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1
المؤلفون: Beth Ann McKenna, Karla Kopec, Greg A. Hostetler, Sankar Chatterjee, Derek Dunn
المصدر: Chemical Biology & Drug Design. 83:666-669
مصطلحات موضوعية: Drug Inverse Agonism, Stereochemistry, Pharmacology, Biochemistry, Benzazepine, chemistry.chemical_compound, Drug Discovery, Humans, Inverse agonist, Potency, Sulfones, Receptor, Sulfonamides, Molecular Structure, Organic Chemistry, Benzazepines, chemistry, Receptors, Serotonin, 5-HT6 receptor, Molecular Medicine, Biological Assay, Enantiomer, Chirality (chemistry), Protein Binding
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2
المؤلفون: Sankar Chatterjee, Karla Kopec, Beth Ann McKenna, Greg A. Hostetler, Derek Dunn
المصدر: Chemical Biology & Drug Design. 83:149-153
مصطلحات موضوعية: Stereochemistry, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Potency, Spiro Compounds, Structural motif, Receptor, Pharmacology, Sulfonamides, Chemistry, Organic Chemistry, Stereoisomerism, Benzazepines, Recombinant Proteins, Receptors, Serotonin, 5-HT6 receptor, Thiazolidines, Molecular Medicine, Serotonin Antagonists, Nonane, Enantiomer, Antagonism, Selectivity, Protein Binding
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3
المؤلفون: Thomas J. Connors, Jie Qian, Zeck Huang, Joanne R. Mathiasen, Edward R. Bacon, Thelma S. Angeles, Mark J. Huffman, Emir Duzic, Joseph M. Salvino, Beth Ann McKenna, Hervé Schaffhauser, Robert J. McHugh, Lily D. Lu, George C. Morton, Beverly P. Holskin, Karla Kopec, Amy DiCamillo, Gerard C. Rosse, Chrysanthe Spais, Rabindranath Tripathy, Lisa D. Aimone
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1421-1426
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Biochemistry, Sulfone, chemistry.chemical_compound, In vivo, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Pharmacophore, Receptor, Molecular Biology, 5-HT receptor
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4
المؤلفون: Beverly P. Holskin, Karla Kopec, Joanne R. Mathiasen, Amy DiCamillo, Babu G. Sundar, Thomas J. Connors, Emir Duzic, Edward R. Bacon, Gerard C. Rosse, Chrysanthe Spais, Thomas R. Bailey, Beth Ann McKenna, Rebecca A. Brown, Jie Qian, Derek Dunn, Mark J. Huffman, Joseph M. Salvino, Huang Zeqi, Lisa D. Aimone, Hervé Schaffhauser, Deborah Galinis, Thelma S. Angeles, Lily D. Lu, George C. Morton
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:120-123
مصطلحات موضوعية: biology, Organic Chemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Biochemistry, Social recognition, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, 5-HT6 receptor, Molecular Medicine, Structure–activity relationship, Serotonin Antagonists, Penetrant (biochemical), Receptor, Molecular Biology, 5-HT receptor
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5
المؤلفون: Donna Bozyczko-Coyne, Beth Ann Thomas, Michael S. Saporito, Zhi-Liang Wu, Ghanashyam D. Ghadge, Stephen P. Trusko, Maroney Anna, Joanne R. Mathiasen, Beth Ann McKenna, Beverly P. Holskin, Raymond P. Roos, Jeffrey C. Thomas, Thomas C. Connors
المصدر: Brain Research. 1003:86-97
مصطلحات موضوعية: 1-Methyl-4-phenylpyridinium, medicine.medical_specialty, Programmed cell death, Indoles, SH-SY5Y, MAP Kinase Signaling System, Carbazoles, CHO Cells, chemistry.chemical_compound, Cell Line, Tumor, Cricetinae, Internal medicine, medicine, Animals, Humans, Molecular Biology, Cell Death, Dose-Response Relationship, Drug, biology, Kinase, General Neuroscience, MPTP, Neurotoxicity, MAP Kinase Kinase Kinases, medicine.disease, Cell biology, Enzyme Activation, Endocrinology, chemistry, Apoptosis, Cell culture, Mitogen-activated protein kinase, biology.protein, Neurology (clinical), Developmental Biology
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6
المؤلفون: Joanne R. Mathiasen, Teresa M. O'Kane, Beth Ann McKenna, Robert L. Hudkins, Donna Bozyczko-Coyne, Masami Kaneko, George W. Gessner, Beth Ann Thomas, Mark A. Ator, Thelma S. Angeles, Chikara Murakata, Michael S. Saporito
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:147-150
مصطلحات موضوعية: Clinical Biochemistry, Carbazoles, Pharmaceutical Science, Indolocarbazole, Biochemistry, Chemical synthesis, Cell Line, Mice, chemistry.chemical_compound, In vivo, Drug Discovery, Animals, Enzyme Inhibitors, Protein kinase A, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, MAP Kinase Kinase Kinases, In vitro, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Signal transduction
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7
المؤلفون: Kurt A. Josef, Donna Bozyczko-Coyne, Zi-Qiang Gu, Sankar Chatterjee, Ming Tao, Rabindranath Tripathy, Ron Bihovsky, Mark A. Ator, Beth Ann McKenna, Shobha E. Senadhi, John P. Mallamo, Teresa M. O'Kane, Satish Mallya, Robert Siman, Derek Dunn
المصدر: Journal of Medicinal Chemistry. 41:2663-2666
مصطلحات موضوعية: Aldehyde, Chemical synthesis, law.invention, law, Drug Discovery, Tumor Cells, Cultured, Humans, Amino Acids, Enzyme Inhibitors, Binding site, chemistry.chemical_classification, Sulfonamides, Binding Sites, biology, Calpain, Stereoisomerism, Dipeptides, Recombinant Proteins, In vitro, Kinetics, Enzyme, chemistry, Biochemistry, Enzyme inhibitor, Recombinant DNA, biology.protein, Molecular Medicine
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8
المؤلفون: Rabindranath, Tripathy, Robert J, McHugh, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Zeck, Huang, Joanne R, Mathiasen, Amy, DiCamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Jie, Qian, Thelma S, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Emir, Duzic, Hervé, Schaffhauser, Gerard C, Rossé
المصدر: Bioorganicmedicinal chemistry letters. 22(3)
مصطلحات موضوعية: Molecular Structure, Brain, Stereoisomerism, Rats, Inhibitory Concentration 50, Mice, Dogs, Receptors, Serotonin, Microsomes, Liver, Animals, Humans, Serotonin Antagonists, Sulfones, Heterocyclic Compounds, 3-Ring
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9
المؤلفون: Babu G, Sundar, Thomas R, Bailey, Derek D, Dunn, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Huang, Zeqi, Joanne R, Mathiasen, Amy, Dicamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Rebecca, Brown, Jie, Qian, Thelma, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Deborah, Galinis, Emir, Duzic, Herve, Schaffhauser, Gerard C, Rosse
المصدر: Bioorganicmedicinal chemistry letters. 22(1)
مصطلحات موضوعية: ERG1 Potassium Channel, Brain, Ether-A-Go-Go Potassium Channels, Rats, Inhibitory Concentration 50, Kinetics, Structure-Activity Relationship, Memory, Short-Term, Models, Chemical, Piperidines, Receptors, Serotonin, Schizophrenia, Animals, Humans, Serotonin Antagonists, Benzofurans
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10
المؤلفون: Beth Ann McKenna, Karla Kopec, Daniel Pauletti
المصدر: Current Protocols in Pharmacology
مصطلحات موضوعية: Pharmacology, Gene isoform, GABA Plasma Membrane Transport Proteins, genetic structures, Cell, GABA transporter activity, Transporter, Transfection, Biology, chemistry.chemical_compound, medicine.anatomical_structure, HEK293 Cells, nervous system, chemistry, Biochemistry, Homogeneous, Cell culture, COS Cells, Chlorocebus aethiops, medicine, Animals, Humans, Neurotransmitter, gamma-Aminobutyric Acid