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1
المؤلفون: W. J. Howe, W. T. Lowther, J. O. Hui, W. G. Tarpley, D. E. Emmert, Chetana Rao, A G Tomasselli, John H. Kinner, V. S. Bradford, D. L. Alexander, Tomi K. Sawyer, B.M. Dunna, Robert A. Conradi, D. L. Decamp, Clark W. Smith, Allen W. Harrison, Charles S. Craik, James Michael Tustin, T. J. Mcquade, Robert L. Heinrikson, Y. Z. Zhang, Philip S. Burton, Jed F. Fisher, Roger A. Poorman, Joseph B. Moon, Jackson B. Hester, D J Staples, L. Liu, P. E. Scarborough, Maggiora Linda Louise
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:819-824
مصطلحات موضوعية: Cathepsin, Protease, Dipeptide, biology, Isostere, Peptidomimetic, Chemistry, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Enzyme binding, chemistry.chemical_compound, Pepsin, Drug Discovery, medicine, biology.protein, Molecular Medicine, Pharmacophore, Molecular Biology
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2
المؤلفون: W. J. Howe, W. T. Lowther, A G Tomasselli, D. E. Emmert, D J Staples, Jackson B. Hester, W. G. Tarpley, J. O. Hui, Ben M. Dunn, John H. Kinner, Robert L. Heinrikson, Y. Z. Zhang, Tomi K. Sawyer, Charles S. Craik, D. L. Decamp, James Michael Tustin, T. J. Mcquade, D. L. Alexander, Allen W. Harrison, P. E. Scarborough, Robert A. Conradi, Jed F. Fisher, Roger A. Poorman, Philip S. Burton, Maggiora Linda Louise, V. S. Bradford, Joseph B. Moon, L. Liu, Clark W. Smith, Chetana Rao
المصدر: ChemInform. 26
مصطلحات موضوعية: Enzyme binding, Protease, Chemistry, Peptidomimetic, medicine.medical_treatment, Human immunodeficiency virus (HIV), medicine, General Medicine, Selectivity, medicine.disease_cause, Cell permeability, Virology
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3
المؤلفون: Gordon L. Bundy, Bob D. Rush, Mary J. Ruwart, Jed F. Fisher, Allen W. Harrison, Karen F. Wilkinson
المصدر: Journal of Medicinal Chemistry. 34:3140-3143
مصطلحات موضوعية: Glycosylation, Peptide, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Renin, Drug Discovery, Renin–angiotensin system, Animals, Bile, chemistry.chemical_classification, Oligopeptide, Molecular Structure, biology, Glycopeptides, Glycopeptide, Rats, Kinetics, Enzyme, Intestinal Absorption, Liver, Biochemistry, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Oligopeptides
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d850e436ec222b9074f4cc9ad7f32c78
https://doi.org/10.1021/jm00114a026 -
4
المؤلفون: David M. Guido, Donald T. Pals, Sally J. Couch, Allen W. Harrison, Garry L. Degraaf, Judy A. Lawson, John Rogers, Dorothy M. Sutter, Mark V. Williams, Jed F. Fisher
المصدر: Bioorganicmedicinal chemistry. 2(12)
مصطلحات موضوعية: medicine.drug_class, Clinical Biochemistry, Molecular Sequence Data, Pharmaceutical Science, Peptide, Blood Pressure, Plasma protein binding, Biochemistry, Renin inhibitor, Structure-Activity Relationship, In vivo, Drug Discovery, Renin, medicine, Structure–activity relationship, Animals, Amino Acid Sequence, Molecular Biology, Antihypertensive Agents, chemistry.chemical_classification, Oligopeptide, Molecular Structure, Chemistry, Organic Chemistry, Glycopeptides, Glycopeptide, Rats, Macaca fascicularis, Carbohydrate Sequence, Solubility, Molecular Medicine, Linker, Oligopeptides, Protein Binding
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5
المؤلفون: Allen W. Harrison, Dong-Chool Kim, Jed F. Fisher, Ronald T. Borchardt, Ismael J. Hidalgo, Karen F. Wilkinson, Mary J. Ruwart
المصدر: Journal of drug targeting. 1(4)
مصطلحات موضوعية: Male, endocrine system, endocrine system diseases, medicine.drug_class, Cell, Pharmaceutical Science, In Vitro Techniques, digestive system, Bile Acids and Salts, Rats, Sprague-Dawley, Intestinal mucosa, In vivo, Ileum, Renin, medicine, Tumor Cells, Cultured, Animals, Humans, Intestinal permeability, Bile acid, Chemistry, Carcinoma, nutritional and metabolic diseases, medicine.disease, G protein-coupled bile acid receptor, Epithelium, Rats, medicine.anatomical_structure, Biochemistry, Intestinal Absorption, Colonic Neoplasms, Carrier Proteins, Oligopeptides, hormones, hormone substitutes, and hormone antagonists, Conjugate
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6
المصدر: The Journal of Organic Chemistry. 49:438-442
مصطلحات موضوعية: Organic Chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::1c4704f0ec5f540feb370b095428be13
https://doi.org/10.1021/jo00177a010 -
7
المؤلفون: Paul A. Aristoff, Anne M. Huber, Allen W. Harrison
المصدر: Tetrahedron Letters. 25:3955-3958
مصطلحات موضوعية: Intramolecular reaction, Bicyclic molecule, Stereochemistry, Chemistry, Organic Chemistry, Prostacyclin, Biochemistry, Benzopyran, chemistry.chemical_compound, Intramolecular force, Drug Discovery, medicine, Mitsunobu reaction, Aliphatic compound, Enone, medicine.drug
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8
المؤلفون: Paul A. Aristoff, Johnson Paul D, Allen W. Harrison
المصدر: Journal of the American Chemical Society. 107:7967-7974
مصطلحات موضوعية: Colloid and Surface Chemistry, Chemistry, Intramolecular force, Wittig reaction, Organic chemistry, Total synthesis, General Chemistry, Biochemistry, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::69cdd9d92841574a40758cac940cf220
https://doi.org/10.1021/ja00312a028 -
9
المؤلفون: Allen W. Harrison, Paul A. Aristoff
المصدر: Tetrahedron Letters. 23:2067-2070
مصطلحات موضوعية: Stereochemistry, Organic Chemistry, Regioselectivity, Prostacyclin, Biochemistry, chemistry.chemical_compound, Prostaglandin analog, chemistry, Drug Discovery, medicine, Organic chemistry, lipids (amino acids, peptides, and proteins), Phenols, Prostaglandin a, medicine.drug
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10
المؤلفون: Paul A. Aristoff, Johnson Paul D, Allen W. Harrison
المصدر: The Journal of Organic Chemistry. 48:5341-5348
مصطلحات موضوعية: chemistry.chemical_classification, Addition reaction, Bicyclic molecule, Chemistry, Carboxylic acid, Organic Chemistry, Organic chemistry, Aliphatic compound, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::04365c6c22c7844e217df93777306088
https://doi.org/10.1021/jo00174a035