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1دورية أكاديمية
المؤلفون: Stefanie Kickinger, Maria E. K. Lie, Akihiro Suemasa, Anas Al-Khawaja, Koichi Fujiwara, Mizuki Watanabe, Kristine S. Wilhelmsen, Christina B. Falk-Petersen, Bente Frølund, Satoshi Shuto, Gerhard F. Ecker, Petrine Wellendorph
المصدر: Frontiers in Chemistry, Vol 9 (2021)
مصطلحات موضوعية: SLC6 neurotransmitter transporters, competitive inhibition, binding mode analysis, computational chemistry, bicyclo-GABA, BGT1, Chemistry, QD1-999
وصف الملف: electronic resource
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2
المؤلفون: Louise Thiesen, Bente Frølund, Anas Al-Khawaja, Maria Damgaard, Aleš Marek, Christoffer Bundgaard, Petrine Wellendorph, Anne S. Haugaard, Mònica Santiveri, Rebekka Löffler
المصدر: ACS Chemical Neuroscience. 9:545-554
مصطلحات موضوعية: 0301 basic medicine, Agonist, Physiology, medicine.drug_class, Cognitive Neuroscience, Biology, Pharmacology, Biochemistry, law.invention, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Betaine, law, medicine, Receptor, GABAA receptor, Substrate (chemistry), Transporter, Cell Biology, General Medicine, 030104 developmental biology, chemistry, Recombinant DNA, 030217 neurology & neurosurgery, Function (biology)
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3
المؤلفون: Anas Al-Khawaja, Stine B. Vogensen, Hans Bräuner-Osborne, Jonas Skovgaard-Petersen, Rasmus P. Clausen, Stefanie Kickinger, Petrine Wellendorph, Arne Schousboe, Rebekka Löffler, Karsten K. Madsen, Gerhard F. Ecker, Emil Rosenthal, Lars N. Jorgensen, Nrupa Borkar
المصدر: Journal of Medicinal Chemistry. 60:8834-8846
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, GABA Plasma Membrane Transport Proteins, Stereochemistry, Allosteric regulation, GABA transporter 1, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Betaine, Piperidines, Drug Discovery, Radioligand, Humans, Structure–activity relationship, Homology modeling, Binding site, Serotonin Plasma Membrane Transport Proteins, biology, Chimera, Chemistry, 030104 developmental biology, Biochemistry, Docking (molecular), Benzamides, biology.protein, Molecular Medicine, GABA Uptake Inhibitors, Carrier Proteins, Allosteric Site
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4
المؤلفون: Rebekka F. Petersen, Maria Damgaard, Anas Al-Khawaja, Mia Nittegaard-Nielsen, Petrine Wellendorph, Bente Frølund
المصدر: European Journal of Medicinal Chemistry. 138:300-312
مصطلحات موضوعية: Pharmacology, Allosteric modulator, 010405 organic chemistry, GABAA receptor, Stereochemistry, Organic Chemistry, General Medicine, Ligand (biochemistry), 01 natural sciences, 0104 chemical sciences, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Monastrol, chemistry, Drug Discovery, Structure–activity relationship, Binding site, Selectivity, Receptor, 030217 neurology & neurosurgery
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5
المؤلفون: Julie T. Christensen, Anas Al-Khawaja, Mia Nittegaard-Nielsen, Petrine Wellendorph, Anders B. Klein
المصدر: MedChemComm. 7:426-432
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, GABAA receptor, Organic Chemistry, Pharmaceutical Science, Bicuculline, Biology, Biochemistry, Cell biology, GABAA-rho receptor, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Muscimol, chemistry, Drug Discovery, medicine, Gabazine, Molecular Medicine, Receptor, Ion channel linked receptors, medicine.drug, G protein-coupled receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::1f74a0dfb7b6f1e0353fe1a58725256c
https://doi.org/10.1039/c5md00442j -
6
المؤلفون: Stefanie Kickinger, Maria Damgaard, Anas Al-Khawaja, Rebekka Löffler, Gerhard F. Ecker, Maria E. K. Lie, Bente Frølund, Petrine Wellendorph, Anne S. Haugaard, Francesco Bavo
المصدر: Biophysical Journal. 118:130a
مصطلحات موضوعية: biology, Biochemistry, Chemistry, Biophysics, biology.protein, Subtype selectivity, GABA transporter
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7
المؤلفون: Anas, Al-Khawaja, Anne S, Haugaard, Ales, Marek, Rebekka, Löffler, Louise, Thiesen, Mònica, Santiveri, Maria, Damgaard, Christoffer, Bundgaard, Bente, Frølund, Petrine, Wellendorph
المصدر: ACS chemical neuroscience. 9(3)
مصطلحات موضوعية: Betaine, Neurons, GABA Plasma Membrane Transport Proteins, Mice, Animals, Membrane Transport Proteins, Biological Transport, gamma-Aminobutyric Acid
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8
المؤلفون: Maria E K, Lie, Anas, Al-Khawaja, Maria, Damgaard, Anne S, Haugaard, Arne, Schousboe, Andrew N, Clarkson, Petrine, Wellendorph
المصدر: Advances in neurobiology. 16
مصطلحات موضوعية: Stroke, GABA Plasma Membrane Transport Proteins, Epilepsy, Animals, Humans, Neuroglia
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::47a9d024c3dffa945e471323337a1c6f
https://pubmed.ncbi.nlm.nih.gov/28828609 -
9
المؤلفون: Maria, Damgaard, Anne Stæhr, Haugaard, Stefanie, Kickinger, Anas, Al-Khawaja, Maria E K, Lie, Gerhard F, Ecker, Rasmus Prætorius, Clausen, Bente, Frølund
المصدر: Advances in neurobiology. 16
مصطلحات موضوعية: GABA Plasma Membrane Transport Proteins, Animals, Brain, Humans, GABA Uptake Inhibitors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::a24459a1c71adde866615832c8e68064
https://pubmed.ncbi.nlm.nih.gov/28828618 -
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المؤلفون: Maria, Damgaard, Anas, Al-Khawaja, Mia, Nittegaard-Nielsen, Rebekka F, Petersen, Petrine, Wellendorph, Bente, Frølund
المصدر: European journal of medicinal chemistry. 138
مصطلحات موضوعية: Structure-Activity Relationship, Binding Sites, Pyrimidines, Dose-Response Relationship, Drug, Molecular Structure, Humans, Thiones, Receptors, GABA-A