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1MWC allosteric model explains unusual hemoglobin-oxygen binding curves from sickle cell drug binding
المؤلفون: Belhu B. Metaferia, Julia Harper, John M. Louis, William A. Eaton, Kristen E. Glass, Eric R. Henry
المصدر: Biophysical Journal. 120:2543-2551
مصطلحات موضوعية: Allosteric regulation, Biophysics, chemistry.chemical_element, Anemia, Sickle Cell, Plasma protein binding, Oxygen, Dissociation (chemistry), Hemoglobins, 03 medical and health sciences, 0302 clinical medicine, Allosteric Regulation, medicine, Humans, 030304 developmental biology, 0303 health sciences, Chemistry, Oxygen–haemoglobin dissociation curve, Kinetics, Pharmaceutical Preparations, Mechanism of action, Hemoglobin, medicine.symptom, 030217 neurology & neurosurgery, Oxygen binding, Protein Binding
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2
المؤلفون: Julia Harper, Eric R. Henry, Swee Lay Thein, Quan Li, William A. Eaton, Emily B. Dunkelberger, Troy Cellmer, H. Franklin Bunn, Kristen E. Glass, Robert B. Best, Belhu B. Metaferia, Anna Conrey
المصدر: Blood. 138(13)
مصطلحات موضوعية: Drug, Models, Molecular, Erythrocytes, media_common.quotation_subject, Immunology, Hemoglobin, Sickle, chemistry.chemical_element, Anemia, Sickle Cell, Pharmacology, Biochemistry, Oxygen, In vivo, Antisickling Agents, medicine, Humans, media_common, Red Cell, Mean corpuscular hemoglobin concentration, medicine.diagnostic_test, Chemistry, Cell Biology, Hematology, medicine.disease, Sickle cell anemia, Hemolysis, Benzaldehydes, Pyrazines, Pyrazoles, Hemoglobin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4643242567d327f4e2c46909f5468d1c
https://pubmed.ncbi.nlm.nih.gov/35815728 -
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المؤلفون: Pablo Bartolucci, William A. Eaton, Quan Li, Emily B. Dunkelberger, David Ostrowski, Swee Lay Thein, Troy Cellmer, Belhu B. Metaferia, James Hofrichter, John M. Louis, Eric R. Henry, Rodolfo Ghirlando, Frédéric Galactéros, Stéphane Moutereau
المصدر: Proceedings of the National Academy of Sciences of the United States of America
مصطلحات موضوعية: Erythrocytes, Hereditary persistence of fetal hemoglobin, Allosteric regulation, Hemoglobin, Sickle, Anemia, Sickle Cell, Compound heterozygosity, sickle cell, Allosteric Regulation, Fetal hemoglobin, medicine, Humans, Fetal Hemoglobin, Multidisciplinary, Chemistry, Biological Sciences, medicine.disease, Abnormal hemoglobin, Oxygen, Kinetics, Biophysics and Computational Biology, polymerization, Biophysics, Protein quaternary structure, Hemoglobin, Intracellular, protein fibers
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b5f8de3a122dfcb1a10edbfaa026a7cc
https://pubmed.ncbi.nlm.nih.gov/32527859 -
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المؤلفون: Emily B. Dunkelberger, Troy Cellmer, Belhu B. Metaferia, Eric R. Henry
المصدر: The Journal of Physical Chemistry B. 122:11579-11590
مصطلحات موضوعية: 0301 basic medicine, Erythrocytes, Hemoglobin, Sickle, Anemia, Sickle Cell, Molecular Dynamics Simulation, Cell morphology, Article, Polymerization, Diffusion, 03 medical and health sciences, 0302 clinical medicine, Materials Chemistry, Humans, Particle Size, Physical and Theoretical Chemistry, Deoxygenation, Sickle Hemoglobin, Hemoglobin s, Red Cell, Chemistry, Surfaces, Coatings and Films, Oxygen, 030104 developmental biology, Time course, Physical chemistry, 030217 neurology & neurosurgery
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5
المؤلفون: Terri H. Wakefield, Eric R. Henry, William A. Eaton, Jeffrey F. Smith, Matthew M. Hsieh, Mary E. Link, Emily B. Dunkelberger, Jeffery L. Miller, James Hofrichter, Troy Cellmer, John F. Tisdale, Dwayne Staton, Belhu B. Metaferia, Garrott W. Christoph, Stacy Jones-Straehle, Quan Li, Sarah Boutom, Erica R. Vass
المصدر: Proceedings of the National Academy of Sciences. 114
مصطلحات موضوعية: 0301 basic medicine, Drug, Erythrocytes, media_common.quotation_subject, Hemoglobin, Sickle, Cell, Mutant, Anemia, Sickle Cell, Disease, Pharmacology, Red cell volume, 03 medical and health sciences, Antisickling Agents, medicine, Humans, Furaldehyde, Cell Size, media_common, Multidisciplinary, Chemistry, Cellular Assay, Oxygen, Kinetics, 030104 developmental biology, medicine.anatomical_structure, PNAS Plus, Biochemistry, Polymerization, Hemoglobin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5594850c3d4be6142aecdb666e07fc70
https://doi.org/10.1073/pnas.1619054114 -
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المؤلفون: Brandon J. Fetterolf, Maria-Teresa Gutierrez-Lugo, Syed Shazad-ul-Hussan, Jeremy A. Smith, Matthew Moravec, Carole A. Bewley, Belhu B. Metaferia, Satyajit Ray
المصدر: Journal of Medicinal Chemistry. 50:6326-6336
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Amidohydrolases, Chemical library, Amidase, chemistry.chemical_compound, Bacterial Proteins, Oxazines, Drug Discovery, Cysteine, Furans, Oxazoles, Pyrans, Antibacterial agent, chemistry.chemical_classification, Sulfonamides, Binding Sites, Natural product, biology, Glycopeptides, Active site, Stereoisomerism, Isoxazoles, Mycobacterium tuberculosis, Mycothiol, Enzyme, chemistry, Biochemistry, Thioglycosides, Enzyme inhibitor, biology.protein, Molecular Medicine, Inositol, Protein Binding
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المؤلفون: David G. I. Kingston, Ami Lakdawala, Jeannine Hoch, James P. Snyder, Susan Bane, Sabarni K. Chatterjee, Thomas E. Glass, Ben Cornett, Belhu B. Metaferia
المصدر: Organic Letters. 3:2461-2464
مصطلحات موضوعية: Models, Molecular, Binding Sites, Paclitaxel, Olefin metathesis, Chemistry, Stereochemistry, Electron crystallography, Organic Chemistry, Molecular Conformation, Crystallography, X-Ray, Antineoplastic Agents, Phytogenic, Biochemistry, Combinatorial chemistry, Taxoid, chemistry.chemical_compound, Cyclization, Tubulin, Tumor Cells, Cultured, Humans, Indicators and Reagents, Physical and Theoretical Chemistry, Binding site, Biological evaluation
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8
المؤلفون: Heidi Hempel, Matthew Rittler, William G. Stetler-Stevenson, Javed Khan, Jinesh S. Gheeya, Alberto Plaza, Carole A. Bewley, Albert Lee, Belhu B. Metaferia
المصدر: Bioorganicmedicinal chemistry letters. 20(24)
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Fluorescence Polarization, Plasma protein binding, CD13 Antigens, Biochemistry, Peptides, Cyclic, Article, Cell Line, Tumor, Drug Discovery, Humans, Molecular Biology, chemistry.chemical_classification, Drug Carriers, Chemistry, Organic Chemistry, Biological activity, Cyclic peptide, Resins, Synthetic, Targeted drug delivery, Cyclization, Cancer cell, Click chemistry, Molecular Medicine, Click Chemistry, Drug carrier, Preclinical imaging, Protein Binding
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9
المؤلفون: James P. Snyder, David G. I. Kingston, Ami Lakdawala, Belhu B. Metaferia, Susan Bane, Sabarni K. Chatterjee, Jeannine Hoch, Thomas E. Glass, Ben Cornett
المصدر: ChemInform. 32
مصطلحات موضوعية: Taxoid, chemistry.chemical_compound, Olefin metathesis, Paclitaxel, Electron crystallography, Stereochemistry, Chemistry, Salt metathesis reaction, General Medicine, Binding site, Biological evaluation
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المؤلفون: Xin-Yun Huang, Lin Chen, Heather L. Baker, Belhu B. Metaferia, Carole A. Bewley
المصدر: Journal of the American Chemical Society. 129(9)
مصطلحات موضوعية: Scaffold, Chemistry, Quinic Acid, Antineoplastic Agents, Breast Neoplasms, General Chemistry, Biochemistry, Combinatorial chemistry, Catalysis, In vitro, Lactones, Colloid and Surface Chemistry, Cell Migration Assay, Models, Chemical, Cell Movement, Ic50 values, Cancer research, Tumor Cells, Cultured, Humans, Female, Breast cancer cells, Wound healing assay, Macrolides, Piperidones