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المؤلفون: Jeffrey W. Johannes, Fiona Pachl, Amber Balazs, Tieguang Yao, C. Larner, Lisa McWilliams, Marianne Schimpl, Scott W. Martin, Kevin J. Embrey, Tom D. Heightman, Paul Hemsley, Jonathan P. Orme, Derek Barratt, Giuditta Illuzzi, Andrew Madin, Paolo Di Fruscia, Avipsa Ghosh, Martin J. Packer, Scott D. Edmondson, Elisabetta Leo, Xiaolan Zheng, Matthew D. Chuba, Xiaohui Pei, Mark J. O'Connor, Verity Talbot, Ke Zhang, Stephen Fawell, Elizabeth Underwood, Anna Staniszewska, Lina Liu, Lin Xue, Sonja J. Gill, Anders Gunnarsson, Andrew Pike, Susan E. Critchlow, Jeffrey G. Varnes, Andrew X. Zhang, Sébastien L. Degorce, J. Lane, Sudhir M. Hande, Hongyao She, Sabina Cosulich, Michal Bista
المصدر: Journal of Medicinal Chemistry. 64:14498-14512
مصطلحات موضوعية: chemistry.chemical_compound, PARP1, Chemistry, In vivo, Poly ADP ribose polymerase, Drug Discovery, Mutant, Cancer research, Molecular Medicine, Progenitor cell, Homologous recombination, DNA, In vitro
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المصدر: The Journal of organic chemistry. 87(14)
مصطلحات موضوعية: Nickel, Organic Chemistry, Iodides, Iridium, Catalysis
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المؤلفون: Avipsa Ghosh, Jeffrey W. Johannes, Christopher S. Gravatt
مصطلحات موضوعية: chemistry.chemical_compound, Nickel, Catalytic cycle, Chemistry, Aryl, Functional group, Photocatalysis, Halide, chemistry.chemical_element, Iridium, Combinatorial chemistry, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bc963fffdd89ad0b587684261d00b8e4
https://doi.org/10.26434/chemrxiv-2021-18xd5 -
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المؤلفون: Jeffrey W, Johannes, Amber, Balazs, Derek, Barratt, Michal, Bista, Matthew D, Chuba, Sabina, Cosulich, Susan E, Critchlow, Sébastien L, Degorce, Paolo, Di Fruscia, Scott D, Edmondson, Kevin, Embrey, Stephen, Fawell, Avipsa, Ghosh, Sonja J, Gill, Anders, Gunnarsson, Sudhir M, Hande, Tom D, Heightman, Paul, Hemsley, Giuditta, Illuzzi, Jordan, Lane, Carrie, Larner, Elisabetta, Leo, Lina, Liu, Andrew, Madin, Scott, Martin, Lisa, McWilliams, Mark J, O'Connor, Jonathan P, Orme, Fiona, Pachl, Martin J, Packer, Xiaohui, Pei, Andrew, Pike, Marianne, Schimpl, Hongyao, She, Anna D, Staniszewska, Verity, Talbot, Elizabeth, Underwood, Jeffrey G, Varnes, Lin, Xue, Tieguang, Yao, Ke, Zhang, Andrew X, Zhang, Xiaolan, Zheng
المصدر: Journal of medicinal chemistry. 64(19)
مصطلحات موضوعية: Poly (ADP-Ribose) Polymerase-1, Humans, DNA, Poly(ADP-ribose) Polymerase Inhibitors, Poly(ADP-ribose) Polymerases, Crystallography, X-Ray, Substrate Specificity
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المؤلفون: Shin‐Ho Kim‐Lee, Alexander T. Radosevich, Morgan Lecomte, Avipsa Ghosh
المصدر: Angewandte Chemie International Edition. 58:2864-2869
مصطلحات موضوعية: Phosphine oxide, Sulfonyl, chemistry.chemical_classification, Trifluoromethyl, 010405 organic chemistry, General Chemistry, 010402 general chemistry, 01 natural sciences, Medicinal chemistry, Catalysis, 0104 chemical sciences, chemistry.chemical_compound, chemistry, Organocatalysis, Electrophile, Deoxygenation, Phosphine
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المؤلفون: Avipsa Ghosh, Morgan Lecomte, Shin‐Ho Kim‐Lee, Alexander T. Radosevich
المصدر: Angewandte Chemie. 131:2890-2895
مصطلحات موضوعية: General Medicine
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المؤلفون: Avipsa Ghosh, Sudhir M. Hande, Amber Balazs, Derek Barratt, Sabina Cosulich, Barry Davies, Sébastien Degorce, Kevin Embrey, Sonja Gill, Anders Gunnarsson, Giuditta Illuzzi, Peter Johnström, Jordan Lane, Carrie Larner, Rachel Lawrence, Elisabetta Leo, Andrew Madin, Elizabeth Martin, Lisa McWilliams, Lenka O’Connor, Mark O’Connor, Jonathan Orme, Fiona Pachl, Martin Packer, Andy Pike, Philip Rawlins, Marianne Schimpl, Magnus Schou, Anna Staniszewska, Wenzhan Yang, James Yates, Andrew Zhang, XiaoLa Zheng, Stephen Fawell, Petra Hamerlik, Jeffrey Johannes
المصدر: Cancer Research. 82:6302-6302
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::288251eb61b3a0254c30186cb54c9b42
https://doi.org/10.1158/1538-7445.am2022-6302 -
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المؤلفون: Andy Pike, Amber Balazs, Zsolt Cselényi, Sébastien L. Degorce, Avipsa Ghosh, Sudhir M. Hande, Jeffrey Johannes, Peter Johnström, Martin J. Packer, Magnus Schou, XiaoLan Zheng
المصدر: Cancer Research. 82:5076-5076
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::9257631ac2f0d93eadc9fa8a4fc52c6f
https://doi.org/10.1158/1538-7445.am2022-5076 -
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المؤلفون: Mark J. O'Connor, Philip B. Rawlins, Kevin J. Embrey, Anders Gunnarsson, Sudhir M. Hande, Anna Staniszewska, Fiona Pachl, Andrew X. Zhang, Jonathan P. Orme, Giuditta Illuzzi, Lisa McWilliams, Sonja J. Gill, Jeffrey W. Johannes, J. Lane, Sébastien L. Degorce, Amber Balazs, Martin J. Packer, Andrew Madin, Marianne Schimpl, Andrew Pike, Elisabetta Leo, Xiaolan Zheng, Avipsa Ghosh, C. Larner
المصدر: Cancer Research. 81:296-296
مصطلحات موضوعية: chemistry.chemical_classification, Cancer Research, Nicotinamide, biology, Poly ADP ribose polymerase, hERG, Olaparib, chemistry.chemical_compound, Enzyme, PARP1, Oncology, chemistry, PARP inhibitor, Cancer research, biology.protein, Binding site
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::5541745268ca2c08d1cdc8f164ef2184
https://doi.org/10.1158/1538-7445.am2021-296