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المؤلفون: Satenig Guler, Maria C. DiPoto, Alejandro Crespo, Richard Caldwell, Benjamin Doerfel, Nina Grossmann, Kevin Ho, Bayard Huck, Christopher CV Jones, Ruoxi Lan, Djordje Musil, Justin Potnick, Heike Schilke, Brian Sherer, Stephanie Simon, Christian Sirrenberg, Zhuo Zhang, Lesley Liu-Bujalski
المصدر: ACS Medicinal Chemistry Letters. 14:566-576
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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2
المؤلفون: Momar Toure, Constantin Neagu, Kevin Ho, Susan Zhang, Filippos Porichis, Zhizhou Fang, Maria DiPoto, Reinaldo Jones, Eugene Chekler, Eva Maria Tanzer, Brian Sherer, Theresa Johnson, Djordje Musil, Bin Li, Ralf Schmidt, Hong Ma, Andrea Unzue Lopez, Yanping Wang, Satenig Guler, YuFang Xiao, Renate Henkes, Chia Lin Chu, Uma Mahesh Gundra, Long Li, Christine Katharina Maurer, Emily Friis, Christopher Jones, James Cummings, Bayard Huck
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::60c4b42c55d861e189da387afa4d82a1
https://doi.org/10.2139/ssrn.4382746 -
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المؤلفون: Rienk Offringa, Lisa Kötzner, Bayard Huck, Klaus Urbahns
المصدر: Nature reviews. Drug discovery. 21(11)
مصطلحات موضوعية: Pharmacology, Neoplasms, T-Lymphocytes, Drug Discovery, Tumor Microenvironment, Humans, Cytokines, General Medicine, Immunotherapy
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المؤلفون: Rinat Zaynagetdinov, Kai Schiemann, Kalyan Nallaparaju, Natalya Belousova, Armine Matevossian, Zhouxiang Chen, Giorgio Kradjian, Meghana Pandya, Nemisha Dawra, Eva-Maria Krauel, Elissaveta Petrova, Oliver Poeschke, David Fischer, Marc Lecomte, Andree Blaukat, Bayard Huck, Jacques Moisan
المصدر: Cancer Research. 82:3499-3499
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4d0f249470dc089a58550abfb940baab
https://doi.org/10.1158/1538-7445.am2022-3499 -
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المؤلفون: Lisa, Kötzner, Bayard, Huck, Sakshi, Garg, Klaus, Urbahns
المصدر: Progress in medicinal chemistry. 59
مصطلحات موضوعية: Small Molecule Libraries, Neoplasms, Humans, Antineoplastic Agents, Amino Acids, Protein Kinase Inhibitors, Protein Kinases
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::837fac698ac6e4ffec531726af3349a8
https://pubmed.ncbi.nlm.nih.gov/32362326 -
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المؤلفون: William F. Hodnick, Luis Llamas, Thomas C. Dent, Jianping Song, Youssef L. Bennani, Michael J. Robarge, John J. Harrington, Alain Stricker-Krongrad, Kurt R. Brunden, Bayard Huck, Chris Crumrine
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:4130-4134
مصطلحات موضوعية: Agonist, Nitrogen, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Dogs, Drug Discovery, medicine, Animals, Structure–activity relationship, Receptor, Molecular Biology, G protein-coupled receptor, chemistry.chemical_classification, Organic Chemistry, Biological activity, Feeding Behavior, Rats, Serotonin Receptor Agonists, chemistry, Drug Design, Molecular Medicine, 5-HT2C receptor agonist, Serotonin 5-HT2 Receptor Agonists, Half-Life, Tricyclic
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المؤلفون: Luis Llamas, William F. Hodnick, Michael J. Robarge, Bayard Huck, Chris Crumrine, Youssef L. Bennani, John J. Harrington, Thomas C. Dent, Alain Stricker-Krongrad, Kurt R. Brunden, Jianping Song
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:2891-2894
مصطلحات موضوعية: Agonist, Pyrimidine, medicine.drug_class, media_common.quotation_subject, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Bridged Bicyclo Compounds, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Receptor, Serotonin, 5-HT2C, medicine, Animals, Amines, Receptor, Molecular Biology, media_common, Octane, Aza Compounds, Molecular Structure, Organic Chemistry, Stereoisomerism, Appetite, Small molecule, Rats, 5-HT2C receptor, Pyrimidines, chemistry, Molecular Medicine, Serotonin 5-HT2 Receptor Agonists
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المؤلفون: Steven M. Murphy, Bruce Sherf, Tom Dent, Daniel P. Silver, Andrew Bailey, L. Nathan Tumey, Jianmin Wang, Youssef L. Bennani, Elizabeth Ann Gleason, David C. Bom, Bayard Huck, Christina Leventhal, Sherry Boozer, John J. Harrington, Stephen Rundlett, Kurt R. Brunden
المصدر: Bioorganicmedicinal chemistry letters. 15(2)
مصطلحات موضوعية: Xeroderma pigmentosum, DNA repair, DNA damage, Flap Endonucleases, Clinical Biochemistry, Flap structure-specific endonuclease 1, Pharmaceutical Science, Biochemistry, Endonuclease, chemistry.chemical_compound, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, medicine, Temozolomide, Humans, Urea, Enzyme Inhibitors, Molecular Biology, Xeroderma Pigmentosum, biology, Organic Chemistry, Base excision repair, medicine.disease, Methyl Methanesulfonate, Methyl methanesulfonate, Dacarbazine, chemistry, Urinary Bladder Neoplasms, biology.protein, Molecular Medicine, Nucleotide excision repair, DNA Damage
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المؤلفون: Jianmin Wang, John J. Harrington, Daniel P. Silver, Bayard Huck, Kurt R. Brunden, Christina Leventhal, Bruce Sherf, L. Nathan Tumey, Tom Dent, Steven M. Murphy, Elizabeth Ann Gleason, Andrew Bailey, Sherry Boozer, Stephen Rundlett, Youssef L. Bennani
المصدر: Bioorganicmedicinal chemistry letters. 14(19)
مصطلحات موضوعية: chemistry.chemical_classification, biology, DNA damage, DNA repair, Flap Endonucleases, Organic Chemistry, Clinical Biochemistry, Flap structure-specific endonuclease 1, Pharmaceutical Science, Base excision repair, Biochemistry, Endonuclease, chemistry.chemical_compound, Butyrates, Structure-Activity Relationship, Enzyme, chemistry, Drug Discovery, biology.protein, Molecular Medicine, Flap endonuclease, Enzyme Inhibitors, Molecular Biology, DNA