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1دورية أكاديمية
المؤلفون: Frank M Szaba, Michael Tighe, Lawrence W Kummer, Kathleen G Lanzer, Jerrold M Ward, Paula Lanthier, In-Jeong Kim, Atsuo Kuki, Marcia A Blackman, Stephen J Thomas, Jr-Shiuan Lin
المصدر: PLoS Pathogens, Vol 14, Iss 4, p e1006994 (2018)
مصطلحات موضوعية: Immunologic diseases. Allergy, RC581-607, Biology (General), QH301-705.5
وصف الملف: electronic resource
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2
المؤلفون: Tran Khanh Tuan, Qiyue Hu, Zhang Junhu, Scott L. Butler, Atsuo Kuki, Qinghai Peng, Erik Jon Flahive, Graham L. Smith, Huichun Zhu, Deepak Dalvie, Plewe Michael Bruno, Jim Solowiej, Dorothy Delisle, Ted William Johnson, Wen Liu, Steven P. Tanis, Klaus Ruprecht Dress, Jon E. Kuehler, Guy A. McClellan, Xiaoming Yu, Hai Wang, Paul F. Richardson
المصدر: Journal of Medicinal Chemistry. 54:3393-3417
مصطلحات موضوعية: Cell Membrane Permeability, Molecular Conformation, Administration, Oral, Biological Availability, Integrase inhibitor, Pharmacology, Structure-Activity Relationship, Dogs, Drug Discovery, Animals, Humans, HIV Integrase Inhibitors, Naphthyridines, Cells, Cultured, chemistry.chemical_classification, biology, Chemistry, virus diseases, Ligand (biochemistry), Integrase, Bioavailability, Enzyme, Liver, Viral replication, Drug Design, HIV-1, Hepatocytes, biology.protein, Hiv 1 integrase, Molecular Medicine, Heterocyclic Compounds, 3-Ring, Tricyclic
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3
المؤلفون: Qinghai Peng, Tran Khanh Tuan, Atsuo Kuki, Steven P. Tanis, Zhang Junhu, Deepak Dalvie, Yang Anle, Xiaoming Yu, Jim Solowiej, Ted William Johnson, Hai Wang, Wen Liu, Plewe Michael Bruno, Buwen Huang, Graham L. Smith, Jon E. Kuehler, Klaus Ruprecht Dress, Chunfeng Yin, Qiyue Hu, Dorothy Delisle, Huichun Zhu, Scott L. Butler
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:7429-7434
مصطلحات موضوعية: Indoles, Stereochemistry, Clinical Biochemistry, Glucuronidation, Administration, Oral, Pharmaceutical Science, Integrase inhibitor, HIV Integrase, Hydroxamic Acids, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Drug Discovery, Animals, Humans, Structure–activity relationship, HIV Integrase Inhibitors, Molecular Biology, ADME, chemistry.chemical_classification, Hydroxamic acid, biology, Organic Chemistry, Integrase, Enzyme, chemistry, Enzyme inhibitor, HIV-1, Hepatocytes, biology.protein, Molecular Medicine, Half-Life
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4
المؤلفون: Qinghai Peng, Nowlin Dawn Marie, Hieu Lam, Ted William Johnson, Yang Anle, Wen Liu, Atsuo Kuki, Steven P. Tanis, Jon E. Kuehler, Zhang Junhu, Hai Wang, Plewe Michael Bruno, Scott L. Butler, Tran Khanh Tuan, Qiyue Hu, Sadayappan V. Rahavendran, Klaus Ruprecht Dress
المصدر: Journal of Medicinal Chemistry. 52:7211-7219
مصطلحات موضوعية: Stereochemistry, Drug Evaluation, Preclinical, Integrase inhibitor, HIV Integrase, Hydroxamic Acids, Ligands, Chemical synthesis, Inhibitory Concentration 50, chemistry.chemical_compound, Drug Discovery, Magnesium, HIV Integrase Inhibitors, chemistry.chemical_classification, Hydroxamic acid, biology, Chemistry, virus diseases, Nucleotidyltransferase, Integrase, Enzyme, Biochemistry, Viral replication, Enzyme inhibitor, Picolines, HIV-1, biology.protein, Molecular Medicine
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5
المؤلفون: Jesper Lau, James Lakis, Shenghua Shi, Javier Gonzalez, Teston Kimberly Ann, Lotte Bjerre Knudsen, Yufeng Hong, John M. May, Douglas E. Murphy, Atsuo Kuki, Dan Kiel, Anthony Lai Ling, Kenna Anderes, Alex Polinsky, Vlad E. Gregor, John B. Porter
المصدر: Journal of Medicinal Chemistry. 44:3141-3149
مصطلحات موضوعية: Blood Glucose, Male, High-throughput screening, In Vitro Techniques, Binding, Competitive, Glucagon, Chemical synthesis, Cell Line, Rats, Sprague-Dawley, Radioligand Assay, Structure-Activity Relationship, In vivo, Drug Discovery, Cyclic AMP, Receptors, Glucagon, Animals, Combinatorial Chemistry Techniques, Humans, Rats, Wistar, Chemistry, Hydrazones, Antagonist, Small molecule, In vitro, Rats, Liver, Biochemistry, Benzamides, Molecular Medicine, Glucagon receptor
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6
المؤلفون: Shenghua Shi, Jaroslaw Kostrowicki, Zhengwei Peng, Atsuo Kuki, Genevieve Paderes
المصدر: Journal of Molecular Graphics and Modelling. 18:478-496
مصطلحات موضوعية: Basis (linear algebra), Chemistry, Component (thermodynamics), Filter (signal processing), Interference (wave propagation), Computer Graphics and Computer-Aided Design, Accessible surface area, symbols.namesake, Models, Chemical, Computational chemistry, Drug Design, Product (mathematics), Materials Chemistry, symbols, Combinatorial Chemistry Techniques, Physical and Theoretical Chemistry, van der Waals force, Representation (mathematics), Biological system, Algorithms, Spectroscopy
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7
المؤلفون: and James M. Gruschus, Atsuo Kuki
المصدر: The Journal of Physical Chemistry B. 103:11407-11414
مصطلحات موضوعية: Physics::Biological Physics, Chemistry, Cytochrome c peroxidase, Electron, Acceptor, Surfaces, Coatings and Films, Coupling (electronics), Delocalized electron, Electron transfer, Atomic orbital, Materials Chemistry, Physical and Theoretical Chemistry, Atomic physics, Wave function
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8
المؤلفون: and Atsuo Kuki, Gautam Basu, Nobuhiro Go, Akio Kitao
المصدر: The Journal of Physical Chemistry B. 102:2076-2084
مصطلحات موضوعية: Coupling, Quantitative Biology::Biomolecules, Chemistry, Solvation, Potential energy, Surfaces, Coatings and Films, Electron transfer, Hyperplane, Normal mode, Energy spectrum, Materials Chemistry, Physical and Theoretical Chemistry, Atomic physics, Vector space
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9
المؤلفون: Gautam Basu, Akio Kitao, and Atsuo Kuki, Nobuhiro Go
المصدر: The Journal of Physical Chemistry B. 102:2085-2094
مصطلحات موضوعية: Coupling (electronics), Electron transfer, Materials science, biology, Normal mode, Cytochrome c, Energy spectrum, Materials Chemistry, biology.protein, Physical and Theoretical Chemistry, Atomic physics, Surfaces, Coatings and Films
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10
المؤلفون: Atsuo Kuki, Kamil Lang, William Chrisman, Enugurthi Brahmachary, Demetrios Anglos, Sambasivarao Kotha, Bakthan Singaram
المصدر: Scopus-Elsevier
مصطلحات موضوعية: chemistry.chemical_classification, Acid derivative, Design, Aminoisobutyric-Acid, Stereochemistry, Carboxylic acid, Metalated Isocyanides, Organic Chemistry, Biochemistry, Amino acid, chemistry.chemical_compound, Quinoxaline, chemistry, Drug Discovery, Side chain, Peptides, Rich