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1دورية أكاديمية
المؤلفون: Nadia M J Rupniak, Elisabetta Perdona, Cristiana Griffante, Palmina Cavallini, Anna Sava, Daniel J Ricca, Karl B Thor, Edward C Burgard, Mauro Corsi
المصدر: PLoS ONE, Vol 13, Iss 10, p e0205894 (2018)
وصف الملف: electronic resource
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المؤلفون: Peng Gao, Paolo Vincetti, Fabio Maria Sabbatini, Holly J. Carlisle, Luisa Mengatto, Stéphane De Lombaert, Anna Sava, Kerry Zobel, Xinying Liu, Claudia Beato, Jessica M. Bright, Alyssa M. A. Toda, Elena Serra, Federica Budassi, Marco Migliore, Laura Caberlotto, Cristiana Griffante, Silvia Bernardi, Mingliang Zhang, Albert W. Garofalo, Daniele Andreotti
المصدر: Journal of Medicinal Chemistry. 63:14821-14839
مصطلحات موضوعية: Indazoles, Tetrazoles, Leucine-Rich Repeat Serine-Threonine Protein Kinase-2, 01 natural sciences, Small Molecule Libraries, Mice, Structure-Activity Relationship, 03 medical and health sciences, Drug Discovery, Animals, Humans, Kinase activity, Protein Kinase Inhibitors, Gene, 030304 developmental biology, 0303 health sciences, Molecular Structure, Chemistry, Kinase, Highly selective, LRRK2, High-Throughput Screening Assays, nervous system diseases, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, HEK293 Cells, Pyrimidines, Mutation, Cancer research, Molecular Medicine
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المؤلفون: Aldo Feriani, Laura Zonzini, Laura Castelletti, Selena Nola, Michele Dal Cin, Teresa Semeraro, Sylvie Gehanne, Silvia Tomelleri, Filippo Visentini, Palmina Cavallini, Susanna Cremonesi, Annalisa Pellacani, Anna Sava, Alessia Bacchi, Andrea Wong, Simone Braggio, Luca Tarsi, Mahmud Kajbaf, Paolo Cavanni, Elisabetta Perdona, Christian Heidbreder, Luciano Marchiò, Beatrice Oliosi, Fabrizio Micheli
المصدر: Journal of Medicinal Chemistry. 59:8549-8576
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Stereochemistry, hERG, CHO Cells, Crystallography, X-Ray, 030226 pharmacology & pharmacy, Heptanes, Structure-Activity Relationship, 03 medical and health sciences, Cricetulus, 0302 clinical medicine, In vivo, Dopamine receptor D3, Dopamine, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Spiro Compounds, biology, Chemistry, Receptors, Dopamine D3, Triazoles, biology.organism_classification, Ether-A-Go-Go Potassium Channels, In vitro, 030104 developmental biology, biology.protein, Molecular Medicine, Selectivity, medicine.drug
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المؤلفون: Nadia M.J. Rupniak, Cristiana Griffante, Mauro Corsi, Palmina Cavallini, Karl B. Thor, Anna Sava, Elisabetta Perdona, Daniel J. Ricca
المصدر: Neurosci Lett
مصطلحات موضوعية: 0301 basic medicine, Agonist, medicine.drug_class, chemistry.chemical_element, CHO Cells, Calcium, Article, law.invention, 03 medical and health sciences, 0302 clinical medicine, Cricetulus, law, medicine, Potency, Animals, Humans, Receptor, AMP synthesis, General Neuroscience, Receptors, Neurokinin-2, Receptors, Neurokinin-1, Recombinant Proteins, 030104 developmental biology, chemistry, Biochemistry, Cell culture, Recombinant DNA, Selectivity, 030217 neurology & neurosurgery
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المؤلفون: Anna Sava, Palmina Cavallini, Daniel J. Ricca, Nadia M.J. Rupniak, Mauro Corsi, Elisabetta Perdona, Edward C. Burgard, Karl B. Thor, Cristiana Griffante
المصدر: PLoS ONE, Vol 13, Iss 10, p e0205894 (2018)
PLoS ONEمصطلحات موضوعية: Neurokinin A, Drug Evaluation, Preclinical, Receptor agonist activity, lcsh:Medicine, Stimulation, Peptide, Biochemistry, Intracellular Receptors, chemistry.chemical_compound, Binding Analysis, 0302 clinical medicine, Cell Signaling, Cricetinae, Cyclic AMP, Membrane Receptor Signaling, Receptor, lcsh:Science, chemistry.chemical_classification, Multidisciplinary, integumentary system, Chemistry, Chinese hamster ovary cell, hemic and immune systems, Receptors, Neurokinin-2, Receptors, Neurokinin-1, respiratory system, Recombinant Proteins, Enzymes, Optical Equipment, 030220 oncology & carcinogenesis, Cell lines, Engineering and Technology, Biological cultures, Oxidoreductases, Luciferase, Research Article, Signal Transduction, Cell Binding, Cell Physiology, Equipment, CHO Cells, Research and Analysis Methods, 03 medical and health sciences, Cricetulus, Potency, Animals, Humans, Receptor Binding Assays, Chemical Characterization, EC50, Dose-Response Relationship, Drug, Cell Membrane, lcsh:R, Biology and Life Sciences, Proteins, Reproducibility of Results, Prisms, Cell Biology, Molecular biology, Enzymology, Calcium, lcsh:Q, Peptides, 030217 neurology & neurosurgery
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المؤلفون: Kay Maltby, Stuart J Mundell, Edward T. Bullmore, Anna Sava, Graeme Henderson, Adelheid Roth, Eamonn Kelly, Antonio Felici, Pradeep J. Nathan
المصدر: Psychopharmacology
مصطلحات موضوعية: Pharmacology, GSK1521498, Binge eating, Receptor pharmacology, medicine.drug_class, Antagonist, μ-Opioid receptor, (+)-Naloxone, Differential effects, Naltrexone, Opioid receptor, Inverse agonism, medicine, medicine.symptom, Psychology, Nalmefene, medicine.drug, Original Investigation
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المؤلفون: Anna Sava, Luca Tarsi, Simone Braggio, Teresa Semeraro, Aldo Feriani, Laura Zonzini, Fabrizio Micheli, Beatrice Oliosi, Susanna Cremonesi, Elisabetta Perdona, Silvia Tomelleri, Paolo Cavanni, Christian Heidbreder
المصدر: Bioorganicmedicinal chemistry letters. 26(4)
مصطلحات موضوعية: 0301 basic medicine, Morpholines, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, 01 natural sciences, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Dopamine receptor D1, Dopamine receptor D3, Dopamine, Morpholine, Dopamine receptor D2, Drug Discovery, Enzyme-linked receptor, medicine, Animals, Molecular Biology, Binding Sites, 010405 organic chemistry, Chemistry, Organic Chemistry, Antagonist, Receptors, Dopamine D3, In vitro, 0104 chemical sciences, Protein Structure, Tertiary, Rats, Molecular Docking Simulation, Dopamine D2 Receptor Antagonists, 030104 developmental biology, Molecular Medicine, medicine.drug, Half-Life
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المؤلفون: Ilaria Sartori, Laura Zonzini, Laurie J. Gordon, Angela Worby, Stefano Fontana, Manuela Borriello, Silvia Bison, Jeannette M. Watson, Steven Mark Bromidge, Giovanna Dal Forno, Colin Philip Leslie, Alessandra Pasquarello, Anna Sava, Luca G. Moccia, Barbara Bertani, Roberto Arban, Daniele Donati, Enrica Granci, Valeria Zucchelli, Paolo Cavanni, Massimo Gianotti, Romano Di-Fabio
المصدر: Journal of Medicinal Chemistry. 53:5827-5843
مصطلحات موضوعية: chemistry.chemical_classification, biology, medicine.drug_class, Stereochemistry, Benzoxazinones, hERG, Carboxamide, Receptor antagonist, chemistry, In vivo, Drug Discovery, medicine, biology.protein, Molecular Medicine, Receptor, Serotonin transporter, Tricyclic
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المؤلفون: Stephen P. Watson, Adelheid Roth, Anna Sava, Greg J. Osborne, David John Nash, Paloma Perez, Ben Powney, Corrado Corti, Magalie Rocheville, Paul W. Smith, Clive Leslie Branch, Federica Bianchi, Pier D’Alessandro, Emma Koppe, Maite de los Frailes, Jesús Ángel de la Fuente, Annarosa Ugolini, Dino Montanari, Stephen L. Garland
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:759-762
مصطلحات موضوعية: Dopamine, High-throughput screening, Clinical Biochemistry, Allosteric regulation, Administration, Oral, Pharmaceutical Science, Receptors, Metabotropic Glutamate, Biochemistry, Piperazines, Structure-Activity Relationship, Allosteric Regulation, Oral administration, Drug Discovery, Animals, Structure–activity relationship, Molecular Biology, Chemistry, Organic Chemistry, Dopaminergic, Long-term potentiation, Synaptic Potentials, High-Throughput Screening Assays, Rats, Metabotropic glutamate receptor, Molecular Medicine, Benzimidazoles, Metabotropic glutamate receptor 2
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المصدر: Neuroscience Letters. 313:37-40
مصطلحات موضوعية: animal structures, Muscle Fibers, Skeletal, Neuromuscular Junction, Protein tyrosine phosphatase, Receptors, Nicotinic, Receptor tyrosine kinase, Neuromuscular junction, Iodine Radioisotopes, Rats, Sprague-Dawley, Radioligand Assay, chemistry.chemical_compound, medicine, Animals, Biotinylation, Enzyme Inhibitors, Phosphorylation, Tyrosine, Phosphotyrosine, Cells, Cultured, Cytoskeleton, Acetylcholine receptor, biology, General Neuroscience, Tyrosine phosphorylation, Bungarotoxins, musculoskeletal system, Rats, Cell biology, Nicotinic acetylcholine receptor, medicine.anatomical_structure, Biochemistry, chemistry, biology.protein, Protein Tyrosine Phosphatases, Vanadates