نتائج البحث - "Angelo Carotti"

المساهمون: Tonelli, Michele, Catto, Marco, Sabaté, Raimon, Francesconi, Valeria, Laurini, Erik, Pricl, Sabrina, Pisani, Leonardo, Miniero, Daniela Valeria, Liuzzi, Grazia Maria, Gatta, Elena, Relini, Annalisa, Gavín, Rosalina, Del Rio, Jose Antonio, Sparatore, Fabio, Carotti, Angelo

المصدر: European Journal of Medicinal Chemistry. 250:115169

مصطلحات موضوعية: Thioxanthene-9-one and xanthen-9-one derivatives, Multitarget-directed ligands (MTDLs), Pharmacology, AChE and BChE inhibition, Organic Chemistry, Drug Discovery, Alzheimer's disease, Aβ and tau aggregation inhibition, General Medicine, Thioxanthene-9-one and xanthen-9-one derivative

وصف الملف: ELETTRONICO

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fb954dcbed2541fdbb4436bce5991df3
https://doi.org/10.1016/j.ejmech.2023.115169

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7

17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer

المؤلفون: Rolf W. Hartmann, Chris J. van Koppen, Matthias W. Laschke, Giuseppe Felice Mangiatordi, Ahmed S. Abdelsamie, Martin Frotscher, Orazio Nicolotti, Abdelrahman Mohamed, Angelo Carotti, Arcangela Mazzini, Hanna Drzewiecka, Emanuele M. Gargano, Paweł P. Jagodziński, Sandrine Marchais-Oberwinkler

المساهمون: HIPS, Helmholtz-Institut für Pharmazeutische Forschung Saarland, Universitätscampus E8.1 66123 Saarbrücken, Germany.

المصدر: ACS medicinal chemistry letters
United States
ACS Med Chem Lett
ACS medicinal chemistry letters (2021). doi:10.1021/acsmedchemlett.1c00462
info:cnr-pdr/source/autori:Emanuele M. Gargano, Abdelrahman Mohamed, Ahmed S. Abdelsamie, Giuseppe F. Mangiatordi, Hanna Drzewiecka, Pawe? P. Jagodzi?ski, Arcangela Mazzini, Chris J. van Koppen, Matthias W. Laschke, Orazio Nicolotti, Angelo Carotti, Sandrine Marchais-Oberwinkler, Rolf W. Hartmann, and Martin Frotscher/titolo:17?-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Potential Treatment Option for Non-Small Cell Lung Cancer/doi:10.1021%2Facsmedchemlett.1c00462/rivista:ACS medicinal chemistry letters/anno:2021/pagina_da:/pagina_a:/intervallo_pagine:/volume

مصطلحات موضوعية: business.industry, Organic Chemistry, Treatment options, medicine.disease, Biochemistry, Docking, respiratory tract diseases, Drug Discovery, Cancer research, Medicine, Non small cell, Hydroxysteroid dehydrogenase, business, Lung cancer, hormones, hormone substitutes, and hormone antagonists

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4b72b1eb9a0d3948ea61df325c6e341e
https://hdl.handle.net/10033/623149

8

Synthesis and Biological Evaluation of Novel Hybrid Molecules Containing Purine, Coumarin and Isoxazoline or Isoxazole Moieties

المؤلفون: Dimitra Hadjipavlou-Litina, Aikaterini Peperidou, Angelo Carotti, Konstantinos E. Litinas, Michael G. Kallitsakis, Marco Catto

المصدر: The Open Medicinal Chemistry Journal

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::23b2cf96ebb7174a9b580c18f81a0462
https://doi.org/10.2174/1874104501711010196

9

Quinolino[3,4- b ]quinoxalines and pyridazino[4,3- c ]quinoline derivatives: Synthesis, inhibition of topoisomerase IIα, G-quadruplex binding and cytotoxic properties

المؤلفون: Odra Pinato, Marco Catto, Fausta Palluotto, Barbara Gatto, Angelo Carotti, Alice Sosic, Grigoris Zoidis, Claudia Sissi

المصدر: European Journal of Medicinal Chemistry. 123:704-717

مصطلحات موضوعية: DNA Topoisomerase IV, 0301 basic medicine, Stereochemistry, Antineoplastic Agents, Chemistry Techniques, Synthetic, G-quadruplex, G-quadruplex stabilizers, 01 natural sciences, Quinoline derivatives, HeLa, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Antigens, Neoplasm, Quinoxalines, Drug Discovery, Humans, Topoisomerase II Inhibitors, Structure–activity relationship, Cytotoxic agents, Cytotoxicity, IC50, Pharmacology, chemistry.chemical_classification, Topoisomerase IIα inhibitors, biology, 010405 organic chemistry, Drug Discovery3003 Pharmaceutical Science, Organic Chemistry, Quinoline, General Medicine, Pyridazine derivatives, biology.organism_classification, 0104 chemical sciences, DNA-Binding Proteins, G-Quadruplexes, DNA Topoisomerases, Type II, 030104 developmental biology, chemistry, Quinolines, Topoisomerase-II Inhibitor, HeLa Cells, Tricyclic

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f4d41cd82204c2a219105b407fb35b8a
https://doi.org/10.1016/j.ejmech.2016.07.063

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10

Exploring Basic Tail Modifications of Coumarin-Based Dual Acetylcholinesterase-Monoamine Oxidase B Inhibitors: Identification of Water-Soluble, Brain-Permeant Neuroprotective Multitarget Agents

المؤلفون: Roberta Farina, Cosimo Altomare, Rosa Maria Iacobazzi, Orazio Nicolotti, Leonardo Pisani, Saverio Cellamare, Angelo Carotti, Giuseppe Felice Mangiatordi, Marco Catto, Nunzio Denora, Ramón Soto-Otero, Lydia Siragusa

المصدر: Journal of medicinal chemistry 59 (2016): 6791–6806. doi:10.1021/acs.jmedchem.6b00562
info:cnr-pdr/source/autori:Pisani, Leonardo; Farina, Roberta; Catto, Marco; Iacobazzi, Rosa Maria; Nicolotti, Orazio; Cellamare, Saverio; Mangiatordi, Giuseppe Felice; Denora, Nunzio; Soto-Otero, Ramon; Siragusa, Lydia; Altomare, Cosimo Damian; Carotti, Angelo/titolo:Exploring Basic Tail Modifications of Coumarin-Based Dual Acetylcholinesterase-Monoamine Oxidase B Inhibitors: Identification of Water-Soluble, Brain-Permeant Neuroprotective Multitarget Agents/doi:10.1021%2Facs.jmedchem.6b00562/rivista:Journal of medicinal chemistry/anno:2016/pagina_da:6791/pagina_a:6806/intervallo_pagine:6791–6806/volume:59

مصطلحات موضوعية: 0301 basic medicine, Monoamine Oxidase Inhibitors, Cell Survival, Monoamine oxidase, 01 natural sciences, Neuroprotection, Madin Darby Canine Kidney Cells, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Dogs, Coumarins, Cell Line, Tumor, Drug Discovery, Animals, Humans, Structure–activity relationship, Cytotoxicity, Monoamine Oxidase, IC50, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Water, Rotenone, Acetylcholinesterase, 0104 chemical sciences, Oxidative Stress, Neuroprotective Agents, 030104 developmental biology, Solubility, chemistry, Biochemistry, Molecular Medicine, Cholinesterase Inhibitors, Monoamine oxidase B, Medicinal Chemistry

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5fd602b86f863e6fb085cd996912bed9
https://doi.org/10.1021/acs.jmedchem.6b00562

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