-
1
المؤلفون: Atul Wavhal, Yogesh Waman, Siddhartha De, Anil M. Deshpande, Manoj Joshi, Sachin Kandalkar, Dinesh A. Barawkar, Amol A. Raje, Venkata P. Palle, Kasim A. Mookhtiar, Ashwini Tambe, Shariq S. Ansari, Parimi Atchuta Ramaiah
المصدر: Bioorganic & Medicinal Chemistry. 25:5799-5819
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, 01 natural sciences, Biochemistry, Nucleobase, Structure-Activity Relationship, 03 medical and health sciences, Adenosine deaminase, Catalytic Domain, Drug Discovery, Adenosine Deaminase Inhibitors, medicine, Molecular Biology, Molecular Structure, biology, 010405 organic chemistry, Chemistry, Adenine, Organic Chemistry, Diastereomer, Active site, 0104 chemical sciences, Enzyme Activation, Molecular Docking Simulation, 030104 developmental biology, Docking (molecular), biology.protein, Microsome, Molecular Medicine, EHNA, Adenosine Deaminase Inhibitor, medicine.drug
-
2
المؤلفون: Kasim A. Mookhtiar, Anita Chugh, Rahul D. Kaduskar, Siddhartha De, Dhananjay N. Umrani, Debnath Bhuniya, Keshav Naik, Santosh Kurhade, Prasad Shitole, Balasaheb Kobal, Pratima Patil, Amol A. Raje, Sandhya Chaturvedi Joshi, Vamsi Madgula, Vaibhav Jain, Satyanarayana Reddy, Vyavahare Vinod, Suhas Tambe, Venkata P. Palle, Jayasagar Gundu, Ganesh Bhat, Bhavesh Dave, Anil M. Deshpande, Sachin Kandalkar, Sujay Basu
المصدر: European Journal of Medicinal Chemistry. 133:268-286
مصطلحات موضوعية: Blood Glucose, 0301 basic medicine, medicine.medical_specialty, Enzyme Activators, Mice, Obese, Type 2 diabetes, Hypoglycemia, 01 natural sciences, 03 medical and health sciences, Pharmacokinetics, Oral administration, Internal medicine, Glucokinase, Drug Discovery, medicine, Animals, Humans, Hypoglycemic Agents, Glucose homeostasis, Cells, Cultured, Pharmacology, 010405 organic chemistry, business.industry, Organic Chemistry, General Medicine, medicine.disease, Rats, 0104 chemical sciences, Molecular Docking Simulation, 030104 developmental biology, medicine.anatomical_structure, Endocrinology, Liver, Hyperglycemia, Hepatocyte, Pancreas, business
-
3
المؤلفون: Helen Krontiras, Venkatram R. Atigadda, Clinton J. Grubbs, Craig D. Smith, Gang Xia, Donald D. Muccio, Anil M. Deshpande, Kirby I. Bland, Wayne J. Brouillette, Lizhi Wu, Natalia Y. Kedishvili
المصدر: Journal of Medicinal Chemistry. 58:7763-7774
مصطلحات موضوعية: Molecular Conformation, Chemistry Techniques, Synthetic, Naphthalenes, Retinoid X receptor, Crystallography, X-Ray, Article, Rats, Sprague-Dawley, Structure-Activity Relationship, Breast cancer, In vivo, Drug Discovery, medicine, Animals, Anticarcinogenic Agents, Humans, Structure–activity relationship, Binding site, Triglycerides, Dyslipidemias, Binding Sites, Retinoid X Receptor alpha, Retinoid X receptor alpha, Chemistry, Mammary Neoplasms, Experimental, medicine.disease, Tamoxifen, Biochemistry, Fatty Acids, Unsaturated, Cancer research, Molecular Medicine, Female, medicine.drug
-
4
المؤلفون: Debnath Bhuniya, Rao Mukkavilli, Rahul Shivahare, Anil M. Deshpande, Ravindra T. Dere, Hari N. Pati, Vadiraj S. Gopinath, Ashok Pradhan, Manjunath Moger, Denis Martin, Suman Gupta, Preeti Vishwakarma, Delphine Launay, Aditya Verma, Sunil K. Puri
المصدر: European Journal of Medicinal Chemistry. 102:582-593
مصطلحات موضوعية: Male, Cell Survival, Antiprotozoal Agents, Administration, Oral, Pharmacology, KB Cells, Compound 32, Cell Line, Mice, Structure-Activity Relationship, Parasitic Sensitivity Tests, Pharmacokinetics, In vivo, Oral administration, Drug Discovery, Animals, Humans, Potency, Structure–activity relationship, Leishmaniasis, IC50, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, General Medicine, Hit to lead, Thiazoles, Leishmania donovani
-
5
المؤلفون: Rahul D. Kaduskar, Dinesh A. Barawkar, Debnath Bhuniya, Anil M. Deshpande, Sachin Kandalkar, Parimi Atchuta Ramaiah
المصدر: Tetrahedron Letters. 54:414-418
مصطلحات موضوعية: Pyridazine, chemistry.chemical_compound, chemistry, Organic Chemistry, Drug Discovery, chemistry.chemical_element, Staudinger reaction, Azide, Carboxylate, Biochemistry, Combinatorial chemistry, Nitrogen, Amination
-
6
المؤلفون: Mahesh Kumar Mone, Summon Koul, Sophie Roy, Anil M. Deshpande, Sachin Kandalkar, Ravi P. Nargund, Jayasagar Gundu, Anita Chugh, Michael P. Graziano, Doris F. Cully, Tian-Quan Cai, Prasun K. Chakravarty, Samir Vyas, Sheo B. Singh, Joseph P. Vacca, Umesh Prasad Singh, Pradeep Rangrao Patil, Ashwin Meru, Dinesh A. Barawkar, Goraksha Khose, Shubhangi Bhosale, Anish Bandyopadhyay, Venkata P. Palle, Kasim A. Mookhtiar, Samuel D. Wright, Siddhartha De
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:4341-4347
مصطلحات موضوعية: Candidate gene, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Carboxylic Acids, Drug Evaluation, Preclinical, Pharmaceutical Science, Thiophenes, Pyrazole, Kidney, Biochemistry, Gene product, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Structure–activity relationship, Computer Simulation, Enzyme Inhibitors, Binding site, Molecular Biology, chemistry.chemical_classification, Oxidase test, Binding Sites, Organic Chemistry, Kidney metabolism, Protein Structure, Tertiary, Rats, Alcohol Oxidoreductases, Liver, chemistry, Pyrazoles, Molecular Medicine
-
7
المؤلفون: Wayne J. Brouillette, Clinton J. Grubbs, Konstantin Christov, Isao Eto, Anil M. Deshpande, Kirby I. Bland, Vivek Tirmal, Donald D. Muccio, Venkatram R. Atigadda, Ronald A. Lubet, Gang Xia
المصدر: Carcinogenesis. 27:1232-1239
مصطلحات موضوعية: Agonist, Cancer Research, medicine.medical_specialty, medicine.drug_class, Molecular Conformation, Mammary Neoplasms, Animal, Biology, Retinoid X receptor, Rats, Sprague-Dawley, Retinoids, In vivo, Internal medicine, Biomarkers, Tumor, medicine, Animals, Anticarcinogenic Agents, Retinoid, Receptor, Triglycerides, Retinoid X Receptor alpha, Cell growth, Cancer, General Medicine, medicine.disease, Lipids, Protein Structure, Tertiary, Rats, Endocrinology, Models, Chemical, Apoptosis, Female
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::45090645bcf6c37da004e5f4a53851b5
https://doi.org/10.1093/carcin/bgi308 -
8
المؤلفون: Joseph Eckman, Narshinha P. Argade, Anil M. Deshpande, Arvind A. Natu
المصدر: Bioorganic & Medicinal Chemistry. 7:1237-1240
مصطلحات موضوعية: Stereochemistry, Leukotriene B4, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, In vitro, chemistry.chemical_compound, chemistry, Drug Discovery, Molecular Medicine, Molecular Biology, IC50, Lead compound, Enone, Naphthalene, Whole blood
-
9
المؤلفون: Parimi Atchuta Ramaiah, Rahul D. Kaduskar, Dinesh A. Barawkar, Anil M. Deshpande, Sachin Kandalkar, Debnath Bhuniya
المصدر: ChemInform. 44
مصطلحات موضوعية: chemistry.chemical_compound, Hydrolysis, Chemistry, Amino derivatives, Organic chemistry, chemistry.chemical_element, General Medicine, Carboxylate, Staudinger reaction, Nitrogen, Amination
-
10
المؤلفون: Narshinha P. Argade, Anil M. Deshpande, Arvind A. Natu
المصدر: Synthesis. 2002:1010-1012
مصطلحات موضوعية: chemistry.chemical_classification, Aqueous solution, Organic Chemistry, Closure (topology), Maleic anhydride, Ring (chemistry), Medicinal chemistry, Catalysis, chemistry.chemical_compound, Dicarboxylic acid, chemistry, Furan, Intramolecular force, Hydroxymethyl
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::851be02904d384fa83371a8bf38c358d
https://doi.org/10.1055/s-2002-31967