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1
المؤلفون: Elisabetta Armani, Andrea Rizzi, Nicolò Iotti, Francesca Saccani, Maria Rosaria Di Lascia, Laura Tigli, Alice Pappani, Gessica Marchini, Annalisa Murgo, Anna Maria Capelli, Maurizio Delcanale, Paola Puccini, Gino Villetti, Maurizio Civelli, Claudia Beato, Marta Giuliani, Claudia Mundi, Francesca Murarolli, Mafalda Pagano, Luca F. Raveglia, Rosaria Remelli, Gabriele Amari
المصدر: Journal of Medicinal Chemistry. 66:5622-5656
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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2
المؤلفون: Valentina Mileo, Anna Maria Capelli, Daniela Miglietta, P. Ronchi, Cataldo Martucci, Maurizio Civelli, Paola Maria Gallo, Matteo Biagetti, Silvia Capacchi, Serena Bertolini, A. Fioni, Gino Villetti
المصدر: C60. ASTHMA: CELLULAR AND ANIMAL MODELS.
مصطلحات موضوعية: Delta, Lung, medicine.anatomical_structure, medicine.drug_class, business.industry, Immunology, medicine, Inflammation, Rodent model, medicine.symptom, business, Anti-inflammatory, PI3K/AKT/mTOR pathway
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4496f1cc3a28786e699e4e0d2de45a32
https://doi.org/10.1164/ajrccm-conference.2020.201.1_meetingabstracts.a5614 -
3
المؤلفون: Alessandro Fioni, Anna Maria Capelli, Chiara Carnini, Gessica Marchini, Fabio Rancati, Valentina Cenacchi, Eleonora Ghidini, Fabrizio Facchinetti
المصدر: Journal of medicinal chemistry. 61(11)
مصطلحات موضوعية: Agonist, Budesonide, medicine.drug_class, Protein Conformation, Drug design, CHO Cells, Pharmacology, 01 natural sciences, 03 medical and health sciences, Mice, 0302 clinical medicine, Cricetulus, Receptors, Glucocorticoid, In vivo, Adrenal Cortex Hormones, Drug Discovery, Administration, Inhalation, medicine, Animals, Humans, Tissue Distribution, Receptor, Asthma, Lung, Inhalation, 010405 organic chemistry, Chemistry, Pneumonia, medicine.disease, 0104 chemical sciences, Molecular Docking Simulation, medicine.anatomical_structure, RAW 264.7 Cells, 030220 oncology & carcinogenesis, Drug Design, Molecular Medicine, medicine.drug
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4
المؤلفون: Fabrizio Facchinetti, Eleonora Ghidini, Valentina Cenacchi, Anna Maria Capelli, A. Virdis, A. Italia, Chiara Carnini, Gessica Marchini
المصدر: Steroids. 95:88-95
مصطلحات موضوعية: Lipopolysaccharides, Male, Transcriptional Activation, Ovalbumin, medicine.drug_class, Administration, Topical, Prednisolone, Myocytes, Smooth Muscle, Clinical Biochemistry, Active Transport, Cell Nucleus, Anti-Inflammatory Agents, Pharmacology, Nitric Oxide, Biochemistry, Anti-inflammatory, Cell Line, Mice, Receptors, Glucocorticoid, Endocrinology, Glucocorticoid receptor, Pharmacokinetics, Drug Discovery, Eosinophilia, medicine, Animals, Humans, Potency, Lung, Molecular Biology, Dexamethasone, Cell Nucleus, Dose-Response Relationship, Drug, Tumor Necrosis Factor-alpha, Chemistry, Macrophages, Interleukin-8, Organic Chemistry, Isoxazoles, Protein Structure, Tertiary, Rats, Molecular Docking Simulation, Receptors, Mineralocorticoid, medicine.anatomical_structure, Corticosteroid, Transcription Factors, medicine.drug
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المؤلفون: Gabriele Costantino, Anna Maria Capelli
المصدر: Journal of Chemical Information and Modeling. 54:3124-3136
مصطلحات موضوعية: Sorafenib, Indoles, General Chemical Engineering, VEGF receptors, Molecular Dynamics Simulation, Library and Information Sciences, urologic and male genital diseases, Molecular dynamics, Catalytic Domain, Sunitinib, medicine, Humans, Pyrroles, Binding site, Protein Kinase Inhibitors, chemistry.chemical_classification, biology, Chemistry, General Chemistry, Vascular Endothelial Growth Factor Receptor-2, female genital diseases and pregnancy complications, Computer Science Applications, Enzyme, biology.protein, Biophysics, medicine.drug
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المؤلفون: Paola Maria Gallo, Fabrizio Facchinetti, Mauro Corsi, Filippo Visentini, Daniele Pala, Matteo Biagetti, Marco Mor, Alice Pappani, Serena Bertolini, Anna Maria Capelli, Silvia Capacchi, Silvia Rivara, Alessio Lodola
المصدر: Journal of medicinal chemistry. 60(10)
مصطلحات موضوعية: Steric effects, Models, Molecular, Molecular model, Stereochemistry, 010402 general chemistry, 01 natural sciences, chemistry.chemical_compound, Mice, Isomerism, Drug Discovery, Animals, Humans, Methylene, Conformational isomerism, Protein Kinase Inhibitors, Phosphoinositide-3 Kinase Inhibitors, Atropisomer, 010405 organic chemistry, Adenine, Biological activity, 0104 chemical sciences, Class Ia Phosphatidylinositol 3-Kinase, chemistry, Axial chirality, Quinazolines, Molecular Medicine, Methyl group
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المؤلفون: Alessio Lodola, Silvia Rivara, Marco Mor, Donatella Callegari, Daniele Pala, Anna Maria Capelli, Andrea Rizzi
المصدر: Journal of chemical information and modeling. 57(2)
مصطلحات موضوعية: 0301 basic medicine, Time Factors, 010304 chemical physics, Drug discovery, Chemistry, Protein Conformation, General Chemical Engineering, Metadynamics, General Chemistry, Library and Information Sciences, Molecular Dynamics Simulation, Cyclin-Dependent Kinase 8, 01 natural sciences, Computer Science Applications, 03 medical and health sciences, 030104 developmental biology, 0103 physical sciences, Cyclin-dependent kinase 8, Collective variables, Thermodynamics, Poor correlation, Biological system, Residence time (statistics), Protein Kinase Inhibitors, Simulation
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8
المصدر: Journal of Medicinal Chemistry. 56:7003-7014
مصطلحات موضوعية: Models, Molecular, medicine.medical_specialty, Chemistry, medicine.medical_treatment, Mutant, Endogeny, Molecular Dynamics Simulation, Ligands, Steroid, Cell biology, Receptors, Glucocorticoid, Glucocorticoid receptor, Endocrinology, Apoptosis, Internal medicine, Mutation, Drug Discovery, medicine, Molecular Medicine, Receptor, Glucocorticoids, Glucocorticoid, Hormone, medicine.drug
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المؤلفون: Federica Tonelli, Elisa Della Turca, Chiara Pecchini, Raffaele Longhi, Romano Di Fabio, Gian Paolo Vallerini, Matteo Biagetti, Dino Montanari, Angelo Giacometti, Anna Maria Capelli, Adelheid Roth, Angela Worby, Marco Mor, Emilio Merlo-Pich, Gabriele Costantino, Giorgio Bonanomi, Fabrizio Micheli, Luca Tarsi
المصدر: ResearcherID
مصطلحات موضوعية: medicine.medical_specialty, Class (set theory), Endocrinology, Chemistry, Stereochemistry, Internal medicine, Drug Discovery, Neuropeptide S, medicine, Pharmaceutical Science, Molecular Medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cd7e266038edffa0e59e037a0182f502
https://doi.org/10.2174/1570180811310050005 -
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المؤلفون: Anna Maria Capelli, Fabrizio Micheli
المصدر: Pharmaceutical Patent Analyst. 1:469-481
مصطلحات موضوعية: Cyclopropanes, biology, Chemistry, General Medicine, Pharmacology, Heptanes, Tryptamines, Reuptake, Norepinephrine, Monoamine neurotransmitter, Norepinephrine transporter, Dopamine, Monoaminergic, medicine, biology.protein, Animals, Hexanes, Humans, Neurotransmitter Uptake Inhibitors, Reuptake inhibitor, Cyclobutanes, Tropanes, medicine.drug