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المؤلفون: Eric Legangneux, Srikanth Neelakantham, Anne Gardin, Kasra Shakeri-Nejad, Cathy Gray, Swati Dumitras
المصدر: Clinical Therapeutics. 42:175-195
مصطلحات موضوعية: Adult, Male, Sphingosine 1 Phosphate Receptor Modulators, medicine.medical_specialty, Administration, Oral, Biological Availability, 02 engineering and technology, 030204 cardiovascular system & hematology, Asymptomatic, Gastroenterology, Young Adult, 03 medical and health sciences, chemistry.chemical_compound, 020210 optoelectronics & photonics, 0302 clinical medicine, Pharmacokinetics, Heart Rate, Internal medicine, Benzyl Compounds, Heart rate, 0202 electrical engineering, electronic engineering, information engineering, medicine, Humans, Pharmacology (medical), Lymphocyte Count, Dosing, Infusions, Intravenous, Pharmacology, business.industry, Middle Aged, Healthy Volunteers, Regimen, Siponimod, Tolerability, chemistry, Pharmacodynamics, Azetidines, Female, medicine.symptom, business
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المؤلفون: Bettina Rudolph, Anna Schubart, Emmanuelle Briard, Florian Muellershausen, Erwin Hermes, Andreas Hofmann, Marc Bigaud, Anne Gardin, Christian Beerli
المصدر: Multiple Sclerosis Journal-Experimental, Translational and Clinical
مصطلحات موضوعية: Agonist, Cerebellum, medicine.drug_class, business.industry, CNS penetration, Central nervous system, Pharmacology, Siponimod, and single-photon emission computed tomography, Olfactory bulb, White matter, Cellular and Molecular Neuroscience, chemistry.chemical_compound, medicine.anatomical_structure, chemistry, rodents, medicine, Medulla oblongata, Distribution (pharmacology), Neurology (clinical), Original Research Article, non-human primates, quantitative whole-body autoradiography, business
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المؤلفون: Anne Gardin, Handan He, Felix Huth, Kenichi Umehara
المصدر: Clinical Pharmacology and Therapeutics
مصطلحات موضوعية: Drug, Physiologically based pharmacokinetic modelling, Cytochrome P-450 CYP2C9 Inhibitors, Genotype, media_common.quotation_subject, Pharmacology, Models, Biological, 030226 pharmacology & pharmacy, Article, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Benzyl Compounds, Cytochrome P-450 Enzyme Inhibitors, Humans, Computer Simulation, Drug Interactions, Pharmacology (medical), CYP2C9, Cytochrome P-450 CYP2C9, media_common, Cytochrome P-450 Enzyme Inducers, CYP3A4, Chemistry, Research, Area under the curve, Cytochrome P-450 CYP3A Inducers, Articles, Drug interaction, Siponimod, Area Under Curve, 030220 oncology & carcinogenesis, Azetidines, Cytochrome P-450 CYP3A Inhibitors, Rifampin, Half-Life
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المؤلفون: Anne Gardin, Swati Dumitras, Srikanth Neelakantham, Felix Huth, Andrea Feller, Kasra Shakeri-Nejad
المصدر: European Journal of Clinical Pharmacology. 75:1565-1574
مصطلحات موضوعية: Adult, Male, Sphingosine 1 Phosphate Receptor Modulators, medicine.medical_specialty, Adolescent, Genotype, Itraconazole, Cmax, 030226 pharmacology & pharmacy, Gastroenterology, Electrocardiography, Young Adult, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Internal medicine, Benzyl Compounds, medicine, Cytochrome P-450 CYP3A, Humans, Drug Interactions, Pharmacology (medical), Lymphocyte Count, 030212 general & internal medicine, Adverse effect, CYP2C9, Cytochrome P-450 CYP2C9, Pharmacology, business.industry, General Medicine, Middle Aged, Healthy Volunteers, Siponimod, Tolerability, chemistry, Area Under Curve, Cohort, Azetidines, Cytochrome P-450 CYP3A Inhibitors, Female, business, medicine.drug
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المصدر: Psychopharmacology
مصطلحات موضوعية: Ozanimod, Sphingosine 1 Phosphate Receptor Modulators, medicine.medical_specialty, Multiple Sclerosis, medicine.medical_treatment, Physical dependence, Review, Siponimod, Abuse, chemistry.chemical_compound, Clinical, Sphingosine, medicine, media_common.cataloged_instance, Animals, Humans, S1P receptor modulator, European union, Psychiatry, Adverse effect, Dependence, media_common, Pharmacology, business.industry, Non-clinical, Fingolimod, Stimulant, chemistry, Ponesimod, medicine.symptom, Lysophospholipids, business, medicine.drug
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المؤلفون: Anne Gardin, Felix Huth, Antonia M Davidson, Eric Legangneux, Kasra Shakeri-Nejad, Cathy Gray, Swati Dumitras, Srikanth Neelakantham
المصدر: European Journal of Clinical Pharmacology. 74:1593-1604
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Adolescent, Cmax, 030226 pharmacology & pharmacy, Gastroenterology, Young Adult, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Internal medicine, Benzyl Compounds, medicine, Humans, Drug Interactions, Pharmacology (medical), Inducer, Lymphocyte Count, CYP2C9, Biotransformation, Cytochrome P-450 CYP2C9, Pharmacology, business.industry, Area under the curve, General Medicine, Healthy Volunteers, Receptors, Lysosphingolipid, Siponimod, chemistry, Tolerability, Area Under Curve, Enzyme Induction, Azetidines, Female, Rifampin, Geometric mean, business, 030217 neurology & neurosurgery
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المؤلفون: Axel Meissner, Ulrike Glaenzel, Gian Camenisch, Eric Legangneux, Sjoerd Peter van Marle, Hubert Borell, Robert Nufer, Kirsten Schroer, Alexander David James, Yi Jin, Wenkui Li, Sylvie Adam-Stitah, Anne Gardin
المصدر: Drug Metabolism and Disposition. 46:1001-1013
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, biology, CYP3A4, Metabolite, Glucuronidation, Pharmaceutical Science, Cytochrome P450, Metabolism, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Siponimod, chemistry, Microsome, biology.protein, 030217 neurology & neurosurgery, ADME
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::03d15a91303385d4488bb9542e37609d
https://doi.org/10.1124/dmd.117.079574 -
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المؤلفون: Srikanth Neelakantham, Xuemei Tan, Kasra Shakeri-Nejad, Angela Dodman, Eric Legangneux, Sampath Kalluri, Anne Gardin
المصدر: Int. Journal of Clinical Pharmacology and Therapeutics. 55:54-65
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Adolescent, Cmax, Administration, Oral, 02 engineering and technology, Severity of Illness Index, Gastroenterology, Young Adult, 03 medical and health sciences, chemistry.chemical_compound, 020210 optoelectronics & photonics, 0302 clinical medicine, Pharmacokinetics, Internal medicine, Benzyl Compounds, 0202 electrical engineering, electronic engineering, information engineering, Humans, Medicine, Pharmacology (medical), Renal Insufficiency, Adverse effect, Aged, Pharmacology, business.industry, Area under the curve, Half-life, Middle Aged, Interim analysis, Receptors, Lysosphingolipid, Siponimod, Tolerability, chemistry, Area Under Curve, Azetidines, Female, business, 030217 neurology & neurosurgery, Half-Life
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9
المؤلفون: Gianluca Rossato, Parasar Pal, Zhenzhong Su, Yi Jin, Eric Legangneux, Kasra Shakeri-Nejad, Mike Ufer, Anne Gardin, Wenkui Li
المصدر: Clinical Pharmacokinetics
مصطلحات موضوعية: Adult, Male, Sphingosine 1 Phosphate Receptor Modulators, Adolescent, Cytochrome P-450 CYP2C9 Inhibitors, Genotype, CYP3A, Cmax, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, chemistry.chemical_compound, Young Adult, 0302 clinical medicine, Pharmacokinetics, Benzyl Compounds, medicine, Humans, Pharmacology (medical), Drug Interactions, Original Research Article, CYP2C9, Fluconazole, Cytochrome P-450 CYP2C9, Polymorphism, Genetic, business.industry, Area under the curve, Middle Aged, Healthy Volunteers, Siponimod, chemistry, Tolerability, Azetidines, Cytochrome P-450 CYP3A Inhibitors, Drug Therapy, Combination, Female, business, 030217 neurology & neurosurgery, medicine.drug
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