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المؤلفون: Elisabetta Armani, Andrea Rizzi, Nicolò Iotti, Francesca Saccani, Maria Rosaria Di Lascia, Laura Tigli, Alice Pappani, Gessica Marchini, Annalisa Murgo, Anna Maria Capelli, Maurizio Delcanale, Paola Puccini, Gino Villetti, Maurizio Civelli, Claudia Beato, Marta Giuliani, Claudia Mundi, Francesca Murarolli, Mafalda Pagano, Luca F. Raveglia, Rosaria Remelli, Gabriele Amari
المصدر: Journal of Medicinal Chemistry. 66:5622-5656
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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المؤلفون: Maurizio Civelli, Anna Rita Pisano, Gino Villetti, Hervé Van de Poël, Francesco Amadei, Vanessa Pitozzi, Carmelida Capaldi, Gabriele Amari, Alice Pappani, Michela Salvadori, Fanti Renato De, Paola Puccini, Valentina Cenacchi, Wesley Blackaby, Maurizio Delcanale, Riccardo Patacchini, Kevin Nash, Andrea Rizzi, Gessica Marchini, Maria Pittelli, Marcello Trevisani, Elisabetta Armani, Charles Baker-Glenn
المصدر: Journal of Medicinal Chemistry. 64:9100-9119
مصطلحات موضوعية: chemistry.chemical_classification, 0303 health sciences, Antagonist, Muscarinic acetylcholine receptor M3, Pharmacology, 01 natural sciences, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Enzyme, chemistry, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, Molecular Medicine, Intracellular, Ex vivo, 030304 developmental biology
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المؤلفون: Elisabetta, Armani, Andrea, Rizzi, Carmelida, Capaldi, Renato, De Fanti, Maurizio, Delcanale, Gino, Villetti, Gessica, Marchini, Anna Rita, Pisano, Vanessa, Pitozzi, Maria Gloria, Pittelli, Marcello, Trevisani, Michela, Salvadori, Valentina, Cenacchi, Paola, Puccini, Francesco, Amadei, Alice, Pappani, Maurizio, Civelli, Riccardo, Patacchini, Charles A G, Baker-Glenn, Hervé, Van de Poël, Wesley P, Blackaby, Kevin, Nash, Gabriele, Amari
المصدر: Journal of medicinal chemistry. 64(13)
مصطلحات موضوعية: Male, Receptor, Muscarinic M3, Dose-Response Relationship, Drug, Molecular Structure, Guinea Pigs, Cyclic Nucleotide Phosphodiesterases, Type 4, Rats, Rats, Sprague-Dawley, Pulmonary Disease, Chronic Obstructive, Structure-Activity Relationship, Rats, Inbred BN, Drug Discovery, Animals, Phosphodiesterase 4 Inhibitors
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المؤلفون: Maurizio Civelli, Alice Pappani, Paola Puccini, Elisabetta Armani, Laura Carzaniga, Silvia Catinella, Roberta Volta, Riccardo Patacchini, Gabriele Amari, Valentina Cenacchi, Maurizio Delcanale, Fabrizio Facchinetti, Chiara Carnini, Carmelida Capaldi, Silvia Capacchi, Andrea Rizzi, Gessica Marchini, Valentina Bagnacani, Gino Villetti, Nadia Moretto, Loredana Battipaglia, Paola Caruso, Francesco Amadei, Eleonora Ghidini, Fanti Renato De
المصدر: Journal of Medicinal Chemistry. 60:10026-10046
مصطلحات موضوعية: Male, 0301 basic medicine, Drug, Pyrrolidines, media_common.quotation_subject, Respiratory Tract Diseases, Drug Evaluation, Preclinical, Pharmacology, Pathogenesis, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Stability, Pharmacokinetics, Rats, Inbred BN, Administration, Inhalation, Drug Discovery, Animals, Humans, Structure–activity relationship, Pulmonary Eosinophilia, ADME, media_common, chemistry.chemical_classification, Binding Sites, Dose-Response Relationship, Drug, Chemistry, Drug discovery, In vitro, Cyclic Nucleotide Phosphodiesterases, Type 4, Thiazoles, 030104 developmental biology, Enzyme, 030220 oncology & carcinogenesis, Molecular Medicine, Phosphodiesterase 4 Inhibitors
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المؤلفون: Silvia Cantoni, Alessandro Fioni, Alice Pappani, Fabrizio Facchinetti, Fiorella Pastore, Stefano Cavalli, Massimiliano Cont, Gino Villetti
المصدر: Vascular Pharmacology. 132:106706
مصطلحات موضوعية: Pharmacology, Physiology, business.industry, Rat model, Molecular Medicine, Medicine, Antagonism, Endothelin receptor, business
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المؤلفون: Andrew Allen, Veronica Puviani, Cataldo Martucci, Gino Villetti, Alice Pappani, Maurizio Civelli, Fabrizio Facchinetti, Chiara Carnini, Daniela Miglietta, Riccardo Patacchini
المصدر: Airway Pharmacology and Treatment.
مصطلحات موضوعية: COPD, Lung, medicine.diagnostic_test, business.industry, p38 mitogen-activated protein kinases, Inflammation, Pharmacology, medicine.disease, Tobacco smoke, respiratory tract diseases, Therapeutic approach, medicine.anatomical_structure, Bronchoalveolar lavage, Medicine, Nasal administration, medicine.symptom, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::beb9e55968e345ec30d3614645793ba9
https://doi.org/10.1183/1393003.congress-2017.oa4831 -
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المؤلفون: Paola Maria Gallo, Fabrizio Facchinetti, Mauro Corsi, Filippo Visentini, Daniele Pala, Matteo Biagetti, Marco Mor, Alice Pappani, Serena Bertolini, Anna Maria Capelli, Silvia Capacchi, Silvia Rivara, Alessio Lodola
المصدر: Journal of medicinal chemistry. 60(10)
مصطلحات موضوعية: Steric effects, Models, Molecular, Molecular model, Stereochemistry, 010402 general chemistry, 01 natural sciences, chemistry.chemical_compound, Mice, Isomerism, Drug Discovery, Animals, Humans, Methylene, Conformational isomerism, Protein Kinase Inhibitors, Phosphoinositide-3 Kinase Inhibitors, Atropisomer, 010405 organic chemistry, Adenine, Biological activity, 0104 chemical sciences, Class Ia Phosphatidylinositol 3-Kinase, chemistry, Axial chirality, Quinazolines, Molecular Medicine, Methyl group
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المؤلفون: Alice Pappani, Cristina Padula, Patrizia Santi
المصدر: International journal of pharmaceutics. 349(1-2)
مصطلحات موضوعية: Drug, media_common.quotation_subject, Chemistry, Pharmaceutical, Skin Absorption, Levothyroxine, Pharmaceutical Science, Absorption (skin), Pharmacology, In Vitro Techniques, Administration, Cutaneous, Diffusion, Excipients, Pharmacokinetics, Drug Stability, medicine, Animals, Solubility, Ear, External, Transdermal, media_common, Cyclodextrins, integumentary system, Chemistry, Permeation, Iontophoresis, Thyroxine, Solvents, Rabbits, medicine.drug, Levothyroxine Sodium