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1دورية أكاديمية
المؤلفون: Helena Pérez-Peña, Anne-Catherine Abel, Maxim Shevelev, Andrea E. Prota, Stefano Pieraccini, Dragos Horvath
المصدر: Biomolecules, Vol 13, Iss 2, p 285 (2023)
مصطلحات موضوعية: computer-aided drug design, microtubules, microtubule targeting agents, virtual screening, molecular docking, molecular dynamics simulations, Microbiology, QR1-502
وصف الملف: electronic resource
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2
المؤلفون: Giorgio Facchetti, Jaime Gracia Vitoria, Martina Moraschi, Raffaella Bucci, Anne Catherine Abel, Stefano Pieraccini, Sara Pellegrino, Isabella Rimoldi
المصدر: European Journal of Organic Chemistry. 26
مصطلحات موضوعية: Organic Chemistry, Physical and Theoretical Chemistry
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3
المؤلفون: Zlata Boiarska, Helena Pérez‐Peña, Anne‐Catherine Abel, Paola Marzullo, Beatriz Álvarez‐Bernad, Francesca Bonato, Benedetta Santini, Dragos Horvath, Daniel Lucena‐Agell, Francesca Vasile, Maurizio Sironi, J. Fernando Díaz, Andrea E. Prota, Stefano Pieraccini, Daniele Passarella
المساهمون: European Commission, Ministerio de Ciencia e Innovación (España), Boiarska, Zlata, Abel, Anne-Catherine, Marzullo, Paola, Álvarez-Bernad, Beatriz, Bonato, Francesca, Horvath, Dragos, Lucena-Agell, Daniel, Vasile, Francesca, Sironi, Maurizio, Díaz, José Fernando, Prota, Andrea E., Pieraccini, Stefano, Passarella, D.
المصدر: Chemistry – A European Journal. 29
مصطلحات موضوعية: microtubules, chemical probes, tubulin, maytansinol functionalization, Organic Chemistry, Settore CHIM/06 - Chimica Organica, General Chemistry, maytansinoids, Catalysis
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4
المؤلفون: Zlata Boiarska, Helena Pérez‐Peña, Anne‐Catherine Abel, Paola Marzullo, Beatriz Álvarez‐Bernad, Francesca Bonato, Benedetta Santini, Dragos Horvath, Daniel Lucena‐Agell, Francesca Vasile, Maurizio Sironi, J. Fernando Díaz, Andrea E. Prota, Stefano Pieraccini, Daniele Passarella
المصدر: Chemistry – A European Journal. 29
مصطلحات موضوعية: Organic Chemistry, General Chemistry, Catalysis
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5
المؤلفون: Marilia, Barreca, Virginia, Spanò, Roberta, Rocca, Roberta, Bivacqua, Anne-Catherine, Abel, Annalisa, Maruca, Alessandra, Montalbano, Maria Valeria, Raimondi, Chiara, Tarantelli, Eugenio, Gaudio, Luciano, Cascione, Andrea, Rinaldi, Ruoli, Bai, Michel O, Steinmetz, Andrea E, Prota, Stefano, Alcaro, Ernest, Hamel, Francesco, Bertoni, Paola, Barraja
المساهمون: Barreca M., Spano' V., Rocca R., Bivacqua R., Abel A.-C., Maruca A., Montalbano A., Raimondi M.V., Tarantelli C., Gaudio E., Cascione L., Rinaldi A., Bai R., Steinmetz M.O., Prota A.E., Alcaro S., Hamel E., Bertoni F., Barraja P.
المصدر: European Journal of Medicinal Chemistry. 243:114744
مصطلحات موضوعية: Pharmacology, Binding Sites, Lymphoma, Antitubulin agents, Colchicine site, Organic Chemistry, Antineoplastic Agents, General Medicine, Isoindoles, Tubulin Modulators, T2R-TTL–Complexes, Structure-Activity Relationship, Tubulin, Neoplasms, Cell Line, Tumor, Drug Discovery, Humans, [1,2]oxazolo[5,4-e]isoindoles, Colchicine, X-ray crystallography
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6
المؤلفون: Paola Marzullo, Zlata Boiarska, Helena Pérez‐Peña, Anne‐Catherine Abel, Beatriz Álvarez‐Bernad, Daniel Lucena‐Agell, Francesca Vasile, Maurizio Sironi, Karl‐Heinz Altmann, Andrea E. Prota, J. Fernando Díaz, Stefano Pieraccini, Daniele Passarella
المصدر: Chemistry – A European Journal. 28
مصطلحات موضوعية: Organic Chemistry, General Chemistry, Catalysis
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7
المؤلفون: Paola Marzullo, Maurizio Sironi, Daniel Lucena-Agell, J. Fernando Díaz, Daniele Passarella, Helena Pérez-Peña, Zlata Boiarska, Stefano Pieraccini, Beatriz Álvarez-Bernad, Anne-Catherine Abel, Karl-Heinz Altmann, Andrea E. Prota, Francesca Vasile
المساهمون: European Commission, Ministerio de Ciencia e Innovación (España), Consejo Superior de Investigaciones Científicas (España), Fundación Tatiana Pérez de Guzmán el Bueno, Università degli Studi di Milano, Marzullo, Paola, Boiarska, Zlata, Abel, Anne-Catherine, Álvarez-Bernad, Beatriz, Lucena-Agell, Daniel, Vasile, Francesca, Sironi, Maurizio, Altmann, Karl-Heinz, Prota, Andrea E., Díaz, José Fernando, Pieraccini, Stefano, Passarella, D., Marzullo, Paola [0000-0003-4249-8794], Boiarska, Zlata [0000-0003-1235-5717], Abel, Anne-Catherine [0000-0002-2392-9029], Álvarez-Bernad, Beatriz [0000-0002-2492-9215], Lucena-Agell, Daniel [0000-0001-7198-2900], Vasile, Francesca [0000-0002-3926-8261], Sironi, Maurizio [0000-0001-5822-4849], Altmann, Karl-Heinz [0000-0002-0747-9734], Prota, Andrea E. [0000-0003-0875-5339], Díaz, José Fernando [0000-0003-2743-3319], Pieraccini, Stefano [0000-0002-7672-0720], Passarella, D. [0000-0001-6180-9581]
المصدر: Chemistry – A European Journal
Digital.CSIC. Repositorio Institucional del CSIC
instname
Chemistry-A European Journal, 28 (2)مصطلحات موضوعية: maytansine binding site, Cancer therapy, 01 natural sciences, Catalysis, microtubules, Acylation, 03 medical and health sciences, Maytansinol, Microtubule, Neoplasms, Humans, Molecule, Maytansine, 030304 developmental biology, 0303 health sciences, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, General Chemistry, maytansinol, tubulin, tubulin binders, Combinatorial chemistry, Tubulin Modulators, 0104 chemical sciences, 3. Good health, Tubulin, Docking (molecular), biology.protein
وصف الملف: application/application/pdf
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8
المؤلفون: Andrea E. Prota, Stefan D. Tomlins, Xuexin Gao, Cassandra Yong, Anne-Catherine Abel, Peter J. Scammells, Shane M. Devine, Michel O. Steinmetz, Ben Capuano, Richard Callaghan, Divya Muthiah
المصدر: ChemMedChem. 16(18)
مصطلحات موضوعية: Stereochemistry, Cell, 1,3-Benzodioxole, Antineoplastic Agents, Dioxoles, Biochemistry, Polymerization, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, 0302 clinical medicine, Tubulin, Drug Discovery, medicine, Tumor Cells, Cultured, Moiety, Humans, General Pharmacology, Toxicology and Pharmaceutics, Cytotoxicity, 030304 developmental biology, Cell Proliferation, Pharmacology, 0303 health sciences, biology, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Tubulin Modulators, 3. Good health, Noscapine, medicine.anatomical_structure, chemistry, 030220 oncology & carcinogenesis, Dioxolane, biology.protein, Molecular Medicine, Efflux, Drug Screening Assays, Antitumor, medicine.drug