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1
المؤلفون: Stefania Meini, Sandro Giuliani, Antonio Guidi, Danilo Giannotti, CarloâAlberto Maggi, Valentina Fedi, Tula Dimoulas, Franco Pasqui, Rossano Nannicini, Manuela Tramontana, Martina Gensini, Maria Altamura, NicholasâJ.âS. Harmat, Antonio Triolo
المصدر: ChemMedChem. 5:65-78
مصطلحات موضوعية: Pharmacology, Stereochemistry, Guinea Pigs, Organic Chemistry, Antagonist, Dipeptides, Receptors, Neurokinin-2, Thiophenes, Tetrahydropyran, Biochemistry, In vitro, Guinea pig, Structure-Activity Relationship, chemistry.chemical_compound, chemistry, In vivo, Drug Design, Drug Discovery, Animals, Humans, Molecular Medicine, Potency, Moiety, General Pharmacology, Toxicology and Pharmaceutics, Receptor
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2
المؤلفون: Sandro Giuliani, Maria Altamura, Carlo Alberto Maggi, Antonio Guidi, Rose-Marie Catalioto, Stefania Meini, Alessandro Giolitti, Danilo Giannotti, Nicholas J. S. Harmat, Alessandro Lecci, Franco Pasqui, and Antonio Triolo, Rossano Nannicini, Manuela Tramontana, Valentina Fedi
المصدر: Journal of Medicinal Chemistry. 50:4793-4807
مصطلحات موضوعية: Male, Colon, Stereochemistry, medicine.drug_class, Guinea Pigs, Urinary Bladder, Substituent, Administration, Oral, Carboxamide, Stereoisomerism, Cyclopentanes, Thiophenes, In Vitro Techniques, Permeability, Intestinal absorption, Injections, Radioligand Assay, chemistry.chemical_compound, Piperidines, Ileum, Drug Discovery, medicine, Animals, Humans, Moiety, Pyrans, Bicyclic molecule, Benzothiophene, Muscle, Smooth, Dipeptides, Receptors, Neurokinin-2, Middle Aged, Ligand (biochemistry), Intestinal Absorption, chemistry, Molecular Medicine, Female, Caco-2 Cells, Muscle Contraction
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3
المؤلفون: Antonio Guidi, Alessandro Giolitti, Paolo Dapporto, Patrizia Rossi, Annalisa Guerri, Valentina Fedi, Paola Paoli, Carlo Alberto Maggi, Maria Altamura
المصدر: Acta Crystallographica Section B Structural Science. 62:889-896
مصطلحات موضوعية: Models, Molecular, chemistry.chemical_classification, animal structures, Molecular Structure, Chemistry, Stereochemistry, Hydrogen Bonding, Peptide, Receptors, Neurokinin-2, General Medicine, Experimental validation, In Vitro Techniques, Crystallography, X-Ray, Peptides, Cyclic, Protein Structure, Secondary, General Biochemistry, Genetics and Molecular Biology, Feature (computer vision), Humans, Receptor, Oligopeptides
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4
المؤلفون: Cristina Nativi, Antonio Guidi, Francesco Cuda, Stefania Meini, Stefano Menichetti, Franco Pasqui, Giuseppe Balacco, Maria Altamura, Annalisa Guerri
المصدر: Tetrahedron. 62:6754-6761
مصطلحات موضوعية: chemistry.chemical_classification, Flexibility (engineering), Chemistry, Ligand, Organic Chemistry, Nuclear magnetic resonance spectroscopy, Biochemistry, Physical chemical, Drug Discovery, Thermal, Organic chemistry, Bioassay, Biological system, Thioamide
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5
المؤلفون: Paolo Dapporto, Annalisa Guerri, Francesco Cuda, Cristina Nativi, Patrizia Rossi, Maria Altamura, Antonio Guidi, Giacomo Coppini, Paola Paoli
المصدر: Journal of Molecular Structure. 749:20-30
مصطلحات موضوعية: Organic Chemistry, Solid-state, Thio, Key features, Force field (chemistry), Analytical Chemistry, Inorganic Chemistry, Phthalic acid, chemistry.chemical_compound, Crystallography, chemistry, Amide, Molecule, Crystallographic database, Spectroscopy
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6
المؤلفون: Maria Altamura, Antonio Guidi, Paola Cucchi, Carlo Alberto Maggi, Alessandro Giolitti, Claudio Catalani, Luigi Rotondaro, Franco Pasqui, Stefania Meini, Sabrina Zappitelli, Sandro Giuliani, Francesca Bellucci
المصدر: European Journal of Pharmacology. 516:104-111
مصطلحات موضوعية: Indoles, Inositol Phosphates, Morpholines, Neurokinin A, Mutation, Missense, Phthalic Acids, Gene Expression, CHO Cells, Substance P, Biology, Ligands, Tritium, Binding, Competitive, Saredutant, Iodine Radioisotopes, Radioligand Assay, Cricetulus, Piperidines, Cricetinae, medicine, Animals, Humans, Protein Isoforms, Binding site, Receptor, G protein-coupled receptor, Pharmacology, Dose-Response Relationship, Drug, Cell Membrane, Antagonist, Receptors, Neurokinin-2, Ligand (biochemistry), Biochemistry, Competitive antagonist, Benzamides, Tachykinin receptor, medicine.drug
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7كتاب إلكتروني
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8Structural investigation on three 3,5-trans disubstituted piperidines. X-ray and theoretical studies
المؤلفون: M. Altamura, Paolo Dapporto, Patrizia Rossi, Paola Paoli, F.R. Calabri, Antonio Guidi, Annalisa Guerri
المصدر: Journal of Molecular Structure: THEOCHEM. 617:189-199
مصطلحات موضوعية: Chemistry, Ab initio, Condensed Matter Physics, Ring (chemistry), Biochemistry, chemistry.chemical_compound, Ab initio quantum chemistry methods, Computational chemistry, Intramolecular force, Molecule, Nitrogen inversion, Piperidine, Physical and Theoretical Chemistry, Conformational isomerism
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9
المؤلفون: Anna Rita Renzetti, Silvia Valenza, Franca M. Cordero, Alessandro Giolitti, Maria Altamura, Alberto Brandi, Francesca Giuntini, Antonio Guidi, Franco Pasqui, Carlo Alberto Maggi
المصدر: The Journal of Organic Chemistry. 65:4003-4008
مصطلحات موضوعية: Models, Molecular, chemistry.chemical_classification, Chemistry, Stereochemistry, Peptidomimetic, Organic Chemistry, Molecular Conformation, Substituent, Regioselectivity, Dipeptides, Receptors, Neurokinin-2, Ligands, Cycloaddition, Nitrone, Structure-Activity Relationship, chemistry.chemical_compound, Tachykinins, Peptide synthesis, Humans, Indicators and Reagents, Nitrogen Oxides, Stereoselectivity, Receptor
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10
المؤلفون: Gloria Menchi, Ernesto G. Occhiato, Fabrizio Machetti, Trabocch A, Sauro Sisi, Dina Scarpi, Antonio Guidi, Antonio Guarna
المصدر: The Journal of Organic Chemistry. 64:7347-7364
مصطلحات موضوعية: chemistry.chemical_classification, Dipeptide, Stereochemistry, Carboxylic acid, Organic Chemistry, Diastereomer, Alpha (ethology), Amino acid, chemistry.chemical_compound, Enantiopure drug, chemistry, Glycine, Tartaric acid, Moiety, Reactivity (chemistry)