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1
المؤلفون: Beverly P. Holskin, Karla Kopec, Joanne R. Mathiasen, Amy DiCamillo, Babu G. Sundar, Thomas J. Connors, Emir Duzic, Edward R. Bacon, Gerard C. Rosse, Chrysanthe Spais, Thomas R. Bailey, Beth Ann McKenna, Rebecca A. Brown, Jie Qian, Derek Dunn, Mark J. Huffman, Joseph M. Salvino, Huang Zeqi, Lisa D. Aimone, Hervé Schaffhauser, Deborah Galinis, Thelma S. Angeles, Lily D. Lu, George C. Morton
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:120-123
مصطلحات موضوعية: biology, Organic Chemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Biochemistry, Social recognition, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, 5-HT6 receptor, Molecular Medicine, Structure–activity relationship, Serotonin Antagonists, Penetrant (biochemical), Receptor, Molecular Biology, 5-HT receptor
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2
المؤلفون: Edward R. Bacon, Jacquelyn A. Lyons, Thomas R. Bailey, Robert L. Hudkins, Rita Raddatz, Zeqi Huang, Lisa D. Aimone, Babu G. Sundar
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5543-5546
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Histamine h, Biochemistry, Pharmacokinetics, In vivo, Drug Discovery, Molecular Medicine, Structure–activity relationship, Amine gas treating, Receptor, Molecular Biology
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3
المؤلفون: Kurt A. Josef, Allison L. Zulli, Lisa D. Aimone, Derek Dunn, Rita Raddatz, Jacquelyn A. Lyons, Ming Tao, Joanne R. Mathiasen, Reddeppa reddy Dandu, Thomas R. Bailey, Val R. Marcy, Babu G. Sundar, John A. Gruner, Edward R. Bacon, Robert L. Hudkins, Robert J. Bendesky, Yin-Guo Lin
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5493-5497
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Histamine h, Biochemistry, In vivo, Drug Discovery, Molecular Medicine, Inverse agonist, Potency, Selectivity, Antagonism, Receptor, Molecular Biology, Linker
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4
المؤلفون: Kurt A. Josef, Curtis R. Haltiwanger, Robert J. McHugh, Babu G. Sundar
المصدر: Synthetic Communications. 41:1481-1485
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Chemistry, Stereochemistry, Hydrogen maleate, Organic Chemistry, Thermal, Salt (chemistry), Amine gas treating, Medicinal chemistry, Derivative (chemistry)
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5
المؤلفون: Babu G, Sundar, Thomas R, Bailey, Derek D, Dunn, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Huang, Zeqi, Joanne R, Mathiasen, Amy, Dicamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Rebecca, Brown, Jie, Qian, Thelma, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Deborah, Galinis, Emir, Duzic, Herve, Schaffhauser, Gerard C, Rosse
المصدر: Bioorganicmedicinal chemistry letters. 22(1)
مصطلحات موضوعية: ERG1 Potassium Channel, Brain, Ether-A-Go-Go Potassium Channels, Rats, Inhibitory Concentration 50, Kinetics, Structure-Activity Relationship, Memory, Short-Term, Models, Chemical, Piperidines, Receptors, Serotonin, Schizophrenia, Animals, Humans, Serotonin Antagonists, Benzofurans
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6
المؤلفون: Robert J. McHugh, Kurt A. Josef, Curtis R. Haltiwanger, Babu G. Sundar
المصدر: ChemInform. 42
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Chemistry, Hydrogen maleate, Salt (chemistry), Amine gas treating, General Medicine, Medicinal chemistry, Derivative (chemistry), Pyrrole derivatives
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7
المؤلفون: Robert L, Hudkins, Lisa D, Aimone, Thomas R, Bailey, Robert J, Bendesky, Reddeppa Reddy, Dandu, Derek, Dunn, John A, Gruner, Kurt A, Josef, Yin-Guo, Lin, Jacquelyn, Lyons, Val R, Marcy, Joanne R, Mathiasen, Babu G, Sundar, Ming, Tao, Allison L, Zulli, Rita, Raddatz, Edward R, Bacon
المصدر: Bioorganicmedicinal chemistry letters. 21(18)
مصطلحات موضوعية: Male, Dose-Response Relationship, Drug, Molecular Structure, Drinking, Stereoisomerism, Rats, Histamine Agonists, Pyridazines, Disease Models, Animal, Structure-Activity Relationship, Animals, Humans, Receptors, Histamine H3, Wakefulness
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8
المؤلفون: Babu G, Sundar, Thomas, Bailey, Edward, Bacon, Lisa, Aimone, Zeqi, Huang, Jacquelyn, Lyons, Rita, Raddatz, Robert, Hudkins
المصدر: Bioorganicmedicinal chemistry letters. 21(18)
مصطلحات موضوعية: Pyridazines, Structure-Activity Relationship, Dose-Response Relationship, Drug, Molecular Structure, Animals, Humans, Receptors, Histamine H3, Stereoisomerism, Amines, Histamine H3 Antagonists, Rats