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1
المؤلفون: Thomas J. Connors, Jie Qian, Zeck Huang, Joanne R. Mathiasen, Edward R. Bacon, Thelma S. Angeles, Mark J. Huffman, Emir Duzic, Joseph M. Salvino, Beth Ann McKenna, Hervé Schaffhauser, Robert J. McHugh, Lily D. Lu, George C. Morton, Beverly P. Holskin, Karla Kopec, Amy DiCamillo, Gerard C. Rosse, Chrysanthe Spais, Rabindranath Tripathy, Lisa D. Aimone
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1421-1426
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Biochemistry, Sulfone, chemistry.chemical_compound, In vivo, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Pharmacophore, Receptor, Molecular Biology, 5-HT receptor
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2
المؤلفون: Beverly P. Holskin, Karla Kopec, Joanne R. Mathiasen, Amy DiCamillo, Babu G. Sundar, Thomas J. Connors, Emir Duzic, Edward R. Bacon, Gerard C. Rosse, Chrysanthe Spais, Thomas R. Bailey, Beth Ann McKenna, Rebecca A. Brown, Jie Qian, Derek Dunn, Mark J. Huffman, Joseph M. Salvino, Huang Zeqi, Lisa D. Aimone, Hervé Schaffhauser, Deborah Galinis, Thelma S. Angeles, Lily D. Lu, George C. Morton
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:120-123
مصطلحات موضوعية: biology, Organic Chemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Biochemistry, Social recognition, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, 5-HT6 receptor, Molecular Medicine, Structure–activity relationship, Serotonin Antagonists, Penetrant (biochemical), Receptor, Molecular Biology, 5-HT receptor
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3
المؤلفون: Beverly P. Holskin, Sheryl L. Meyer, Emmanuel Burgeon, Bruce Jones, Thao Ung, Emir Duzic, Sandra Y. Flores, Mark A. Ator, Vincent J. Dupriez
المصدر: Analytical Biochemistry. 400:184-189
مصطلحات موضوعية: Biophysics, Aequorin, Photoprotein, Digitonin, CHO Cells, Transfection, Biochemistry, Receptors, G-Protein-Coupled, law.invention, Cricetulus, law, Cricetinae, Animals, Humans, Receptor, Molecular Biology, G protein-coupled receptor, Cryopreservation, biology, Oxotremorine, Receptor, Muscarinic M1, Cell Biology, Acetylcholine, Cell biology, Cell culture, biology.protein, Recombinant DNA, Calcium, Function (biology)
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4
المؤلفون: Donna Bozyczko-Coyne, Steven C. Almo, Jean Husten, Michael S. Saporito, Richard W. Scott, Alexander A. Fedorov, Mark A. Ator, Chung Ho Park, Diebold James L, Ming Tao, Thelma S. Angeles, Sheryl L. Meyer, John P. Mallamo, Lisa D. Aimone, Elena V. Fedorov, Kurt A. Josef, Beverly P. Holskin, Robert L. Hudkins, Joanne R. Mathiasen, John T. Durkin
المصدر: Journal of Medicinal Chemistry. 51:5680-5689
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Molecular model, Stereochemistry, Carbazoles, Administration, Oral, In Vitro Techniques, Crystallography, X-Ray, Mice, In vivo, Cell Line, Tumor, Drug Discovery, Animals, Humans, Transferase, Protein Kinase Inhibitors, chemistry.chemical_classification, Molecular Structure, MAP kinase kinase kinase, biology, Chemistry, MAP Kinase Kinase Kinases, Pyrrolidinones, Rats, Enzyme, Enzyme inhibitor, Mitogen-activated protein kinase, biology.protein, Molecular Medicine, Signal transduction
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المؤلفون: George Gessner, Beverly P. Holskin, Matthew S. Reed, Jan Pohl, John T. Durkin, Karla K. Kopec, Brian M. Steffy, Chrysanthe M. Spais, Sheryl L. Meyer, Thelma S. Angeles, Mark A. Ator
المصدر: Biochemistry. 43:16348-16355
مصطلحات موضوعية: Threonine, Molecular Sequence Data, CHO Cells, Protein Serine-Threonine Kinases, Mitogen-activated protein kinase kinase, Biochemistry, Mass Spectrometry, MAP2K7, Cricetinae, Animals, Humans, Amino Acid Sequence, Phosphorylation, Serine/threonine-specific protein kinase, biology, MAP kinase kinase kinase, Cyclin-dependent kinase 5, Autophosphorylation, Cyclin-dependent kinase 2, JNK Mitogen-Activated Protein Kinases, MAP Kinase Kinase Kinases, Molecular biology, Protein Structure, Tertiary, Kinetics, Mutation, biology.protein, Cyclin-dependent kinase 9
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المؤلفون: Donna Bozyczko-Coyne, Beth Ann Thomas, Michael S. Saporito, Zhi-Liang Wu, Ghanashyam D. Ghadge, Stephen P. Trusko, Maroney Anna, Joanne R. Mathiasen, Beth Ann McKenna, Beverly P. Holskin, Raymond P. Roos, Jeffrey C. Thomas, Thomas C. Connors
المصدر: Brain Research. 1003:86-97
مصطلحات موضوعية: 1-Methyl-4-phenylpyridinium, medicine.medical_specialty, Programmed cell death, Indoles, SH-SY5Y, MAP Kinase Signaling System, Carbazoles, CHO Cells, chemistry.chemical_compound, Cell Line, Tumor, Cricetinae, Internal medicine, medicine, Animals, Humans, Molecular Biology, Cell Death, Dose-Response Relationship, Drug, biology, Kinase, General Neuroscience, MPTP, Neurotoxicity, MAP Kinase Kinase Kinases, medicine.disease, Cell biology, Enzyme Activation, Endocrinology, chemistry, Apoptosis, Cell culture, Mitogen-activated protein kinase, biology.protein, Neurology (clinical), Developmental Biology
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7
المؤلفون: Ted L. Underiner, Sheryl L. Meyer, Beverly P. Holskin, Thelma S. Angeles, Jay P. Theroff, Jie Qian
المصدر: Assay and drug development technologies. 10(4)
مصطلحات موضوعية: Boron Compounds, DNA, Complementary, biology, Chemistry, Ligand binding assay, Lactams, Macrocyclic, Drug Evaluation, Preclinical, Gene Expression, Fluorescence Polarization, Geldanamycin, Cysteine Proteinase Inhibitors, Hsp90, chemistry.chemical_compound, Biochemistry, Heat shock protein, Drug Discovery, biology.protein, Benzoquinones, Molecular Medicine, Atpase activity, HSP90 Heat-Shock Proteins, BODIPY, Fluorescence anisotropy, Function (biology), Fluorescent Dyes
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::55bc3c1fcd0722ed37fdab3a82a4e043
https://pubmed.ncbi.nlm.nih.gov/22428803 -
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المؤلفون: Kristen A. Murray, Jennifer L. Mason, Beverly P. Holskin, Thelma S. Angeles, Jie Qian, Mark A. Ator, Sheryl L. Meyer
المصدر: Assay and drug development technologies. 10(2)
مصطلحات موضوعية: Fluorescence, Cell Line, Small Molecule Libraries, hemic and lymphatic diseases, High-Throughput Screening Assays, Drug Discovery, Fluorescence Resonance Energy Transfer, STAT5 Transcription Factor, Humans, Phosphorylation, Protein Kinase Inhibitors, STAT5, Myeloproliferative Disorders, biology, Kinase, Janus Kinase 2, Molecular biology, Small molecule, Förster resonance energy transfer, Mutation, STAT protein, biology.protein, Molecular Medicine, Signal transduction, Janus kinase, Software
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e57642afcf141f5ea1254a5573194633
https://pubmed.ncbi.nlm.nih.gov/22132729 -
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المؤلفون: Kevin J. Wells-Knecht, Sheryl L. Meyer, Kristen A. Murray, Jennifer L. Mason, Mark A. Ator, Beverly P. Holskin, Thelma S. Angeles
المصدر: Assay and drug development technologies. 9(3)
مصطلحات موضوعية: Reporter gene, Cell growth, Activator (genetics), Response element, Mutant, Wild type, Biology, Janus Kinase 2, Protein Engineering, Molecular biology, Cell Line, IRF1, hemic and lymphatic diseases, Drug Discovery, Fluorescence Resonance Energy Transfer, Molecular Medicine, Humans, Biological Assay, Janus kinase, Protein Kinase Inhibitors, Interferon Regulatory Factor-1
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ca4d546991c8fdd8735fb298f4e27796
https://pubmed.ncbi.nlm.nih.gov/21133674 -
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المؤلفون: Kristen A. Murray, Beverly P. Holskin, Jennifer L. Mason, Mark A. Ator, Thelma S. Angeles, Jie Qian, Sheryl L. Meyer
المصدر: The FASEB Journal. 23
مصطلحات موضوعية: Förster resonance energy transfer, Homogeneous, Kinase, Chemistry, Genetics, Biophysics, Molecular Biology, Biochemistry, JAK2 V617F, Biotechnology, Cell based