras C. Wong, David J. Carini, Ruth R. Wexler
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:895-898
مصطلحات موضوعية: medicine.medical_specialty, Angiotensin receptor, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Selective antagonist, Biochemistry, Angiotensin II, Blood pressure, Endocrinology, Internal medicine, Drug Discovery, dup, medicine, Molecular Medicine, Molecular Biology
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9
المؤلفون: David J. Carini, Ruth R. Wexler, P. C. Wong, William A. Price, Andrew T. Chiu, S. E. Yoo, J. B. Iii Santella, Michael E. Pierce, J. V. Duncia, Alexander L. Johnson, P. B. M. W. M. Timmermans, Paul E. Aldrich, Gregory James Wells
المصدر: ChemInform. 22
مصطلحات موضوعية: Angiotensin receptor, Orally active, Chemistry, General Medicine, Pharmacology
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10
المؤلفون: S W Tam, Gary A. Cain, Thomas E. Christos, Paul J. Gilligan, D. E. Grigoriadis, Alexander L. Johnson, Charles J. Eyermann
المصدر: ChemInform. 25
مصطلحات موضوعية: Chemistry, Stereochemistry, Sigma receptor, General Medicine