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المؤلفون: Jane Hughes, Iain Chessell, Arjan Snijder, Peter E. Thornton, Maria A T Groves, Bojana Popovic, James Button, Claire Dobson, Tristan J Vaughan, Bruck Taddese, Darren J. Schofield, Trevor Wilkinson, Wendy A Williams, Ling Huang, Jon P. Hatcher, Clare A. Jones, Yoko Shibata, George Thom, Bhupinder Dosanjh, Andy Billinton, Carl I Webster, John E. Linley
المصدر: Pain. 160:1989-2003
مصطلحات موضوعية: Purinergic P2X Receptor Antagonists, medicine.drug_class, Pharmacology, Inhibitory postsynaptic potential, Monoclonal antibody, Rats, Sprague-Dawley, Mice, 03 medical and health sciences, 0302 clinical medicine, 030202 anesthesiology, medicine, Animals, Humans, Receptor, Cells, Cultured, Injections, Spinal, Ion channel, biology, Chemistry, Drug discovery, HEK 293 cells, Antibodies, Monoclonal, Rats, Mice, Inbred C57BL, HEK293 Cells, Anesthesiology and Pain Medicine, Neurology, Neuropathic pain, biology.protein, Neuralgia, Female, Neurology (clinical), Antibody, Receptors, Purinergic P2X4, 030217 neurology & neurosurgery, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9866af38e140ef1e2b18bcb9f4825b5b
https://doi.org/10.1097/j.pain.0000000000001587 -
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المؤلفون: Tarik Khaznadar, Helen Susanne Price, Andy Billinton, Martin E. Swarbrick, David Andrew Stevens, Gerard Martin Paul Giblin, Melanie A. Kay, Anton D. Michel, Nicholas Maughan Clayton, David J. Spalding, Alan Naylor, Alex W. Wilson, Amanda C. Allan, Mark Patrick Healy, Iain P. Chessell, Kristin Bailey
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:1892-1896
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, EP4 Receptor, Pharmaceutical Science, Inflammatory pain, Biochemistry, Partial agonist, Anti-inflammatory, 03 medical and health sciences, Acetic acid, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, chemistry, Drug Discovery, Neuropathic pain, medicine, Molecular Medicine, Inhibitory concentration 50, lipids (amino acids, peptides, and proteins), Molecular Biology, 030217 neurology & neurosurgery
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المؤلفون: Robert A. Rissman, Jonathan M. Schott, Aaron P. Schultz, Doug R. Galasko, David Mengel, Reisa A. Sperling, Keith A. Johnson, Michael J. Properzi, Andy Billinton, Zhicheng Chen, Dominic M. Walsh, Ashvini Keshavan, Henrik Zetterberg, Michael S. Perkinton, Jennifer L. Percival-Alwyn, Purvish P. Patel
المصدر: Alzheimer's & Dementia. 14
مصطلحات موضوعية: Psychiatry and Mental health, Cellular and Molecular Neuroscience, medicine.medical_specialty, Endocrinology, Developmental Neuroscience, Terminal (electronics), Epidemiology, Chemistry, Health Policy, Internal medicine, medicine, Neurology (clinical), Geriatrics and Gerontology
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المؤلفون: Mark P, Healy, Amanda C, Allan, Kristin, Bailey, Andy, Billinton, Iain P, Chessell, Nicholas M, Clayton, Gerard M P, Giblin, Melanie A, Kay, Tarik, Khaznadar, Anton D, Michel, Alan, Naylor, Helen, Price, David J, Spalding, David A, Stevens, Martin E, Swarbrick, Alexander W, Wilson
المصدر: Bioorganicmedicinal chemistry letters. 28(10)
مصطلحات موضوعية: Lipopolysaccharides, Blood Cells, Tumor Necrosis Factor-alpha, Anti-Inflammatory Agents, Drug Evaluation, Preclinical, Pain, Isoindoles, Dinoprostone, Rats, Inhibitory Concentration 50, Animals, Humans, Protein Isoforms, Receptors, Prostaglandin E, EP4 Subtype, Half-Life
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المؤلفون: Phil Newton, Michael S. Perkinton, Maria Groves, Tristan J. Vaughan, Anna Bogstedt, Iain P. Chessell, Amanda Dudley, Fraser Welsh, Chris Lloyd, Rajesh Narwal, Keith Tan, Mary McFarlane, Andy Billinton, Susanna Eketjäll
المصدر: Alzheimer's & Dementia. 13
مصطلحات موضوعية: 0301 basic medicine, Amyloid, Epidemiology, medicine.drug_class, business.industry, Health Policy, Monoclonal antibody, 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Psychiatry and Mental health, Cellular and Molecular Neuroscience, 030104 developmental biology, Developmental Neuroscience, medicine, Cancer research, Neurology (clinical), Geriatrics and Gerontology, Beta (finance), business
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المؤلفون: Tomas Ondrejcak, Andy Billinton, Dominic M. Walsh, Maria Groves, Michael S. Perkinton, Tiernan T. O'Malley, Iain P. Chessell, Michael J. Rowan, Amanda Dudley
المصدر: Alzheimer's & Dementia. 13
مصطلحات موضوعية: biology, Epidemiology, Chemistry, Health Policy, C-terminus, Cell biology, Psychiatry and Mental health, Cellular and Molecular Neuroscience, Developmental Neuroscience, Biochemistry, In vivo, Synaptic plasticity, biology.protein, Neurology (clinical), Geriatrics and Gerontology, Antibody
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المؤلفون: Thor Ostenfeld, Richard Turner, Eva Lindqvist, Amanda Dudley, Iain P. Chessell, Michael Pomfret, Manasa Tatipalli, Rajesh Narwal, Nancy Y. Lee, Maria Groves, Andy Billinton, Keith Tan, Zulma Santisteban Valencia, Tharani Chessell
المصدر: Alzheimer's & Dementia. 13
مصطلحات موضوعية: 0301 basic medicine, Amyloid, Epidemiology, business.industry, Health Policy, Safety tolerability, Disease, Pharmacology, 03 medical and health sciences, Psychiatry and Mental health, Cellular and Molecular Neuroscience, Specific antibody, 030104 developmental biology, 0302 clinical medicine, Developmental Neuroscience, Pharmacokinetics, Medicine, In patient, Neurology (clinical), Geriatrics and Gerontology, business, 030217 neurology & neurosurgery
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المؤلفون: Amanda Dudley, Andy Billinton, Iain Chessell
المصدر: Drug Discovery Today. 17:875-879
مصطلحات موضوعية: Pharmacology, Analgesics, Biological Products, medicine.medical_specialty, business.industry, Analgesic, Biologic therapies, Chronic pain, Alternative medicine, Antibodies, Monoclonal, Pain, Inflammatory pain, medicine.disease, Broad spectrum, Drug Discovery, Neuropathic pain, medicine, Physical therapy, Animals, Humans, Intensive care medicine, Cancer pain, business
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المؤلفون: Andrew Charlton, Stephen J. Medhurst, Laura J. Chambers, Livermore David, Brian Peter Slingsby, Andy Billinton, Lee William Page, Anton D. Michel, Daryl S. Walter, Jon Graham Anthony Steadman, Shilina Roman, Sadhana Patel, Elena Fonfria, Robert Gleave, Stefan Senger, Katharine Laura Collis, Andrew P. Moses, Sue D. Collins, Muna H. Abdi, Paul John Beswick, Clarisse L. Lejeune, David Kenneth Dean, Alexander J. Stevens
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5080-5084
مصطلحات موضوعية: Models, Molecular, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Amide, Drug Discovery, Purinergic P2 Receptor Antagonists, medicine, Structure–activity relationship, Receptor, Molecular Biology, Drug discovery, Organic Chemistry, Antagonist, Receptor antagonist, Amides, Pyrrolidonecarboxylic Acid, chemistry, Molecular Medicine, Receptors, Purinergic P2X7, Pyroglutamic acid
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المؤلفون: Andy Billinton, Sue Roomans, Stefan Senger, Anton D. Michel, Stephen J. Medhurst, Robert Gleave, Daryl S. Walter, Elena Fonfria, Laura J. Chambers, Andrew P. Moses, Shilina Roman, David Kenneth Dean, Alexander J. Stevens, Paul John Beswick, Sadhana Patel
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4653-4656
مصطلحات موضوعية: Purinergic P2X Receptor Antagonists, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Analgesic, Administration, Oral, Pain, Pharmaceutical Science, Carboxamide, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Acetamides, Drug Discovery, medicine, Animals, Humans, Molecular Biology, Organic Chemistry, Antagonist, In vitro, Rats, Disease Models, Animal, chemistry, Hyperalgesia, Pyrazoles, Molecular Medicine, Receptors, Purinergic P2X7, medicine.symptom, Lead compound, Acetamide