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1
المؤلفون: Laurence Dumais, Gilles Ouvry, Laurent Chantalat, Angélique Feret, Sandrine Chambon, Thibaud Portal, Sandrine Talano, Gwenaëlle Duvert, Catherine Soulet, Jean-Marie Arlabosse, Samuel Tabet, Sebastien Daver, Jonathan Pascau, Nicolas Rodeville, Catherine Raffin, Claire Bouix-Peter, Etienne Thoreau
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:1736-1741
مصطلحات موضوعية: 0301 basic medicine, Agonist, Receptors, Retinoic Acid, medicine.drug_class, Clinical Biochemistry, Trifarotene, Pharmaceutical Science, Pharmacology, Biochemistry, Retinoids, Structure-Activity Relationship, 030207 dermatology & venereal diseases, 03 medical and health sciences, 0302 clinical medicine, Acne Vulgaris, Drug Discovery, medicine, Humans, Tissue distribution, Molecular Biology, Acne, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Acne treatment, medicine.disease, Molecular Docking Simulation, 030104 developmental biology, Drug Design, Molecular Medicine, Structure based
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2
المؤلفون: Craig S. Harris, Isabelle Cardinaud, Feriel Hacini-Rachinel, Nicolas Rodeville, Audrey Beillard, Arnaud Reitz, Marilyne Bourotte, Benoit Deprez, Laetitia Bonnary, Catherine Comino, Corinne Millois, Delphine Spiesse, Claire Bouix-Peter, Denis Duvert, Jean-Guy Boiteau, Jean-Marie Arlabosse, Yushma Bhurruth-Alcor, Anne-Pascale Luzy, Laurent F. Hennequin, Gaëlle Polge, Emmanuel Vial, Loïc Tomas, Samuel Tabet, Kevin Reverse, Arnaud Mathieu, Artur Pinto, Angélique Feret, Karine Bouquet, Gilles Ouvry, Stéphanie Astri, Nicolas Orsini, Jonathan Pascau, Nathalie Taquet, David Piwnica, Patricia Rossio
المصدر: Bioorganic & Medicinal Chemistry. 26:945-956
مصطلحات موضوعية: 0301 basic medicine, Process development, Administration, Topical, Clinical Biochemistry, Druggability, Pharmaceutical Science, Topical treatment, ADAM17 Protein, Pharmacology, Hydroxamic Acids, Skin Diseases, 01 natural sciences, Biochemistry, Mice, 03 medical and health sciences, In vivo, Psoriasis, Drug Discovery, medicine, Animals, Humans, Enzyme Inhibitors, Molecular Biology, Mice, Hairless, Sulfonamides, Tumor Necrosis Factor-alpha, 010405 organic chemistry, Chemistry, Organic Chemistry, Oxazolone, medicine.disease, Tace inhibitor, 0104 chemical sciences, 030104 developmental biology, Solubility, Drug Design, Microsomes, Liver, Molecular Medicine, Female