-
1
المؤلفون: Marc L. Reitman, Cheng Guo, Theresa M. Kelly, Constantin Tamvakopoulos, Joseph M. Metzger, Tianying Jian, Howard Y. Chen, Arthur A. Patchett, Oksana C. Palyha, Alison M. Strack, Allan J. Goodman, Ravi P. Nargund, Peter H. Dobbelaar, Yanqing Kan, Mark Hadden, Larry Yet, Peter R. Guzzo, Qianping Peng, Linus S. Lin, Shuwen He, Lauren P. Shearman, Alan J. Henderson, Carina P. Tan, Sargent Bruce J, Xiao-Ming Guan, Scott D. Feighner, Iyassu K. Sebhat, Jie Pan, Jian Liu, Donald J. Marsh, Matthew J. Wyvratt, Andrew D. Howard, Megan Ruenz
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1913-1917
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Structure–activity relationship, Molecular Biology, Biphenyl, Chemistry, Drug discovery, fungi, Organic Chemistry, Imidazoles, Rats, Bombesin receptor, Bioavailability, Receptors, Bombesin, Molecular Medicine, Bombesin Receptor Subtype-3
-
2
المؤلفون: Doreen E. Cashen, Constantin Tamvakopoulos, Qianping Peng, William J. Martin, David H. Weinberg, Charles Rosenblum, Arthur A. Patchett, Tanya MacNeil, Patrick G. Pollard, Zhixiong Ye, Raman K. Bakshi, Ralph A. Stearns, Rubana N. Kalyani, Palucki Brenda, Joseph M. Metzger, Alison M. Strack, Lex H.T. Van der Ploeg, D. Euan MacIntyre, Iyassu K. Sebhat, Aurawan Vongs, Airu S. Chen, Ravi P. Nargund, Liangqin Guo, Matthew J. Wyvratt, Randy R. Miller, Rui Tang, Howard Y. Chen, Khaled J. Barakat
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:3501-3505
مصطلحات موضوعية: Male, Agonist, Quinuclidines, Time Factors, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Rodentia, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Rats, Sprague-Dawley, Eating, Structure-Activity Relationship, Piperidines, In vivo, Drug Discovery, medicine, Animals, Humans, Receptor, Molecular Biology, Aza Compounds, Bicyclic molecule, Chemistry, Penile Erection, digestive, oral, and skin physiology, Organic Chemistry, Small molecule, Rats, Microsomes, Liver, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin, Protein Binding
-
3
المؤلفون: George A. Doss, Lex H.T. Van der Ploeg, Qianping Peng, Ravi P. Nargund, Charles Rosenblum, Randall R. Miller, Aurawan Vongs, Palucki Brenda, Tanya MacNeil, Ralph A. Stearns, Min K. Park, David H. Weinberg, Rui Tang, Arthur A. Patchett, Constantin Tamvakopoulos
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:1993-1996
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Receptor, Molecular Biology, biology, Chemistry, Organic Chemistry, biology.organism_classification, In vitro, Piperazine, Microsoma, Microsome, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
-
4
المؤلفون: William J. Martin, D. Euan MacIntyre, Ravi P. Nargund, Rubana N. Kalyani, Rui Tang, George A. Doss, Min K. Park, Alison M. Strack, Erin McGowan, Joseph M. Metzger, Charles Rosenblum, Randall R. Miller, Palucki Brenda, Qianping Peng, Arthur A. Patchett, Ralph A. Stearns, Patrick G. Pollard, Lex H.T. Van der Ploeg, Iyassu K. Sebhat, Constantin Tamvakopoulos, Cherrie Shepherd, Aurawan Vongs, Tanya MacNeil, David H. Weinberg, Zhixiong Ye
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:171-175
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Piperazines, Mice, Dogs, Erectile Dysfunction, Piperidines, In vivo, Drug Discovery, medicine, Animals, Obesity, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Haplorhini, In vitro, Rats, Receptor, Melanocortin, Type 4, Molecular Medicine, Melanocortin
-
5
المؤلفون: James M. Schaeffer, Lihu Yang, Ralph T. Mosley, Elizabeth T. Birzin, Alexander Pasternak, Susan P. Rohrer, Yanping Pan, Arthur A. Patchett
المصدر: Letters in Drug Design & Discovery. 1:121-125
مصطلحات موضوعية: Biochemistry, Chemistry, Somatostatin receptor, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Somatostatin receptor 2, Somatostatin receptor 1
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::90a812c1b95fe12969db74b56255181b
https://doi.org/10.2174/1570180043485563 -
6
المؤلفون: Arthur A. Patchett
المصدر: Journal of Medicinal Chemistry. 45:5609-5616
مصطلحات موضوعية: Chemistry, Management science, Drug discovery, Peptidyl-Dipeptidase A, Drug Discovery, Molecular Medicine, Natural (music), General Medicine, Medicinal chemistry, Somatotropin-releasing factor, Natural (archaeology), Lovastatine
-
7
المؤلفون: Ralph A. Stearns, Randy R. Miller, William J. Martin, Ravi P. Nargund, Erin McGowan, Lex H.T. Van der Ploeg, and Arthur A. Patchett, Andrew D. Howard, David B. R. Johnston, D. Euan MacIntyre, Rubana N. Kalyani, Khaled Barakat, Raman K. Bakshi, Ralph T. Mosley, Jennifer E. Drisko, Constantin Tamvakopoulos, Rui Tang, Alison M. Strack, Zhixiong Ye, Doreen E. Cashen, Tanya MacNeil, David H. Weinberg, Palucki Brenda, Gary J Hom, Iyassu K. Sebhat
المصدر: Journal of Medicinal Chemistry. 45:4589-4593
مصطلحات موضوعية: Agonist, Chemistry, medicine.drug_class, Biological activity, Pharmacology, Melanocortin receptor, THIQ, Drug Discovery, medicine, Anorectic, Molecular Medicine, Structure–activity relationship, Melanocortin, Receptor, medicine.drug
-
8
المؤلفون: Christopher P. Austin, Doreen E. Cashen, Sheng-Shung Pong, Brian D. Spar, Brett Connolly, Tung Ming Fong, D. Euan MacIntyre, Carina P. Tan, Michael R. Tota, Ravi P. Nargund, R. S. L. Chang, Oksana C. Palyha, Constantin Tamvakopoulos, Deborah L. Drazen, Anthony G. DiLella, Jennifer E. Drisko, David J. Figueroa, Tanya MacNeil, Andreas W. Sailer, David H. Weinberg, Randy J. Nelson, Charles Rosenblum, Cathy R.-R.C. Huang, Rui Tang, Arthur A. Patchett, Xiao-Ming Guan, Hong Yu, George J. Christ, Andrew D. Howard, Lex H.T. Van der Ploeg, William J. Martin, Aurawan Vongs, Iyassu K. Sebhat, Ralph A. Stearns
المصدر: Proceedings of the National Academy of Sciences. 99:11381-11386
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, DNA, Complementary, Intracranial Pressure, medicine.drug_class, Blood Pressure, In Vitro Techniques, Biology, Somatosensory system, Mice, Sexual Behavior, Animal, Nerve Fibers, Internal medicine, Copulation, medicine, Animals, Glans, In Situ Hybridization, DNA Primers, Multidisciplinary, Reverse Transcriptase Polymerase Chain Reaction, Human penis, Feeding Behavior, Ribonuclease, Pancreatic, Biological Sciences, Spinal cord, Electric Stimulation, Mice, Inbred C57BL, Melanocortin 4 receptor, medicine.anatomical_structure, Endocrinology, Receptors, Corticotropin, Models, Animal, Receptor, Melanocortin, Type 4, Brainstem, Energy Metabolism, Penis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::341db11f0e12a0307d07e04176cd4aad
https://doi.org/10.1073/pnas.172378699 -
9
المؤلفون: Zhixiong Ye, Elizabeth T. Birzin, Meng-Hsin Chen, Louis Locco, Sheng-Shung Pong, Ravi P. Nargund, Rupa M. Parmar, Roy G. Smith, Ying-Duo Gao, Scott D. Feighner, Wanda W.-S. Chan, James M. Schaeffer, Arthur A. Patchett, Raman K. Bakshi, Allan D. Blake, Andrew D. Howard, Susan P. Rohrer
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:5-8
مصطلحات موضوعية: Models, Molecular, Agonist, Molecular model, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Receptors, Cell Surface, Carboxamide, Pharmacology, Biochemistry, Chemical synthesis, Receptors, G-Protein-Coupled, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Receptors, Ghrelin, Molecular Biology, Quinazolinone, Binding Sites, Human Growth Hormone, Chemistry, Organic Chemistry, In vitro, Rats, Kinetics, Drug Design, Quinazolines, Molecular Medicine, Secretagogue, Secretory Rate
-
10
المؤلفون: Sheng-Shung Pong, Mark Abramovitz, Andrew D. Howard, Rino Stocco, Ploeg, Raman K. Bakshi, Stacia Kargman, Carina P. Tan, Donna L. Hreniuk, Margaret A. Cascieri, David J. Figueroa, Ravi P. Nargund, Karen K. McKee, Jilly F. Evans, Scott D. Feighner, Lex H. T. Van Der, Christopher P. Austin, Oksana C. Palyha, Roy G. Smith, Douglas J. MacNeil, Arthur A. Patchett, Gary P. O'Neill
المصدر: Science. 284:2184-2188
مصطلحات موضوعية: Receptors, Neuropeptide, medicine.medical_specialty, Colon, G protein, Motilin receptor, Molecular Sequence Data, Thyroid Gland, Gastric motility, Peptide hormone, Biology, Ligands, Transfection, Cell Line, Receptors, Gastrointestinal Hormone, Motilin, GTP-Binding Proteins, Internal medicine, Heterotrimeric G protein, Intestine, Small, medicine, Humans, Amino Acid Sequence, Cloning, Molecular, Receptor, Antrum, In Situ Hybridization, Binding Sites, Multidisciplinary, Base Sequence, Chromosomes, Human, Pair 13, digestive, oral, and skin physiology, Chromosome Mapping, Erythromycin, Alternative Splicing, Endocrinology, Gastric Mucosa, Calcium, hormones, hormone substitutes, and hormone antagonists